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2-[3-(4-tert-butylphenoxymethyl)-5-[(2S,4R)-4-hydroxypyrrolidin-2-yl]-1H-1,2,4-triazol-1-yl]acetic acid
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(2-methylpropyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(1-hydroxybutan-2-yl)-5,6-dimethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
4-ethyl-6-{4-[1-(propan-2-yl)piperidine-3-carbonyl]piperazin-1-yl}pyrimidine
(3S,9aR)-3-(2-methylpropyl)-8-(quinolin-5-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-{[4-(2-phenylpropyl)-1H-1,2,3-triazol-1-yl]methyl}pyridine
(3S,4S)-1-[(2,6-difluorophenyl)methyl]-4-(4-fluorophenyl)piperidin-3-ol
3-[5-(aminomethyl)pyridin-2-yl]-5-[2-(piperidin-2-yl)ethyl]phenol
(3R,9aR)-3-[(benzylsulfanyl)methyl]-8-(2,3-difluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-{1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}-1H-pyrazole-4-carboxamide
N-[(3-chlorophenyl)methyl]-3-{1-[3-(pyrazin-2-yl)propanoyl]piperidin-4-yl}propanamide
2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)-N-[3-(pyridin-3-yl)propyl]acetamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-7-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide
1-{2-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
4-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridin-2-amine
N-[(3-methylphenyl)methyl]-N-(oxolan-2-ylmethyl)-3-(4H-1,2,4-triazol-4-yl)benzamide
3-[1-(6-aminopyrimidin-4-yl)piperidin-3-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(1-hydroxybutan-2-yl)-N-(pyridin-2-ylmethyl)quinoline-8-carboxamide
7-ethyl-2-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
1-{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-[(4-fluorophenyl)sulfanyl]piperidine
3-chloro-5-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
5-(3-chloropyridine-4-carbonyl)-1-(cyclopropylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-{[4-(pyrrolidine-1-sulfonyl)-1,4-diazepan-1-yl]methyl}benzoic acid
5,5-dimethyl-1-{2-oxo-2-[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]ethyl}imidazolidine-2,4-dione
N-[(5-amino-1,3,4-thiadiazol-2-yl)(phenyl)methyl]-4H-thieno[3,2-b]pyrrole-5-carboxamide
N-[(2,4-difluorophenyl)methyl]-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
ethyl[2-(1H-pyrazol-1-yl)ethyl]{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
5-[(1-methyl-1H-imidazol-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
N-[(1-methyl-2,3-dihydro-1H-indol-5-yl)methyl]-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-2-(methylsulfanyl)acetamide
2-(4-{[2-(1H-imidazol-1-yl)-1-phenylethyl]amino}piperidin-1-yl)pyridine-4-carbonitrile
N-(1-benzylpiperidin-4-yl)-1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
2,7,8-trimethyl-4-(thiomorpholine-4-carbonyl)quinoline
5-methoxy-2-{[2-(3-methoxyphenyl)piperidin-1-yl]methyl}-4H-pyran-4-one
N-{2-[2-(4-chlorophenyl)morpholin-4-yl]-2-oxoethyl}-2-methylpropanamide
ethyl 4-{[4-(pyridin-4-yl)pyrimidin-2-yl]amino}piperidine-1-carboxylate
methyl 2-[6-(1H-pyrazol-1-yl)pyrimidin-4-yl]benzoate
2,5-dioxo-6-{2-[2-(trifluoromethyl)phenyl]ethyl}-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
methyl 3-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}benzoate
N-[1-({methyl[(4-phenoxyphenyl)methyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-4-oxo-4-phenylbutanamide
(1S,4R)-4,7,7-trimethyl-N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-3-oxo-2-oxabicyclo[2.2.1]heptane-1-carboxamide
3-({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-1-(pyrrolidin-1-yl)propan-1-one
(3S,9aR)-2-methyl-3-(2-methylpropyl)-8-[4-(trifluoromethoxy)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(2-ethyl-1H-1,3-benzodiazol-6-yl)-3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine-1-carboxamide
N-({1-[1-(4-fluorophenyl)piperidin-4-yl]piperidin-3-yl}methyl)thiophene-2-carboxamide
4-{[(3S,5R)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-5-(pyrrolidine-1-carbonyl)piperidin-3-yl]methyl}morpholine
N-ethyl-6-methyl-4-(4-methyl-1H-imidazol-2-yl)-N-(2-methylprop-2-en-1-yl)-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
(2-methoxyethyl)[(3-methyl-1H-pyrazol-5-yl)methyl][(2E)-3-phenylprop-2-en-1-yl]amine
N-({1-[3-(1H-pyrazol-1-yl)propyl]piperidin-3-yl}methyl)pyridine-3-carboxamide
4-({5-methanesulfonyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-(trifluoromethyl)morpholine