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N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-methoxypyridine-4-carboxamide
{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}(methyl){[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
(2S,3R)-2-({[2-(adamantan-1-yl)-1,3-thiazol-4-yl]methyl}amino)-3-hydroxybutanamide
ethyl 4-(2-{1-[2-(dimethylamino)ethyl]-3-(3-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl}acetyl)piperazine-1-carboxylate
N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1,9-dioxaspiro[5.5]undecan-4-amine
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-4-oxo-3,4-dihydroquinazoline-2-carboxamide
dimethyl(2-{2-[1-(5-phenyl-1,3,4-thiadiazol-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)amine
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-[(2-methoxyphenyl)methyl]piperazine
4,4,4-trifluoro-1-[3-(naphthalene-1-carbonyl)piperidin-1-yl]butan-1-one
N-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)-1H-pyrazole-4-carboxamide
5-chloro-9-(2-fluorophenyl)-15-methyl-12-(morpholine-4-carbonyl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaen-13-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
(3aS,6aS)-2-(2,6-dimethoxypyridine-3-carbonyl)-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
8-(4-carboxyquinolin-2-yl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-(4-methyl-1,2,5-oxadiazol-3-yl)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}acetamide
(1R,5R)-6-(naphthalen-2-ylmethyl)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-[2-(thiophen-2-yl)ethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-[(3R,4S)-1-(6-aminopyrimidin-4-yl)-4-propylpyrrolidin-3-yl]-2-(2-oxopyrrolidin-1-yl)acetamide
N-[4-(2-oxopyrrolidin-1-yl)phenyl]-3-phenylpiperazine-1-carboxamide
(2S)-2-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-4-(methylsulfanyl)butan-1-ol
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-5-ethylpyrimidin-2-amine
6-[(diethylamino)methyl]-N-(2,3-dihydro-1,4-benzodioxin-6-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-[1-(4-fluoro-2-methylbenzoyl)piperidin-3-yl]-2-phenylethan-1-one
2-(2,6-difluorophenyl)-N-(3,4-dimethyl-1H-pyrazol-5-yl)acetamide
N-(3-phenylpropyl)-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-[6-amino-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-N,N-bis(propan-2-yl)benzamide
(1R,5S,6R)-3-cyclopentyl-N-[(5-methylpyrazin-2-yl)methyl]-3-azabicyclo[3.1.0]hexane-6-carboxamide
3-[2-(3,4-difluorophenyl)ethyl]-1-(3-fluoro-2-methoxybenzoyl)piperidine
1-{2-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}piperidin-2-one
2-(diethylamino)-N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
3-(5-{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanoic acid
6-methyl-3-[4-(1H-pyrazol-5-yl)phenyl]pyridin-2-amine
N3-[(3,5-dimethoxyphenyl)methyl]-1-[(5-methylfuran-2-yl)methyl]-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-[2-methyl-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]-2-oxo-1-oxaspiro[4.4]nonane-4-carboxamide
{5-methyl-7-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
(2S,4S)-N-[2-(2-fluorophenyl)ethyl]-4-{[(3-hydroxy-4-methoxyphenyl)methyl]amino}-1-(2-methylpropyl)pyrrolidine-2-carboxamide
1-[(4-fluorophenyl)methyl]-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-[(1s,4s)-4-aminocyclohexyl]-N-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-1H-1,2,3-triazole-4-carboxamide
(3S,9aR)-3-(1H-indol-3-ylmethyl)-8-(3-methoxybenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1-(propan-2-yl)piperidine-4-carboxamide
4-benzyl-3-{2-oxo-2-[4-(pyridin-3-yloxy)piperidin-1-yl]ethyl}piperazin-2-one
1-tert-butyl-N-[(3R,4S)-4-cyclopropyl-1-methanesulfonylpyrrolidin-3-yl]-1H-pyrrole-3-carboxamide
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-(5-phenyl-1,2-oxazole-3-carbonyl)pyrrolidin-3-yl]acetamide
4-(2-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-2-oxoethyl)-5-methyl-2,3-dihydro-1H-pyrazol-3-one
[1-(2,3-dihydro-1H-inden-2-yl)-4-[(4-methoxyphenyl)methyl]piperidin-4-yl]methanol
N-[3-chloro-2-(propan-2-yloxy)phenyl]-4-(dimethylamino)azepane-1-carboxamide
1-[(2,4-difluoro-3-methoxyphenyl)methyl]-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
N-ethyl-N-methyl-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
1-[4-(2-aminopyrimidin-4-yl)piperidin-1-yl]-2-(thiophen-2-yl)ethan-1-one
1-{4-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]piperidin-1-yl}ethan-1-one