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7-{[(butan-2-yl)(pyridin-4-ylmethyl)amino]methyl}-4-methyl-2H-chromen-2-one
4-({1-[methyl(pyrazin-2-ylmethyl)amino]hex-5-en-2-yl}oxy)benzonitrile
5-cyclobutyl-N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-1,3,4-oxadiazol-2-amine
2-{4-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]morpholin-3-yl}acetic acid
N-[2-(1H-indol-3-yl)ethyl]-6-(2,3,6-trifluorobenzoyl)-6-azaspiro[2.5]octane-1-carboxamide
4-[1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-1-(2-phenylethyl)piperidine
3-(furan-2-yl)-1-[4-(hydroxymethyl)-4-(2-phenoxyethyl)piperidin-1-yl]-3-phenylpropan-1-one
2-[4-(1-benzothiophen-3-yl)-2-(morpholin-4-ylmethyl)phenoxy]-N-cyclohexyl-N-methylacetamide
6-(benzyloxy)-1-cyclohexyl-4-(1,3-thiazole-4-carbonyl)-1,4-diazepan-2-one
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
[2-({4-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperazin-1-yl}methyl)phenyl]methanol
1-ethyl-N-[(5-ethylpyridin-2-yl)methyl]-N-[2-(pyridin-2-yl)ethyl]piperidin-4-amine
[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl](methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
N-methyl-N-({4-oxo-3H,4H-thieno[3,2-d]pyrimidin-2-yl}methyl)-5-(1H-pyrazol-1-ylmethyl)furan-2-carboxamide
5-{[benzyl(methyl)amino]methyl}-N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-1,2-oxazole-3-carboxamide
2-methoxy-N-({1-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)benzamide
1-cyclopropanecarbonyl-N-[3-(1H-indol-2-yl)phenyl]piperidine-4-carboxamide
3-(4-methanesulfonyl-1,4-diazepane-1-carbonyl)-6-phenyl-1,2-dihydropyridin-2-one
2-({6-[2-(aminomethyl)-7-chloro-2,3-dihydro-1-benzofuran-5-yl]quinazolin-4-yl}amino)ethan-1-ol
1-cyclobutanecarbonyl-4-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-1,4-diazepane
{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}[(1-methyl-1H-imidazol-2-yl)methyl](propan-2-yl)amine
1-[7-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
3-[1-(carbamoylmethyl)-1H-imidazol-2-yl]-N-[(4-fluorophenyl)methyl]piperidine-1-carboxamide
N-(cyclohex-3-en-1-ylmethyl)-1-methyl-N-(pyridin-4-ylmethyl)piperidin-4-amine
ethyl 4-{1-[2-(dimethylamino)benzoyl]piperidin-3-yl}piperazine-1-carboxylate
3,5-dimethyl-7-(5-phenoxyfuran-2-carbonyl)-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazine
1-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]-2-(pyrrolidin-1-ylmethyl)piperidine
2-{[4-methyl-1-(pyridin-4-yl)-1H-1,3-benzodiazol-2-yl]methoxy}acetic acid
4-{5-[(4-cyclobutanecarbonyl-1,4-diazepan-1-yl)methyl]thiophen-2-yl}-2-methylbut-3-yn-2-ol
3-fluoro-2-methoxy-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]benzamide
3-[(3R,4S)-1-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
(3aS,6aS)-2-methyl-5-[(2-oxo-1,2,3,4-tetrahydroquinolin-6-yl)sulfonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-(4-oxo-1,4-dihydropyridin-1-yl)acetamide
5-{[(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinolin-2-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
1-(carbamoylmethyl)-N-[(dimethyl-1,3-thiazol-5-yl)methyl]piperidine-3-carboxamide
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}cyclopropanamine
N-[3-(1H-pyrazol-1-yl)propyl]-2-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzamide
3,5-dimethyl-4-{1-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}-1,2-oxazole
N,3,5-trimethyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1,2-oxazole-4-carboxamide
1-[1-(hydroxymethyl)-9-[3-(1H-pyrazol-1-yl)propyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-(methylsulfanyl)ethan-1-one
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
1-(carbamoylmethyl)-N-methyl-N-[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]piperidine-3-carboxamide
1-{7,7-dimethyl-5-[(propan-2-yl)amino]-5,6,7,8-tetrahydroquinazolin-2-yl}piperidin-4-ol
4-butyl-11-(ethylamino)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
methyl 7-oxo-3-[(1R,2R)-2-phenylcyclopropanecarbonyl]-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-1-(2-propyl-1,3-thiazole-4-carbonyl)piperidine
N-(adamantan-1-yl)-8-methyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
4-(4-methanesulfonylphenyl)-5,6-dimethyl-2-(pyrrolidin-1-yl)pyrimidine
3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(2-methylpropyl)piperidin-4-yl]oxy}benzamide
N5-cyclopropyl-N6-[1-(3-methylpyridin-2-yl)propan-2-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine