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1-{6-[2-(morpholin-4-ylmethyl)phenyl]pyridin-2-yl}ethan-1-ol
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-4-ethyl-2-methyl-1,3-thiazole-5-carboxamide
2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-methyl-N-(oxan-4-ylmethyl)acetamide
ethyl 1-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carbonyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
(4aR,8aS)-6-{[4-(benzyloxy)phenyl]methyl}-1-[(4-fluorophenyl)methyl]-decahydro-1,6-naphthyridin-2-one
2-(3,5-difluorophenyl)-1-[4-(1-methylpiperidin-4-yl)piperazin-1-yl]ethan-1-one
3-chloro-N-methyl-N-(pyrazin-2-ylmethyl)thiophene-2-carboxamide
2-[benzyl(methyl)amino]-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
3-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-3H,4H-pyrido[3,4-d]pyrimidin-4-one
methyl 3-cyclohexaneamido-5-{[(4-methyl-1,3-oxazol-5-yl)formamido]methyl}benzoate
1-(3-fluoro-4-methoxybenzoyl)-3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine
(3aR,6aS)-N-(1,3-diethyl-6-methyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-octahydropyrrolo[3,4-c]pyrrole-2-carboxamide
methyl 3-benzamido-5-{[(2-fluoro-5-methoxyphenyl)methyl]amino}-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(3S,4S)-1-[2-amino-6-(methylamino)pyrimidin-4-yl]-4-(naphthalen-2-yl)piperidin-3-ol
N-({1-[(4-methyl-1H-imidazol-5-yl)methyl]pyrrolidin-3-yl}methyl)isoquinoline-5-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methylimidazo[1,2-a]pyrimidine-2-carboxamide
{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[2-(1H-pyrazol-4-yl)ethyl]amine
1-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-hydroxy-2-[4-(trifluoromethyl)phenyl]ethan-1-one
1-(1-ethyl-1H-pyrazole-4-carbonyl)-4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine
N4-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-N2,N2,N4-trimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
1-[cyclohexyl(methyl)amino]-3-{2-methoxy-4-[(4-methoxypiperidin-1-yl)methyl]phenoxy}propan-2-ol
ethyl 1-benzyl-5-(oxan-4-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-(4-{[(4-hydroxyphenyl)methyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
2-[2-(azocan-1-yl)acetyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
(3aR,6aR)-2-methanesulfonyl-5-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]pyrazin-2-ol
{2-[2-(2,3-dimethoxy-5-methylphenyl)phenoxy]ethyl}dimethylamine
2-[2-({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]-3,4-dihydroquinazolin-4-one
1-[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]-2-(4,6,7-trimethyl-1-benzofuran-3-yl)ethan-1-one
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
2-amino-N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)pyridine-4-carboxamide
N-({7-[(3,5-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-5-(methoxymethyl)furan-2-carboxamide
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-3-phenyl-1H-pyrazole-5-carboxamide
N-(2-methylpropyl)-1-[(1s,4s)-4-{[(3,4,5-trimethoxyphenyl)methyl]amino}cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-(2-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenyl)ethan-1-one
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N-methyl-2-(3-methyl-2-oxopyrrolidin-1-yl)acetamide
N-[(2E)-3-phenylprop-2-en-1-yl]-N-propyl-4-(pyrrolidin-1-ylmethyl)benzamide
N-(1-{1-[(2R)-2-aminopropanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-phenylmethanesulfonamide
6-methyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-oxo-4-(pyridin-3-yl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
(1R,9aR)-1-(2-chloro-4-fluorophenoxymethyl)-octahydro-1H-quinolizine
ethyl 2-{1-[2-(3-methoxyphenyl)acetyl]piperidin-2-yl}acetate
2-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-6-methylpyridine-3-carbonitrile
2-(cyclopropylmethyl)-9-(1-methyl-1H-pyrazole-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N,N-dimethyl-2-{[(7-methyl-1-benzofuran-2-yl)formamido]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
N-{[2-(dimethylamino)-7-fluoroquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-3,4-dimethoxybenzamide
6-(2,5-dimethylfuran-3-yl)-N-(1-hydroxypropan-2-yl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-1-[(4-methoxyphenyl)methyl]piperazin-2-one
methyl 2-[4-({[1-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]carbamoyl}amino)phenoxy]acetate
1-(4-methylphenyl)-4-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}piperazin-2-one
2-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-3-fluoro-6-methylimidazo[1,2-a]pyridine