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N,5,6-trimethyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-2-(pyrrolidin-1-yl)pyrimidin-4-amine
(2,1,3-benzoxadiazol-4-ylmethyl)(methyl)[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]amine
1-[2-(2-methyl-1H-imidazol-1-yl)propanoyl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-2,3-dihydro-1H-indene-1-carboxamide
1-benzyl-4-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-3-methoxybenzamide
3-(3-chlorophenyl)-3-(2-hydroxyphenyl)-N-(pyridin-4-ylmethyl)propanamide
N-(1,3-benzothiazol-2-ylmethyl)-2-[(4-methoxyphenyl)methyl]-1,3-benzoxazole-6-carboxamide
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-2-(2-methoxyethyl)-N-methyl-1,3-benzoxazole-6-carboxamide
2-chloro-5-acetamido-N-[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]benzamide
N-ethyl-3-{[1-(4-hydroxyphenyl)propyl]sulfamoyl}-N-methylbenzamide
1-(2-chlorophenyl)-4-[1-oxo-1-(pyrrolidin-1-yl)propan-2-yl]piperazin-2-one
2-methoxy-N-[1-methyl-2-(pyridin-3-yl)-5-[2-(1,3-thiazol-2-yl)piperidine-1-carbonyl]-1H-1,3-benzodiazol-7-yl]acetamide
2-ethoxy-6-{1-[(3-fluorophenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenol
3-(2-phenylethyl)-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,2-oxazole-5-carboxamide
2-{4-[(2-aminopyridin-3-yl)methyl]morpholin-3-yl}acetic acid
4-(piperidin-1-yl)-1-[2-(1,3-thiazol-2-yl)piperidin-1-yl]butan-1-one
(3S,4R)-1-(5-hydroxypyrazine-2-carbonyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-5-{cyclopropyl[(trimethyl-1H-pyrazol-4-yl)methyl]amino}azepan-2-one
(2S,6S)-1-(1-cycloheptyl-1H-1,2,3-triazole-4-carbonyl)-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
6-(propan-2-yloxy)-N4-[2-(1H-1,2,3,4-tetrazol-5-yl)ethyl]pyrimidine-2,4-diamine
2-{[3-(2-hydroxyethyl)-4-(2-methylpropyl)piperazin-1-yl]methyl}quinolin-4-ol
1-[4-(furan-2-ylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]-3-(1,2-oxazinan-2-yl)propan-1-one
ethyl 4-benzyl-1-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxylate
(2E)-N-({4-[(4-fluorophenyl)methoxy]phenyl}methyl)-N-(pyridin-3-ylmethyl)-3-(thiophen-2-yl)prop-2-enamide
methyl 1-[2-(propan-2-yl)-1,3-benzoxazole-5-carbonyl]piperidine-2-carboxylate
1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(methoxymethyl)-N-[2-(pyridin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
N-{[5,8-dimethoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)propanamide
3-{3-[6-(morpholin-4-yl)pyrimidin-4-yl]piperidine-1-carbonyl}phenol
3-{1-[2-(methylamino)pyrimidine-5-carbonyl]piperidin-4-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[2-(4-acetylpiperazin-1-yl)-5,8-dimethoxyquinolin-3-yl]methyl}-4-methyl-N-(oxolan-2-ylmethyl)benzamide
6-methyl-2-[(2-propylpyrrolidin-1-yl)methyl]quinolin-4-ol
4-chloro-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
7,7-dimethyl-2-{2-[(6-methyl-2-propylpyrimidin-4-yl)amino]ethyl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
8-[6-(dimethylamino)pyrimidin-4-yl]-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[(1S,3S,3aR,6aS)-5-ethyl-3-(hydroxymethyl)-3-phenyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]-4-methylphenol
4-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phthalazin-1-ol
N-[(1-propyl-1H-imidazol-2-yl)methyl]-4-(pyridin-3-yl)pyrimidin-2-amine
N-(2-methoxyethyl)-N-[(3-methoxyphenyl)methyl]oxolane-3-carboxamide
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-2-propyl-1,3-thiazole-4-carboxamide
4-{6-[2-methyl-4-(pyrrolidin-1-ylmethyl)phenoxy]pyrazine-2-carbonyl}morpholine
8-fluoro-4-oxo-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-1,4-dihydroquinoline-2-carboxamide
N-{[(2R)-1-ethylpyrrolidin-2-yl]methyl}-5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
(2S,4S)-4-[(1-benzylpiperidin-4-yl)amino]-1-(2,2-diphenylethyl)-N-methylpyrrolidine-2-carboxamide
4-[3-(4-phenoxybenzoyl)piperidine-1-carbonyl]pyridin-1-ium-1-olate
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(1H-imidazol-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(3S,4R)-1-{5-methyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carbonyl}-4-phenylpyrrolidine-3-carboxylic acid
2-(3,4-dichlorophenyl)-4-(1-methylpiperidin-4-yl)morpholine
4-[(1-phenoxypropan-2-yl)amino]-N-phenylpiperidine-1-carboxamide
4-methyl-N-[4-(1,3-thiazol-4-yl)phenyl]-1,4-diazepane-1-carboxamide