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1-(2-ethoxyphenyl)-4-[(1-ethyl-1H-imidazol-2-yl)methyl]piperazine
1-{4-[(1,3-benzothiazol-5-yl)amino]piperidin-1-yl}ethan-1-one
2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)-N-[2-(pyrazin-2-yl)ethyl]acetamide
1-(azocan-1-yl)-3-(4-{[benzyl(methyl)amino]methyl}-2-methoxyphenoxy)propan-2-ol
(4aS,7aR)-1-[(2-chlorophenyl)methyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{1-[2-(dimethylamino)ethyl]-4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl}-N-phenylpiperidine-1-carboxamide
2-{1-cyclopentyl-4-[(3-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N,N,4-trimethyl-3-({[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]carbamoyl}methyl)-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
1-{[3-(2-chlorophenyl)-1,2-oxazol-5-yl]methyl}-4-(1H-imidazol-2-yl)-1H-1,2,3-triazole
4-methoxy-1-[5-(phenoxymethyl)-1,2-oxazole-3-carbonyl]piperidine
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-5-(1,3-oxazol-5-yl)thiophene-2-sulfonamide
4-{3-[3-(3-{pyrazolo[1,5-a]pyrimidin-3-yl}phenyl)-1H-pyrazol-1-yl]propyl}morpholine
N-(1-{[1-(carbamoylmethyl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}piperidin-3-yl)pyrrolidine-1-carboxamide
methyl 1-[(3R,5S)-5-[4-(4-fluorophenyl)piperazine-1-carbonyl]-1-{[3-(2-methylphenyl)phenyl]methyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
4-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]-3-methyl-2-propyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(2S,4R)-N-(2-phenylethyl)-1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
7-[3-(2-methoxyethyl)-1-(4-methylpyridin-2-yl)-1H-1,2,4-triazol-5-yl]-1,2,3,4-tetrahydroquinoxalin-2-one
4-[2-(3-fluorophenyl)ethyl]-11-{methyl[(4-methyl-1,3-thiazol-2-yl)methyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-ethyl-3-{1-[2-(1H-indol-1-yl)acetyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(4-chlorophenyl)-5-methyl-4-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)piperazin-2-one
2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]acetamide
4-{2-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]-2-oxoethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
3-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-4-(1-phenylethyl)-4H-1,2,4-triazole
9-methyl-3-[6-(4H-1,2,4-triazol-4-yl)pyridine-2-carbonyl]-3,9-diazaspiro[5.6]dodecane
N3-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]piperidine-1,3-dicarboxamide
2-methyl-7-(oxolane-2-carbonyl)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-[2-(4-chlorophenyl)ethyl]-N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-6-oxopiperidine-3-carboxamide
methyl 3-[4-(2-methoxybenzoyl)piperazine-1-carbonyl]benzoate
methyl 4-(5-chloro-2-{[(1-methylpiperidin-3-yl)formamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)benzoate
2-(cyclopropylmethyl)-N-(prop-2-en-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[2-(2-hydroxyethoxy)ethyl]-2-[(prop-2-en-1-yl)amino]benzamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(4-methylphenyl)acetamide
N-(1-carbamoylcyclopentyl)-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
3-hydroxy-1-(2-methoxyethyl)-3-{[(thiophen-2-ylmethyl)amino]methyl}piperidin-2-one
1-ethyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]benzamide
1-(4-phenylpiperazin-1-yl)-3-[1-(1,2,3,4-tetrahydronaphthalen-2-yl)piperidin-4-yl]propan-1-one
(1R,5R)-6-(cyclobutylmethyl)-3-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-3,6-diazabicyclo[3.2.2]nonane
1-[2-(dimethylamino)ethyl]-4-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}pyrrolidin-2-one
N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
9-[2-(5-fluoro-2-methylphenyl)acetyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
3-cyclopropyl-1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazole
2-{4-[(5,8-dimethoxy-4-methylquinolin-2-yl)amino]piperidin-1-yl}acetamide
3-({3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}methyl)benzonitrile
4-(4-{[(4-methoxyphenyl)methyl]amino}piperidin-1-yl)-N-[2-(morpholin-4-yl)ethyl]benzamide
N-[2-(N-methylmethanesulfonamido)ethyl]-1-oxo-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
4-{2-[5-(hydroxymethyl)furan-2-yl]-1H-imidazol-1-yl}benzene-1-sulfonamide
N-[3-(3-ethylphenoxy)propyl]-N-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-{[2-(trifluoromethyl)phenyl]methyl}propanamide
methyl 2-[3-(2-{[(2-fluorophenyl)methyl]carbamoyl}ethyl)piperidine-1-carbonyl]benzoate