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1-{2-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
N-[(5-chlorothiophen-2-yl)methyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-[1'-(2-methoxypyridine-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
N-(6-methylpyridin-3-yl)-4-[(oxolan-3-yl)sulfamoyl]benzamide
2-(cyclopropanesulfonamidomethyl)-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
6-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
ethyl 3-{[4-(3-hydroxypiperidin-1-yl)pyrimidin-2-yl]amino}propanoate
9-(4-methoxyquinoline-2-carbonyl)-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
[2-(4-fluoro-2-methoxyphenyl)pyridin-4-yl]methanol
1,3-dimethyl-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-(2-phenyl-1H-imidazol-1-yl)-1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
2-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]benzonitrile
4-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[2-(2-oxoimidazolidin-1-yl)ethyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
3-(1-methyl-1H-imidazol-2-yl)-1-{[2-(trifluoromethyl)phenyl]methyl}piperidine
(2S,4S)-4-amino-N,N-diethyl-1-(2-phenylbenzoyl)pyrrolidine-2-carboxamide
7-(2,3-dihydro-1,4-benzodioxine-6-sulfonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[(2S,4R)-4-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]-1-{[4-(methylsulfanyl)phenyl]methyl}pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane
6-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carbonyl}-2-methyl-2,3-dihydropyridazin-3-one
3-cyclopropyl-5-(4-fluoro-2-methoxyphenyl)-1-methyl-1H,4H-pyrazolo[3,4-d]imidazole
5-({3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)-2-(methylsulfanyl)pyrimidine
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
N-cyclopropyl-3-(dimethyl-1H-1,2,4-triazol-1-yl)-N-[(2-methoxyphenyl)methyl]-2-methylpropanamide
2-(dimethylamino)-2-(2-fluorophenyl)-N-methyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]acetamide
1-[4-(1H-indol-7-ylmethyl)-1,4-diazepan-1-yl]-2-methoxyethan-1-one
2-(4-fluoro-3-methylphenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]ethan-1-one
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-(2-methylphenyl)-3-phenylpropanamide
N,N-diethyl-1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperidine-4-carboxamide
N-[2-(2-chlorophenyl)-2-hydroxyethyl]-N'-(4-methylphenyl)propanediamide
N-{[1-(4-fluorophenyl)cyclopentyl]methyl}-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
4-benzyl-3-{2-oxo-2-[4-(pyridin-2-yl)piperazin-1-yl]ethyl}piperazin-2-one
(3S,4R)-1-(1H-1,3-benzodiazol-2-ylmethyl)-N,N-dimethyl-4-propylpyrrolidin-3-amine
3-{1-[(2-aminopyrimidin-5-yl)methyl]piperidin-4-yl}-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
5-methyl-N-propyl-2-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzamide
2-{[1-ethyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1-methyl-1H-1,3-benzodiazole
N-[cyclopropyl(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-3,5-dimethyl-1-benzofuran-2-carboxamide
3-(3-cyclopropyl-1H-pyrazol-5-yl)-4-(2-ethoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
[(4-ethyl-5-{1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
3-chloro-6-{4-[3-(methylsulfanyl)propyl]piperazin-1-yl}pyridine-2-carboxylic acid
1-methyl-N-[phenyl(pyridin-2-yl)methyl]-3-propyl-1H-pyrazole-5-carboxamide
3-[({[6-chloro-2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(methyl)amino)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{6-[(3-methoxyphenyl)methoxy]-4-(2-methylpropyl)-3-oxo-1,4-diazepane-1-carbonyl}-1,2,3,4-tetrahydroquinolin-2-one
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
ethyl 1-(2,1,3-benzoxadiazol-4-ylmethyl)-4-(2-phenoxyethyl)piperidine-4-carboxylate
8-cyclopropanecarbonyl-2-[(4-hydroxy-3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
ethyl 1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-pyrazole-4-carboxylate
N-{[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]methyl}-2-(pyrrolidin-3-yl)benzamide
2,4-dichloro-3-{[4-(2-methoxyethoxy)piperidin-1-yl]methyl}phenol
6-{1-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperidin-3-yl}pyrimidin-4-ol
1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-2-(1H-imidazol-1-yl)ethan-1-one