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N-[(4-{[(2-fluorophenyl)methyl]amino}-8-methylquinazolin-2-yl)methyl]-3,5-dimethyl-1,2-oxazole-4-sulfonamide
N-(2-fluorophenyl)-2-(3-methoxypropyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
N,N,1-triethyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]-N-(2-fluorophenyl)piperidine-1-carboxamide
[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]({[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl})methylamine
N-(3-methoxypropyl)-5,6-dimethyl-N-{[6-(2-methylphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
5-(1-benzothiophen-2-ylmethyl)-8-ethoxy-2-(3,4,5-trimethoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]-1-(1,2-oxazole-3-carbonyl)piperidine
2,4-dichloro-3-({methyl[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]amino}methyl)phenol
1-[6-(methoxymethyl)pyrimidin-4-yl]spiro[azepane-4,2'-chromene]
1'-[(3,5-dimethoxyphenyl)methyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
3-[2-methyl-4-(4-methylphenyl)-5-oxopiperazine-1-carbonyl]benzonitrile
2-(2-phenyl-1,3-thiazol-4-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(3R,4R)-4-cyclopropyl-3-methyl-1-[(4-phenoxyphenyl)methyl]piperidin-4-ol
(2R)-2-amino-N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]-3-hydroxypropanamide
1-[4-(2-chlorophenyl)piperazin-1-yl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propan-1-one
3-cyclohexyl-N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-1H-pyrazole-4-carboxamide
N-[2-(furan-2-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-3-(4-methylphenyl)propanamide
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}spiro[2.3]hexane-1-carboxamide
(1s,4s)-4-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]cyclohexan-1-ol
ethyl 2-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-1,3-oxazole-4-carboxylate
2-(2-fluorophenoxymethyl)-N-[(1S)-2-hydroxy-1-phenylethyl]-1,3-oxazole-4-carboxamide
N-(isoquinolin-5-ylmethyl)-1-methyl-N-(pyridin-3-ylmethyl)piperidin-4-amine
3-[({1-[ethyl(methyl)amino]cyclohexyl}methyl)sulfamoyl]-N,N-dimethylbenzamide
2-{6,8-dioxo-2,7-diazaspiro[4.4]nonan-2-yl}-6-phenylpyridine-3-carboxylic acid
(4aS,8aR)-1-butyl-6-[4-(1H-imidazol-1-yl)butanoyl]-decahydro-1,6-naphthyridin-2-one
2-(3-methylbutyl)-8-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2,8-diazaspiro[5.5]undecan-3-one
3-{4-[(ethylcarbamoyl)amino]phenyl}-4-methylbenzamide
1-{4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}butan-1-one
2-(3-methyl-1,2-oxazol-5-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}acetamide
1-[(2-fluorophenyl)methoxy]-8-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)-1,8-diazaspiro[4.5]decan-2-one
N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
3-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[2-(4-fluorophenoxy)pyridin-3-yl]urea
N-{1-[2-oxo-2-(4-phenylazepan-1-yl)ethyl]-1H-pyrazol-4-yl}-2-phenoxyacetamide
(1H-imidazol-4-ylmethyl)({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)amine
N-[2-(1H-imidazol-4-yl)ethyl]-4-(trifluoromethyl)pyrimidin-2-amine
3-(pyrrolidine-1-carbonyl)-1-[(2,4,6-trimethoxyphenyl)methyl]piperazine
1-[2-(methylsulfanyl)phenyl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}urea
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
ethyl 4-[(4-chlorophenyl)methyl]-1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidine-4-carboxylate
1-(2-amino-5,6,7,8-tetrahydroquinazolin-4-yl)-3-[(dimethylamino)methyl]pyrrolidin-3-ol
4-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-1-(2-phenylphenyl)piperazin-2-one
(3S,4S)-4-(dimethylamino)-1-(trimethylpyrimidin-4-yl)pyrrolidin-3-ol
N-[(3S,4R)-4-(4-methoxyphenyl)-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]pyrrolidin-3-yl]acetamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-5-(methoxymethyl)thiophene-2-carboxamide
6-(1-benzofuran-2-yl)-5-chloro-2-methylpyrimidin-4-ol
2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-N-[2-(1H-pyrazol-4-yl)ethyl]-1,3-oxazole-4-carboxamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-6-methyl-2-(morpholin-4-yl)pyrimidin-4-amine
1-cyclopentyl-N-methyl-6-oxo-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidine-3-carboxamide
N-[4-(3-methylphenyl)phenyl]-1-(1,3-thiazole-4-carbonyl)piperidine-4-carboxamide