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1-[2-(2,3-dihydro-1H-isoindol-2-ylmethyl)-4-methoxyphenoxy]-3-(dimethylamino)propan-2-ol
2-[(3-hydroxyphenyl)methyl]-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
(2S,4R)-4-amino-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
(3S)-3-{[1-methyl-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}azepan-2-one
4-(4-{4-[(2,2-dimethylmorpholin-4-yl)methyl]-1H-1,2,3-triazol-1-yl}piperidin-1-yl)pyrimidin-2-amine
2-(dimethylamino)-2-(4-methylphenyl)-N-(1-phenylpiperidin-4-yl)acetamide
1-[4-(2-ethoxyphenyl)piperazin-1-yl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
methyl 2-[8-benzyl-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
2-chloro-N-{[1-(1H-imidazol-4-ylmethyl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}pyridine-4-carboxamide
9-oxo-N-(4H-1,2,4-triazol-4-yl)-9,10-dihydroacridine-4-carboxamide
N-(3-methyl-1,2,4-thiadiazol-5-yl)-3-(2-methylphenyl)piperidine-1-carboxamide
2-amino-6-{4-[3-(5-methylfuran-2-yl)butyl]piperazin-1-yl}-3,4-dihydropyrimidin-4-one
4-[2-(2,5-dimethyl-1H-pyrrol-1-yl)-4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl]-1,4-oxazepan-6-ol
(3aR,6aR)-2-cyclopentyl-N-[(4-sulfamoylphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
5-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}-1H-1,3-benzodiazole
1-(2-benzyl-1,3-thiazole-4-carbonyl)-4-(1-methyl-1H-imidazol-2-yl)piperidine
1-(2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-amido)cyclopentane-1-carboxylic acid
3-(2-chlorophenyl)-3-(3-hydroxyphenyl)-1-(4-methoxypiperidin-1-yl)propan-1-one
3-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propanoic acid
N-(2,2-dimethyloxan-4-yl)-2-(4-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
2-[3-(2-fluorophenyl)pyrrolidin-1-yl]-4-(1-methyl-1H-pyrazol-4-yl)pyrimidine
1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-3-methoxypropan-1-one
N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
4-(1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carbonyl)morpholine
4-methyl-5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-2-phenylpyrimidine
N4-[1-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-2-methylpropyl]-5-ethylpyrimidine-2,4-diamine
5-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2-methyl-1H-1,3-benzodiazole
5-{[(1S,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-2,1,3-benzothiadiazole
3-[(3S,4R)-1-benzyl-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]-N-(2-methoxyethyl)propanamide
2-(2-methyl-1,3-thiazol-4-yl)-1-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]ethan-1-one
3-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-6-phenyl-1,2-dihydropyridin-2-one
N-ethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
{1-[1-(6-ethoxy-4-methylquinazolin-2-yl)piperidin-4-yl]piperidin-4-yl}(pyridin-3-yl)methanol
3-(4-chloro-1H-pyrazol-1-yl)-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]propanamide
(3S,5R)-N3-(6-methylpyridin-3-yl)-N5-(pyridin-2-ylmethyl)piperidine-3,5-dicarboxamide
4-[5-({4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}methyl)pyrimidin-2-yl]morpholine
2-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-6,7-dimethoxyquinazolin-4-amine
1-(4-{[1-(1H-1,3-benzodiazol-2-yl)ethyl]amino}-2-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
2-[(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]-3-methoxyphenol
4-[(2-butyl-1H-imidazol-4-yl)methyl]-1-[(2-fluorophenyl)methyl]piperazin-2-one
2-chloro-N-methyl-5-(1H-pyrazol-3-yl)benzamide
N-[(3S,4R)-1-[(4-acetamidophenyl)methyl]-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
N-[3-(4-fluorophenyl)phenyl]-1-(4-methyl-2-oxopentanoyl)piperidine-3-carboxamide
2-[1-(cyclohexylmethyl)-4-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperazin-2-yl]ethan-1-ol
(1S,3R)-3-amino-N-{[2-chloro-5-(trifluoromethyl)phenyl]methyl}cyclopentane-1-carboxamide
{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[1-(pyridin-2-yl)ethyl]amine
4-{[4-(3-hydroxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-pyrazole-3-carboxylic acid
1-(3-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-3-oxopropyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
3-(3-chloro-1,2-oxazol-5-yl)-1-[2-(pyrrolidine-1-carbonyl)piperazin-1-yl]propan-1-one
4-chloro-2-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenol