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6,6-dimethyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-5-oxothiomorpholine-3-carboxamide
N-[2-(4-methoxyphenoxy)ethyl]-2-(1H-1,2,3,4-tetrazol-5-yl)aniline
3-cyclopropyl-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-1H-pyrazole-5-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyridazine-3-carboxamide
2-(4-{[4-(4-methoxybenzoyl)piperazin-1-yl]methyl}-3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-ol
2-[2-(oxolan-3-yl)ethyl]-2,3-dihydro-1,2-benzothiazol-3-one
6-[2-hydroxy-2-(2-methoxyphenyl)ethyl]-2-methoxy-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
{[2-chloro-5-ethoxy-4-(propan-2-yloxy)phenyl]methyl}[1-(1H-1,2,4-triazol-5-yl)ethyl]amine
N-[(3R,5S)-5-(ethylcarbamoyl)-1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]-4-methyl-1,2,3-thiadiazole-5-carboxamide
4-({5-[1-(cyclopentylmethyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)morpholine
3-[(3R,4S)-4-(morpholin-4-yl)-1-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}piperidin-3-yl]propan-1-ol
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}benzamide
9-(3-methanesulfonylpropanoyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{[(1R,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzoic acid
15-methyl-12-(3-methylpiperidine-1-carbonyl)-9-(pyridin-3-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaen-13-one
methyl 3-{[1-(cyclopropylmethyl)-5-(naphthalene-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]formamido}propanoate
4-(1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)pyridine
8-[4-(1H-imidazol-1-yl)butanoyl]-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
5-(1-benzoxepine-4-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
4-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]benzamide
6-(1-benzofuran-2-yl)-5-cyano-2-methylpyridine-3-carboxylic acid
N-methyl-N-(pyridin-2-ylmethyl)-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-methyl-5-{[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}furan-2-carboxamide
ethyl 4-(6-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}-6-azaspiro[2.5]octane-1-carbonyl)piperazine-1-carboxylate
3-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carbonyl}-6-methyl-1,2-dihydropyridin-2-one
1-ethyl-N-(furan-3-ylmethyl)-5-[(2-methoxyethyl)(methyl)amino]-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-(2-methoxyethyl)-2-methyl-3-({[2-(1-methyl-1H-pyrazol-5-yl)ethyl]carbamoyl}amino)benzamide
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-4-(1H-1,2,4-triazol-3-yl)benzamide
3-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidine-1-carbonyl}quinoline
2-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
3-methyl-1-{1-[6-(quinolin-3-yl)pyridine-3-carbonyl]piperidin-3-yl}butan-1-one
4-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-6-(propan-2-yloxy)pyrimidin-2-amine
[(4aS,8aR)-6-{[4-(1H-imidazol-1-yl)phenyl]methyl}-decahydro-1,6-naphthyridin-4a-yl]methanol
methyl 2-{[(2,4-dimethoxyphenyl)methyl]amino}pyridine-4-carboxylate
5-methoxy-1-methyl-2-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-1-carbonyl}-1H-indole
1-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}azepane
{2-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}urea
1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-3-(pyridin-3-yl)propan-1-one
methyl 5-{[4-(4-methoxyphenyl)-2-methyl-3-oxopiperazin-1-yl]methyl}furan-2-carboxylate
(3S,4R)-1-[2-(2,4-dioxoimidazolidin-1-yl)acetyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
1-[(3,5-dimethylphenyl)methyl]-4-(3-fluoropyridin-4-yl)piperazin-2-one
4-(methoxymethyl)-6-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyrimidine
N,N-dimethyl-2-[(1S,5R)-6-(3-phenoxypropanoyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
(2S,4S)-N-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-5-yl}-1-[(4-methoxy-3-methylphenyl)methyl]-4-(pyrimidin-2-ylsulfanyl)pyrrolidine-2-carboxamide
3-[1-(1-cyclopentanecarbonylpiperidin-4-yl)-1H-pyrazol-5-yl]-1-(2-methylphenyl)urea
2,3-dimethyl-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]quinoxaline-6-carboxamide
(1R,5R)-6-(cyclopropylmethyl)-3-{1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-8-(4-phenylbutan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-4-(pyrrolidin-1-yl)butan-1-one
2-(2-methoxyethyl)-9-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one