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N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}-2-(4-methyl-1H-pyrazol-1-yl)acetamide
(4aS,7aR)-1-(2-phenylacetyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N'-cyclopentyl-N-[1-(thiophen-2-yl)butyl]butanediamide
4-[4-methyl-2-(pyridin-3-yl)pyrimidine-5-carbonyl]-2-(trifluoromethyl)morpholine
4-(2-{1-[(5-fluoro-2-methylphenyl)methyl]piperidin-2-yl}ethyl)morpholine
3-(4-{3-[(2-chlorophenyl)methoxy]phenyl}-1H-pyrazol-1-yl)propanamide
1-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
5-benzamido-1-cyclopentyl-N-(furan-2-ylmethyl)-N-(prop-2-yn-1-yl)-1H-1,3-benzodiazole-7-carboxamide
N3-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-N1-(pyridin-3-yl)propane-1,3-diamine
methyl (2S)-2-(3-{5-oxo-2-[(4-phenylphenyl)methyl]pyrrolidin-2-yl}propanamido)-2-phenylacetate
3-(4-chlorophenyl)-1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}propan-1-one
6-(2,5-dimethylphenyl)-N-(1,2-oxazol-3-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-{4-[(6-ethoxyquinolin-2-yl)methyl]-1-(3-methylbut-2-en-1-yl)piperazin-2-yl}ethan-1-ol
4-[3-(4-methylphenyl)phenyl]-4H-1,2,4-triazole
N-{2-[4-(1-benzofuran-5-yl)-1H-1,2,3-triazol-1-yl]ethyl}-3-methylpyridin-4-amine
N-(1-benzothiophen-5-ylmethyl)-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
N,N,2-trimethyl-7-{4H-thieno[3,2-b]pyrrole-5-carbonyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
5-{[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-3-propylimidazolidine-2,4-dione
({3-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}methyl)diethylamine
1-[2-(3-methylphenyl)benzoyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
1-cyclopropyl-4-[4-(2-methoxyphenyl)piperidine-1-carbonyl]pyrrolidin-2-one
N-(1H-imidazol-2-ylmethyl)-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-methylpropan-2-amine
N-[(4-methoxyphenyl)methyl]-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{1-[1-(3,4-dichlorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
2-(2,6-dioxo-1,3-diazinan-1-yl)-N-[1-(4-methoxyphenyl)propyl]-N-methylacetamide
1-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}-3-(4-methoxy-2-methylphenyl)urea
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-[2-(pyrazin-2-yl)acetyl]piperidin-3-yl]propanoic acid
4-(azepane-1-carbonyl)-N-(1,2-oxazol-3-ylmethyl)benzene-1-sulfonamide
N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
(4aR,7aS)-1-ethyl-4-[2-(phenylsulfanyl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[1-(1H-imidazol-4-ylmethyl)pyrrolidin-3-yl]methyl}adamantane-1-carboxamide
5-methoxy-N,1-dimethyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1H-indole-2-carboxamide
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
4-[(2,4,5-trifluorophenyl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
8-fluoro-2-({[1-(furan-2-carbonyl)piperidin-3-yl]amino}methyl)quinolin-4-ol
5-(2-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(2,1,3-benzoxadiazol-4-ylmethyl)-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
N-[1-(3-fluoro-4-hydroxyphenyl)ethyl]-1-(2-hydroxyethyl)-1H-1,3-benzodiazole-5-carboxamide
3-[5-(pyridine-4-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl]pyridine
8-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-3-(2-methylpropyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{3-[3-(pyrazin-2-yl)phenyl]-1H-pyrazol-1-yl}butan-2-ol
3-{[1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)piperidin-4-yl]oxy}pyridine
[1-(1-benzofuran-2-ylmethyl)-3-[(3-methoxyphenyl)methyl]piperidin-3-yl]methanol
2-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidine-1-carbonyl]-3,5,7-trimethyl-1H-indole
N-methyl-2-({5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)ethane-1-sulfonamide
1-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine-3-carbonitrile
4-(1-{2-amino-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}-1-oxopropan-2-yl)-1,2-dihydrophthalazin-1-one
1-(1-{6-[(thiophen-2-ylmethyl)amino]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}piperidin-4-yl)piperidin-3-ol
3-(2-amino-1,3-thiazol-4-yl)-1-[3-(3-fluorophenoxymethyl)piperidin-1-yl]propan-1-one