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N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetamide
(2S)-N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-5-oxopyrrolidine-2-carboxamide
1-[(2-methyl-1,3-thiazol-5-yl)methyl]-3-[2-(methylsulfanyl)benzoyl]piperidine
4-[(4-fluorophenyl)methyl]-N,N-dimethyl-3-(propan-2-yl)-1,4-diazepane-1-sulfonamide
3-[(oxan-4-yl)sulfamoyl]-N-(piperidin-4-ylmethyl)benzamide
N-methyl-4-[4-(oxolan-2-ylmethyl)piperazine-1-carbonyl]pyridin-2-amine
N-{[3-(2-chlorophenyl)-1,2-oxazol-5-yl]methyl}-3-(1-methylpiperidin-3-yl)propanamide
(2S)-3-hydroxy-2-(methylamino)-1-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propan-1-one
3-acetyl-N-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-1H-pyrazole-5-carboxamide
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
methyl N-{[(2S,4S)-4-fluoro-1-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl]methyl}carbamate
methyl 3-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-7-oxo-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]-2-methyl-1,3-thiazole-4-carboxamide
3-{[1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)pyrrolidin-3-yl]methyl}benzoic acid
(3R,4S)-4-[4-(2-ethylpyrimidine-5-carbonyl)-1,4-diazepan-1-yl]oxolan-3-ol
ethyl 1-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
3-{2-[2-(furan-2-yl)-1H-imidazol-1-yl]ethyl}-1H-indole
N-(1-ethyl-5-oxopyrrolidin-3-yl)-2-(1H-1,2,4-triazol-3-yl)benzamide
N-[3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)propyl]-2-(ethylamino)pyrimidine-5-carboxamide
1-methyl-N-{2-[methyl(phenyl)amino]ethyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide
1-{[2-(4-chlorophenyl)-5,8-dimethoxyquinolin-3-yl]methyl}azetidin-3-ol
6-methoxy-3-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
2-{2-[1-(2-methyl-2-phenylpropanoyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
4-[5-(pyrrolidin-1-ylmethyl)pyridin-2-yl]benzonitrile
(3S,4S)-N-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-methoxypyrrolidin-3-amine
4-{1-[1-(5-ethyl-2-methylpyrimidin-4-yl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
(2S,4S)-N-ethyl-1-(propan-2-yl)-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
1-{2-[2-(1H-imidazol-1-yl)ethyl]piperidin-1-yl}-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
5-{3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}-2-methylphenol
(1R,3S)-3-(2-aminoethoxy)-7-[2-(pyrrolidin-1-yl)benzoyl]-7-azaspiro[3.5]nonan-1-ol
8-methoxy-N-(2-methylpropyl)-N-(pyridin-4-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-methyl-N-{[3-(2-methylpropyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}aniline
1-{6-oxa-9-azaspiro[4.5]decan-9-yl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethan-1-one
4-amino-2-[4-(4-benzyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]pyrimidine-5-carbonitrile
N-(3-methoxypropyl)-2,5-dimethyl-N-(1-methylpiperidin-4-yl)-1,3-thiazole-4-carboxamide
N-(adamantan-1-yl)-1-[(3-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
1-[(3R,4R)-3-hydroxy-4-(4-methylpiperazin-1-yl)piperidin-1-yl]-3-phenylprop-2-yn-1-one
2-amino-6-(1-ethyl-1H-indol-3-yl)-4-[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]pyridine-3-carbonitrile
1-(2,5-dimethylfuran-3-carbonyl)-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
(1S,4S)-5-(2,3-dihydro-1H-inden-2-yl)-2-(2-fluorophenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-(oxolan-2-ylmethyl)-N-({4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
6-({1-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]hex-5-en-2-yl}oxy)-N,N-dimethylpyridazin-3-amine
1-(carbamoylmethyl)-N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]piperidine-3-carboxamide
N-[2-(dimethylamino)ethyl]-3-(1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)propanamide
N-benzyl-N-[(1R,2R)-2-hydroxycyclohexyl]-1H-1,2,3-triazole-5-carboxamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[3-(oxolan-3-yl)propyl]-1H-pyrazole-3-carboxamide
4-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]-2-[3-(1H-pyrazol-1-yl)azetidin-1-yl]pyrimidine
2-{4-[(3-hydroxyazetidin-1-yl)methyl]phenoxy}-1-(morpholin-4-yl)ethan-1-one
(5S,9aS,9bS)-2-[(4-methoxyphenyl)methyl]-5-(thiophen-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one