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dimethyl[2-(1-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}piperidin-2-yl)ethyl]amine
{[6-chloro-2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}[3-(methylsulfanyl)propyl]amine
1-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
N-{4-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]phenyl}acetamide
N-[1-(cyclohexylmethyl)piperidin-3-yl]-2-[methyl(pyridin-4-ylmethyl)amino]acetamide
N3-{[5-(2-chlorophenyl)furan-2-yl]methyl}piperidine-1,3-dicarboxamide
2-{3-[3-(trifluoromethyl)benzoyl]piperidine-1-carbonyl}pyridin-3-ol
5-(1H-pyrazol-1-ylmethyl)-N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}furan-2-carboxamide
2-(4-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}morpholin-2-yl)ethan-1-ol
N3-tert-butyl-N5-(2,2-diphenylethyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
1-cyclohexyl-N-[1-(1-methyl-1H-imidazol-2-yl)butyl]piperidine-4-carboxamide
5-methoxy-1-methyl-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-1H-indole-2-carboxamide
1-ethyl-N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1H-pyrazole-4-carboxamide
1-[5-(3-chloro-2-fluorobenzoyl)-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-4-phenylpiperazine
(1r,4r)-4-({[1-(4-fluorophenyl)-2,2-dimethylcyclopropyl]formamido}methyl)cyclohexane-1-carboxylic acid
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-phenylacetamide
2-(4-methyl-1H-imidazol-5-yl)-1-[3-(pyrrolidin-1-ylmethyl)phenyl]-1H-imidazole
N-{[7-chloro-2-(4-methoxyphenyl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)propanamide
(3aS,6aS)-2-(dimethylcarbamoyl)-5-(naphthalene-2-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-benzyl-4-[5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carbonyl]piperazin-2-one
N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-4-(pyridin-2-yl)pyrimidin-2-amine
[(3R,4R)-1-(5-chlorofuran-2-carbonyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
2-(5-acetylthiophen-3-yl)-N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)acetamide
2-{4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenoxy}-1-(piperidin-1-yl)ethan-1-one
N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]-1-(2-phenylethyl)piperidin-4-amine
(2E)-N-({3-methyl-7-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-(thiophen-2-yl)prop-2-enamide
4-{2-oxo-4-[3-(trifluoromethyl)benzoyl]piperazin-1-yl}benzonitrile
3-[1-(3,4-dimethylbenzenesulfonyl)piperidin-4-yl]-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
5-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
2-[1-(dimethyl-1,3-thiazol-2-yl)-1H-pyrazol-4-yl]-7-fluoro-N,N-dimethylquinoline-4-carboxamide
3-(4-fluorophenyl)-N-(2-{4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)benzamide
4-(1H-pyrazol-3-yl)-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
N,N-diethyl-1-{1-[4-(1H-imidazol-1-yl)phenyl]piperidin-4-yl}pyrrolidin-3-amine
1-{2-[4-(2-methoxybenzoyl)piperazine-1-carbonyl]pyrrolidin-1-yl}propan-1-one
(3aR,6aS)-5-[(4-ethoxyphenyl)methyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-chloro-N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
ethyl 2-({2-[(4-methoxyphenyl)methyl]morpholine-4-carbonyl}amino)acetate
1-{2-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]pyrimidin-4-yl}piperidin-3-ol
2-[3-(2-hydroxyethyl)-4-[(5-methylfuran-2-yl)methyl]piperazin-1-yl]-6-methylpyridine-3-carboxylic acid
5-chloro-6-(3,5-difluorophenyl)-2-methylpyrimidin-4-ol
8-(1-benzofuran-2-ylmethyl)-1-methyl-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(2H-1,2,3,4-tetrazol-2-yl)ethan-1-one
4,6-dimethyl-N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
1-(4-fluorophenyl)-4-(1-propylpiperidin-4-yl)piperazine
(2S,4R)-4-amino-N-ethyl-1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]pyrrolidine-2-carboxamide
N4-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-5-methylpyrimidine-2,4-diamine
ethyl 2-({[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)acetate
1,6-dimethyl-3-[2-(pyridin-2-yl)piperidine-1-carbonyl]-1,4-dihydroquinolin-4-one
1-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-3-(1-ethyl-2-methyl-1H-indol-5-yl)urea
methyl 6-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-2-[methyl(2-methylpropyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate