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3-methyl-5-[3-(piperazin-1-yl)phenyl]pyridin-2-amine
N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-N-methyl-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-methyl-N-[1-(pyridin-3-yl)pentyl]acetamide
4-hydroxy-1-methyl-N-[(4-sulfamoylphenyl)methyl]piperidine-4-carboxamide
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
N-(propan-2-yl)-1-{1-[1-(pyrrolidin-1-yl)cyclopentanecarbonyl]piperidin-4-yl}piperidine-4-carboxamide
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-3-phenyl-1H-pyrazole-4-carboxamide
2-(4-fluorophenyl)-2-hydroxy-1-[4-(2-methylphenoxy)piperidin-1-yl]ethan-1-one
N-[3-(1H-imidazol-1-yl)propyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
11-{[(3-methylphenyl)methyl]amino}-4-(pyridin-2-ylmethyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-[(2R)-1-hydroxypropan-2-yl]-5-{[methyl(2-phenylethyl)amino]methyl}-1,2-oxazole-3-carboxamide
N-{1-[3-(2-methylphenyl)-3-phenylpropanoyl]piperidin-4-yl}methanesulfonamide
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-2-(4-propanoylphenoxy)acetamide
N-methyl-2-{4-[(E)-2-phenylethenyl]phenoxy}acetamide
N-(4-{2-[2-(4-hydroxyphenyl)ethyl]piperidine-1-carbonyl}phenyl)acetamide
(4aR,7aS)-1-propanoyl-4-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(4-chloro-1H-pyrazol-1-yl)-1-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
4-acetyl-N-[4-(3-acetylphenyl)phenyl]-1,4-diazepane-1-carboxamide
N,N-dimethyl-2-[(1S,5R)-6-{[3-(trifluoromethyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-4-(1-phenyl-1H-pyrazol-4-yl)pyrimidin-2-amine
3-[2-(2-fluorophenyl)ethyl]-1-(1,4-oxazepan-6-ylmethyl)urea
3-(4-methyl-1H-pyrazol-5-yl)-1-(naphthalene-1-sulfonyl)piperidine
3-{1-[(3-ethoxy-2-hydroxyphenyl)methyl]piperidin-3-yl}-N-[(2-fluorophenyl)methyl]propanamide
1-[(4-fluorophenyl)methyl]-5-[methyl(2-methylpropyl)amino]azepan-2-one
N-(oxan-3-ylmethyl)-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl](methyl)[(5-methyl-1H-pyrazol-3-yl)methyl]amine
(3R,4R)-4-cyclobutyl-1-(2-ethoxybenzoyl)-3-methylpiperidin-4-ol
N3-(1-benzylpiperidin-4-yl)-N5-cycloheptyl-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N,2-dimethyl-1-benzofuran-5-carboxamide
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(pyridin-3-yl)propan-1-one
4-fluoro-3-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]benzene-1-sulfonamide
3-(6-methoxynaphthalene-2-carbonyl)-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]piperidine
N-(pyridin-4-ylmethyl)-4-(quinolin-4-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
2-{2-[(pyridin-4-ylmethyl)amino]pyrimidin-4-yl}pyridine-4-carboxylic acid
4,6-dimethyl-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}pyrimidin-2-amine
N-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-1-[2-(methylsulfanyl)ethyl]piperidin-4-amine
2-[(2,4-dimethoxyphenyl)methyl]-4-{4-[4-(2,4-dimethylphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
(3S,4R)-4-methyl-1-[(2,3,5,6-tetrafluoro-4-methoxyphenyl)methyl]piperidine-3,4-diol
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-2-cyclopropyl-4-hydroxypyrimidine-5-carboxamide
2-methyl-8-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-2,8-diazaspiro[5.5]undecane
methyl 1-methoxy-2-oxo-8-[3-(prop-2-en-1-yloxy)benzoyl]-1,8-diazaspiro[4.5]decane-4-carboxylate
[(2S)-1-{[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}pyrrolidin-2-yl]methanol
[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl][(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amine
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
1-{2-[4-hydroxy-4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-4-methylpyrimidin-5-yl}ethan-1-one
1-[cyclohexyl(methyl)amino]-3-[2-methoxy-4-({methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
4-amino-1-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}butan-1-one
2-({4-[(4-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenol
1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-4-(pyridin-3-yl)piperazine
2-methyl-6-(1-{[3-(pyridin-2-yl)phenyl]methyl}piperidin-4-yl)pyrimidin-4-ol