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2-{[5-(2-chlorophenyl)-1,2-oxazol-3-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
3-(1H-imidazol-2-yl)-1-(oxane-4-carbonyl)piperidine
4-{[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]amino}-5-methyl-N-[(1-phenylcyclopentyl)methyl]thieno[2,3-d]pyrimidine-6-carboxamide
1-[(3-methoxyphenyl)methyl]-N-[(2-propylpyrimidin-5-yl)methyl]piperidin-3-amine
(1R,5R)-6-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
5-acetamido-1-ethyl-2-(2-fluorophenyl)-N-[2-(1,3-thiazol-4-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
N-(1-{1-[2-(4-acetylphenoxy)acetyl]piperidin-4-yl}-2-(3-methoxyphenyl)ethyl)-N-methylcyclopropanecarboxamide
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(4-fluorophenoxy)ethan-1-one
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-2-(pyridin-3-yl)acetamide
2-amino-4-(5-ethylfuran-2-yl)-6-(3-hydroxyphenyl)pyridine-3-carbonitrile
2-[5-({8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)-1,2,4-oxadiazol-3-yl]pyrazine
(3S,4S)-4-(naphthalen-2-yl)-1-(pyridine-3-carbonyl)piperidin-3-ol
N-{[2-(dimethylamino)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
7-(oxan-4-yl)-2-(1,2-oxazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]-N-(2-oxoazepan-3-yl)acetamide
3-(2-{[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}ethyl)-1,3-oxazolidin-2-one
1-[7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-2-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
2-(4-acetylphenoxy)-1-{3-[benzyl(methyl)amino]piperidin-1-yl}ethan-1-one
N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
N,N-dimethyl-6-(4-methylthiophen-3-yl)pyridine-2-carboxamide
2-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-4H-chromen-4-one
3-amino-N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]propanamide
1-{9-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-1-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl}-2-(methylsulfanyl)ethan-1-one
4-(1-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}ethyl)morpholine
1-(morpholin-4-yl)-3-[1-(pyridin-4-ylmethyl)piperidin-4-yl]propan-1-one
3-{3-hydroxy-5-[2-(piperidin-2-yl)ethyl]phenyl}-4-methylbenzamide
N-{[2-(dimethylamino)-5,6,7-trimethoxyquinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]-3-(4-methylphenyl)propanamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[(4-methoxypyridin-2-yl)methyl]-N-methylacetamide
2-(4-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}piperazin-1-yl)pyrimidine
N-[2-(3-methoxyphenyl)-1-{1-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}ethyl]-N,3-dimethylbutanamide
2-cyclopropyl-4-phenyl-9-(pyridine-4-carbonyl)-2,9-diazaspiro[5.5]undecane
3-(cyclohex-1-en-1-yl)-5-[(pyridin-2-ylmethyl)sulfamoyl]benzoic acid
5-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-N-methyl-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-chloro-6-[3-(1H-imidazol-2-yl)piperidin-1-yl]pyridine-3-carboxylic acid
1-(2-methoxyphenyl)-3-{1-[1-(pyridine-4-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
3-(3-{1-[(4-methanesulfonylphenyl)methyl]-1H-pyrazol-3-yl}phenyl)-6-methylpyridazine
1-(2,2-difluoroethyl)-3-(2,3-dimethoxyphenyl)pyrrolidine
N-(1-methanesulfonylpiperidin-4-yl)-5-methyl-2-phenyl-1H-imidazole-4-carboxamide
1-cyclopentyl-4-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
N-[2-phenyl-2-(piperidin-1-yl)ethyl]-3-(pyridin-3-yl)propanamide
3-ethyl-8-(5-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-[(2S)-1-(3,6-dimethyl-1-benzofuran-2-carbonyl)pyrrolidin-2-yl]-3-methyl-1,2,4-oxadiazole
1-(2,3-dihydro-1H-inden-4-yl)-3-{2-[5-(hydroxymethyl)-1,2,4-oxadiazol-3-yl]ethyl}urea
{5-[3-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]furan-2-yl}methanol
(2,1,3-benzoxadiazol-4-ylmethyl)(methyl)[3-(oxolan-2-yl)propyl]amine
6-fluoro-4-[2-(6-methylpyridin-2-yl)ethyl]-3,4-dihydro-2H-1,4-benzoxazin-3-one
3-(4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}phenyl)-1H-1,2,4-triazole
N-methyl-7-oxo-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-3-(2-oxopyrrolidin-1-yl)propanamide
1-[4-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(4-ethylpiperazin-1-yl)ethan-1-one