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1-(2-methyl-5-propylpyrimidin-4-yl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
2-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}butanamide
8-{2-[2-(pyridin-2-yl)pyrimidin-5-yl]-1H-imidazol-1-yl}quinoline
2-[(3,5-difluorophenyl)methyl]-3-oxo-N-propyl-2,8-diazaspiro[4.5]decane-8-carboxamide
3-[4-(dimethylamino)phenyl]-N-methyl-N-{[1-(propan-2-yl)piperidin-3-yl]methyl}propanamide
2-[2-(dimethylamino)ethyl]-8-(5-ethyl-2,6-dimethylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
N-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3-{2-[(4-methylphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
2-(1H-indol-3-yl)-N-[(2-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
(1R,5S)-3-(furan-3-carbonyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-(5-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
3-(4-chlorophenyl)-1-(6-hydroxy-1,4-diazepan-1-yl)propan-1-one
9-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-1-oxa-9-azaspiro[5.5]undecan-5-ol
5-(4-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperazin-1-yl)-2-methyl-2,3-dihydropyridazin-3-one
N-[(1-ethylpiperidin-3-yl)methyl]-3-(trimethyl-1H-pyrazol-1-yl)propanamide
4-(4-{1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(methoxymethyl)-1H-pyrazole-4-carbonyl}piperazin-1-yl)phenol
3-[2-(2,6-difluorophenyl)ethyl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine
6-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-2-methyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-1-(propan-2-yl)piperidine-4-carboxamide
4-[2-(2,3-difluorophenyl)pyridine-4-carbonyl]morpholine
7-(2,3-dimethoxyphenyl)-9-methoxy-4-{[2-(trifluoromethyl)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-({[(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)amino}methyl)pyrrolidin-3-ol
6-(methoxymethyl)-N-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)pyrimidin-4-amine
N-(3-hydroxypropyl)-1-(1-{[4-(2-methylphenyl)phenyl]methyl}piperidin-3-yl)-1H-1,2,3-triazole-4-carboxamide
6-[4-(furan-2-yl)benzoyl]-N-[2-(3-methoxyphenyl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
3-[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]-6-propyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-{4-[(8-methoxyquinolin-2-yl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
6,7-dimethoxy-2-{[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}quinazolin-4-amine
3-[4-(1-methoxyethyl)phenyl]-1H-1,2,4-triazole-5-carboxamide
2-cyclopentyl-9-(6-methylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
6-methyl-2-(morpholin-4-ylmethyl)quinolin-4-ol
(3R,4S)-1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)-4-propylpyrrolidin-3-amine
N-(furan-2-ylmethyl)-1-methyl-2-oxo-N-(pyridin-2-ylmethyl)-1,2-dihydroquinoline-4-carboxamide
2-methoxy-N-[(1-methyl-1H-imidazol-2-yl)methyl]-5-{[1,3]oxazolo[4,5-b]pyridin-2-yl}aniline
N-(1,4-oxazepan-6-ylmethyl)-1-phenyl-1H-1,2,3,4-tetrazol-5-amine
(3R,4R)-1-[1-(benzenesulfonyl)cyclopropanecarbonyl]-4-(hydroxymethyl)piperidin-3-ol
4-{3-[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]propyl}morpholine
4-[(benzyloxy)methyl]-1-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1H-1,2,3-triazole
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-4-(1H-1,2,4-triazol-1-yl)butanamide
5-amino-3-(6-methoxy-2H-1,3-benzodioxol-5-yl)-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-triene-4-carbonitrile
3-[2-(2,4-difluorophenyl)ethyl]-1-(1H-imidazol-2-ylmethyl)piperidine
4-(4-{1-[(1R,2S)-2-phenylcyclopropyl]-1H-imidazol-2-yl}-1H-1,2,3-triazol-1-yl)piperidine
3-[2-(dimethylamino)ethyl]-1-ethyl-8-[(1-methyl-1H-indol-3-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[2-(trifluoromethoxy)phenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
(furan-3-ylmethyl)({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)amine
2-{[2-(1,3-benzothiazol-2-yl)ethyl]amino}-N-(4-methylphenyl)propanamide
N-(2-ethylphenyl)-4-oxo-4-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]butanamide
N-ethyl-N-(2-methylphenyl)-3-(1,2,3,6-tetrahydropyridin-1-yl)propanamide
N-tert-butyl-4-(1-methyl-1H-imidazol-5-yl)benzene-1-sulfonamide
2-phenyl-5-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}pyrimidine
4-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane