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3-[1-(5-methoxyfuran-2-carbonyl)piperidin-3-yl]-N-[(3-methoxyphenyl)methyl]propanamide
3-{2-[4-(1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindol-1-one
(2R)-2-amino-3-(1H-indol-3-yl)-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}propanamide
(2S,4R)-4-amino-1-[2-(2-cyclopropyl-1H-1,3-benzodiazol-1-yl)acetyl]-N-methylpyrrolidine-2-carboxamide
7-methyl-3-({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)-3,7,11-triazaspiro[5.6]dodecan-12-one
N-{[1-(1H-1,3-benzodiazol-2-ylmethyl)pyrrolidin-3-yl]methyl}cyclohexanecarboxamide
(2R,3R,6R)-5-[(2-methyl-1,3-oxazol-4-yl)methyl]-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
4-ethyl-1-{[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl}-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-methyl-2-[3-oxo-1-(2,6,8-trimethylquinoline-4-carbonyl)piperazin-2-yl]acetamide
4-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-5-(propan-2-yl)pyrimidine
(3S,4S)-1-[6-(3-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-4-(propan-2-yloxy)pyrrolidin-3-ol
N-[(2R,3R)-1'-(4-methylbenzoyl)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
[(3R,4R)-1-(2-ethoxypyridine-3-carbonyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
3-methyl-1-(2-methylphenyl)-3-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)urea
(1R,3s,6r,8S)-4-[1-(pyridin-3-ylmethyl)piperidine-4-carbonyl]-4-azatricyclo[4.3.1.13,8]undecane
2-[2-(dimethylamino)ethyl]-8-[3-(pyridin-2-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
6-{1-[2,2-dimethyl-1-(thiophen-2-yl)cyclopropanecarbonyl]piperidin-3-yl}-3,4-dihydropyrimidin-4-one
4-{2-chloro-4-[3-(methoxymethyl)pyrrolidine-1-carbonyl]phenoxy}-1-(2,2-dimethylpropyl)piperidine
N-(1-hydroxyhexan-2-yl)-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
3-(2-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl)phenol
1-[2-(azepan-1-ylmethyl)-6-methoxyphenoxy]-3-(morpholin-4-yl)propan-2-ol
3-(3-hydroxy-3-methylbutyl)-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}benzamide
2-(2-methoxyphenoxy)-N-[(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-3-yl)methyl]acetamide
4-methoxy-N-[2-(7-{[4-(pyrrolidin-1-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]benzamide
2-[3-(2-chlorophenyl)-1-(2-methoxyethyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(oxan-2-ylmethyl)acetamide
5-(3-fluoro-2-methoxyphenyl)-3-methyl-1H-1,2,4-triazole
2-{4-[2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)acetyl]piperazin-1-yl}pyridine-3-carbonitrile
2-(propan-2-yl)-N-(pyridin-2-ylmethyl)-1,3-benzoxazole-5-carboxamide
methyl({1-[1-(quinoline-6-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)amine
5-({4-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carbonyl]-1,3-oxazol-2-yl}methoxy)isoquinoline
4-(benzyloxy)-1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidine
2-(1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1,4-diazepan-6-yl)acetic acid
4-{4-[(2-fluorophenyl)methyl]piperidine-1-carbonyl}-1λ6-thiane-1,1-dione
5-(hydroxymethyl)-2-methyl-4-{[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]methyl}pyridin-3-ol
1-(4-fluorobenzoyl)-4-(2-methylpropyl)-1,4-diazepan-5-one
8-(2-ethoxyacetyl)-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
methyl 4-{1-methyl-2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-ylmethyl}-1H-pyrazole-3-carboxylate
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-2-(3-methylphenyl)acetamide
N-[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
({3-[(1R,5S)-3,8-diazabicyclo[3.2.1]octane-3-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}methyl)diethylamine
({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]amine
(4aS,8aR)-6-(1-benzothiophene-5-carbonyl)-1-propyl-decahydro-1,6-naphthyridin-2-one
4-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-2-[2-(2-methoxyethyl)-2H-1,2,3,4-tetrazol-5-yl]morpholine
(1R,5S)-6-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-6-azabicyclo[3.2.1]octane
6-(oxolan-2-ylmethyl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
2-({4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]phenyl}formamido)-N-methylbutanamide
5-ethoxy-N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]furan-2-carboxamide
3-[(3,6-dimethylpyrazin-2-yl)methyl]-1λ6-thiane-1,1-dione
2-(3-chlorophenoxy)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]propanamide
4-{[4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}pyridine