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N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5-hydroxy-N-methylpyrazine-2-carboxamide
1-(2-{[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)carbamoyl]amino}ethyl)piperidine-3-carboxamide
4-{[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl}morpholine
4-{5-[4-(thiophen-3-ylmethyl)piperazine-1-carbonyl]-1H-pyrazol-3-yl}phenol
3-(4-hydroxyphenyl)-N-[3-(1H-1,2,4-triazol-1-yl)propyl]benzamide
1-[6-(4-{4-[hydroxy(phenyl)methyl]-1H-1,2,3-triazol-1-yl}piperidin-1-yl)pyridin-3-yl]ethan-1-one
(3R,4S)-1-[6-(methoxymethyl)pyrimidin-4-yl]-N,N-dimethyl-4-propylpyrrolidin-3-amine
1-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]cyclopropane-1-carboxamide
4-{[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]methyl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
2-(dimethylamino)-N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-(3-methylphenyl)acetamide
N4-{[4-(pyrrolidine-1-carbonyl)phenyl]methyl}-5,6,7,8-tetrahydroquinazoline-2,4-diamine
N-cyclopentyl-4-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-3-(piperidin-3-yl)benzamide
10-[4-(4-methylphenyl)piperazine-1-carbonyl]-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraen-9-one
1-{4-[4-(benzyloxy)piperidin-1-yl]-4-oxobutyl}piperidin-2-one
4-(2,6-dimethylpyridin-3-yl)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}pyrimidin-2-amine
2-ethyl-2-hydroxy-1-{4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazin-1-yl}butan-1-one
N-(2-{1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidin-3-yl}ethyl)-1,3-thiazole-5-carboxamide
4-(2-methyl-1,3-thiazole-4-carbonyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(5-{2-[2-(oxolan-3-yl)-1H-imidazol-1-yl]ethyl}-1H-1,2,4-triazol-3-yl)pyridine
9-(3-ethyl-1H-pyrazole-5-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-1,4-dioxane-2-carboxamide
(3S,4S)-1-(3-hydroxypyridine-2-carbonyl)-4-propylpyrrolidine-3-carboxylic acid
1-(2-{1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperidin-2-yl}ethyl)pyrrolidin-2-one
1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}-3-(2-methyl-1H-1,3-benzodiazol-1-yl)propan-1-one
(5S)-5-[({[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}(pyridin-2-ylmethyl)amino)methyl]pyrrolidin-2-one
3-(2-phenylethyl)-N-(1,3-thiazol-2-ylmethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
3-[(3R,4S)-4-(dimethylamino)-1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-3-yl]propan-1-ol
N-benzyl-3-{2-[(4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}propanamide
4-[1-(5-chloronaphthalene-1-carbonyl)piperidin-4-yl]thiomorpholine
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(1H-pyrazol-1-yl)propanamide
N-[(2R,3R)-2-ethoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-4-(1H-1,2,4-triazol-1-yl)butanamide
4-(1-benzofuran-2-yl)pyridin-2-amine
4,6-dimethyl-1-{2-[3-(4-methylphenoxymethyl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one
2-[(4-acetyl-6-hydroxy-1,4-diazepan-1-yl)methyl]-8-chloro-1,4-dihydroquinolin-4-one
N-{[4-(cycloheptyloxy)-3-methoxyphenyl]methyl}-3,5-dimethyl-N-(pyridin-2-ylmethyl)-1,2-oxazole-4-sulfonamide
1-{1'-[(3-methyl-1H-indol-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
7-methoxy-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-1,2,3,4-tetrahydronaphthalen-2-amine
1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
methyl 2-{[3-(morpholin-4-yl)piperidin-1-yl]sulfonyl}benzoate
N-[(7S,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,3-dihydro-1-benzofuran-7-carboxamide
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-6-methylpyridine-3-carboxamide
1-[(2-chlorophenyl)methyl]-4-(1-propyl-1H-imidazol-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-(1-benzyl-1H-pyrazole-4-carbonyl)-3-[4-(trifluoromethyl)benzoyl]piperidine
1-[(3aS,6aS)-5-(pyridazine-3-carbonyl)-octahydropyrrolo[2,3-c]pyrrol-1-yl]-3-(methylsulfanyl)propan-1-one
N-({5-[3-(trifluoromethoxy)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)cyclopropanecarboxamide
2-chloro-N-propyl-5-({[(3R)-pyrrolidin-3-yl]carbamoyl}amino)benzamide
N-methyl-2-[4-(3-methylphenyl)piperazin-1-yl]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
2-[(4-methoxyphenyl)methyl]-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-1,3-benzoxazole-6-carboxamide
1-[(2-fluorophenyl)methyl]-N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-6-oxopiperidine-3-carboxamide