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N-(2-{7-[(4-methoxy-2,3-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-4-methylbenzamide
N-tert-butyl-2-[6-oxo-4-(piperazin-1-yl)-1,6-dihydropyridazin-1-yl]propanamide
N-[(2S,4R,6S)-2-benzyl-6-(1-methyl-1H-imidazol-2-yl)oxan-4-yl]benzamide
N-(5-{[3-(2-chlorophenyl)-1-(cyclopropylmethyl)-2-oxo-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-6-yl]methyl}thiophen-2-yl)acetamide
N-methyl-2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-N-(1H-pyrazol-5-ylmethyl)acetamide
2-({[2-(dimethylamino)ethyl]({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)amino}methyl)-3-methoxyphenol
N-(3-chloro-4-fluorophenyl)-3-{1-[2-(4H-1,2,4-triazol-4-yl)ethyl]piperidin-4-yl}propanamide
3-(3,4-difluorophenyl)-5-(2-phenylethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
N-ethyl-2-[3-ethyl-3-(hydroxymethyl)piperidin-1-yl]acetamide
4-[(1-{[1-(pyrimidin-2-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]thiomorpholine
2-(2,6-dimethoxypyridin-3-yl)-2-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}acetic acid
3-methoxy-N-[1-(7-{[4-(2-methylphenyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]benzamide
5-(1H-1,3-benzodiazole-5-carbonyl)-1-[2-(4-methoxyphenyl)ethyl]-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(furan-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-[(1S,5R)-3-[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
5-methanesulfonyl-2-methyl-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}pyrimidin-4-amine
2-({[(3R,4R)-4-(hydroxymethyl)-1-[1-(3-methylphenyl)piperidin-4-yl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-[(3S,4R)-4-(4-methoxyphenyl)-1-(propane-2-sulfonyl)pyrrolidin-3-yl]acetamide
1-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)-2-(2,3,6-trimethylphenoxy)ethan-1-one
2-{1-[(1-{7-methylthieno[3,2-d]pyrimidin-4-yl}piperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}propan-2-amine
N-ethyl-N-[2-(morpholin-4-yl)ethyl]quinoline-2-carboxamide
4-(2,6-dimethylquinoline-4-carbonyl)-1-(3-methoxyphenyl)-6-methylpiperazin-2-one
1-butyl-4-{1-[4-(1H-pyrazol-1-yl)phenyl]piperidin-4-yl}piperazine
3-(3,4-dimethoxyphenyl)-1-[4-(4H-1,2,4-triazol-3-ylmethyl)piperazin-1-yl]propan-1-one
(1S,3R)-3-[1-(4-methylpyridin-2-yl)-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-5-yl]cyclohexan-1-amine
N-[(3-chlorophenyl)methyl]-3-(1-cyclohexylpiperidin-4-yl)propanamide
{1-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
N,N-dimethyl-7-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-cyclopropyl-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}piperazine-2-carboxamide
5-methyl-4-(4-methylpiperazin-1-yl)-N-[(1-phenylcyclopentyl)methyl]thieno[2,3-d]pyrimidine-6-carboxamide
3-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-3-methyl-1-[3-(piperidin-1-ylmethyl)phenyl]urea
N-[2-(azepan-1-yl)-2-phenylethyl]pyrimidin-2-amine
N-{[4-methoxy-3-(pyridin-3-ylmethoxy)phenyl]methyl}-4-oxo-N-[(3S)-2-oxoazepan-3-yl]-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
4-methyl-N-[1-(thiophen-2-ylmethyl)piperidin-3-yl]pyrimidin-2-amine
(1R,3S)-3-methoxy-7-[4-(2-methoxyphenyl)benzoyl]-7-azaspiro[3.5]nonan-1-ol
2-(1-ethylpiperidin-4-yl)-N-{1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}acetamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(2,3-dihydro-1,4-benzodioxine-5-carbonyl)piperidin-3-ol
(3S)-1-[4-(2-methoxyphenyl)benzoyl]-N,N-dimethylazepan-3-amine
2-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]thiophen-3-amine
N-(2-methoxyethyl)-3-(1H-pyrazol-1-yl)-N-(1,3-thiazol-2-ylmethyl)benzamide
N-(2,2-dimethyloxan-4-yl)-N-ethyl-4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
1-(4-{[4-(2-methanesulfonylethyl)piperazin-1-yl]methyl}thiophen-2-yl)ethan-1-one
4-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}-1-(thiophene-2-carbonyl)piperidine
methyl (2S,4R)-1-[(3-chlorophenyl)methyl]-4-[3-(4-methylphenyl)propanamido]pyrrolidine-2-carboxylate
(2E)-N-{[4-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)-3-(thiophen-2-yl)prop-2-enamide
3-methyl-3-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1-[3-(sulfamoylmethyl)phenyl]urea
N-ethyl-1-[(3-methoxyphenyl)methyl]-5-(quinolin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-cyclopropyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(1H-pyrrol-1-yl)propanamide
1,3,6-trimethyl-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N,N-dimethyl-4-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]aniline