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2-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]pyridin-3-ol
4-{[4-(4-fluorophenoxy)piperidin-1-yl]methyl}-2-(propan-2-yl)pyrimidine
N,8-dimethyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
5-(2-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-methyl-3-(2-methylpropyl)-N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-5-carboxamide
2-({2-[1-(1-tert-butyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N-[2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-3-(thiophen-2-yl)propanamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2-(dimethylamino)-2-(3-fluorophenyl)acetamide
1,6-dimethyl-3-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-1,2-dihydropyridin-2-one
5-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]-4-methyl-1,3-thiazol-2-amine
3-(4-methyl-1,3-thiazol-5-yl)-1-(3-{5-methyl-2-[(pyridin-3-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidin-1-yl)propan-1-one
2-[5-(oxolan-3-yl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl]acetic acid
N-[(2,5-dimethylphenyl)(pyridin-3-yl)methyl]-1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-{[6-(3,5-dimethyl-1H-pyrazol-4-yl)quinazolin-4-yl]amino}ethan-1-ol
1-ethyl-5-{4-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
(3R,4S)-1-(5-chloro-2-fluorobenzoyl)-4-cyclopropylpyrrolidin-3-amine
N5-[(5-chlorothiophen-2-yl)methyl]-1-cyclopentyl-N3,N3-diethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
7-fluoro-2-methyl-4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]quinoline
N-[3-(4-fluorophenyl)-3-(furan-2-yl)propyl]-2-hydroxyacetamide
1-(2-amino-9H-purin-6-yl)-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
4-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1-(2-methoxyphenyl)-1H-pyrazole
3-(2-fluorophenoxymethyl)-1-[4-(1H-pyrazol-3-yl)benzoyl]piperidine
4-(4-methyl-1H-pyrazol-1-yl)-1-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperidine-4-carboxylic acid
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(3-methylfuran-2-carbonyl)piperidin-3-yl]propanamide
(4aR,7aS)-N,N-dimethyl-6,6-dioxo-4-(3-phenoxypropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
{[2-(cycloheptanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
N-(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)-3-methyl-5,6-dihydro-1,4-dioxine-2-carboxamide
1-({[(2-ethoxypyridin-3-yl)methyl]carbamoyl}methyl)piperidine-4-carboxamide
methyl 8-(2-ethylbutyl)-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
2-(1-{1-[3-(furan-2-yl)benzoyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-2-amine
[(2-cyclohexylpyrimidin-5-yl)methyl](methyl){[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}amine
1-(1-carbamoylcyclopropanecarbonyl)-4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
5-[(4S,4aS,8aR)-4-hydroxy-4-phenyl-decahydroquinoline-1-carbonyl]-N-ethyl-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
2-{[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
N-(1-{1-[(2-chloro-4-fluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-methylbutanamide
[(3R,4R)-4-(morpholin-4-ylmethyl)-1-(3-phenyl-1H-pyrazole-5-carbonyl)pyrrolidin-3-yl]methanol
5-(2-methoxybenzoyl)-1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[2-methoxy-5-({methyl[(4-methyl-1,3-thiazol-2-yl)methyl]amino}methyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
(1-methoxypropan-2-yl)({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)amine
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
1-(1-methyl-1H-pyrazole-4-carbonyl)-3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-[4-(4-methoxybenzoyl)piperazin-1-yl]-2-(2-methyl-1H-imidazol-1-yl)propan-1-one
(2S)-2-amino-3-(4-hydroxyphenyl)-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)propanamide
(1H-imidazol-2-ylmethyl)(methyl){[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}amine
N-{[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-(2,3-dihydro-1H-inden-1-yl)acetamide
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzamide
2-{3,5-dimethyl-4-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-amido]-1H-pyrazol-1-yl}acetic acid
1-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-4-(3-methylpyridin-2-yl)piperazine
N-(2,3-dihydro-1H-inden-1-yl)-4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}benzamide
ethyl 4-{[3-(5-chloro-2-methoxybenzoyl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylate