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1-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-(pyrrolidine-1-carbonyl)piperidine
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-{[(4-methoxy-2,3-dimethylphenyl)methyl]amino}-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
3-(3-methoxyphenoxymethyl)-1-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
2-butyl-N-(3-methanesulfonamidophenyl)-2,5-dihydro-1H-pyrrole-1-carboxamide
(3R,5S)-N-(2-phenylethyl)-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
2-(2-methoxypyridine-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-{[3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]methyl}quinolin-4-ol
2-methylpropyl 9-oxo-8-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecane-2-carboxylate
N-[2-(1-benzylpiperidin-2-yl)ethyl]pyrimidin-4-amine
1-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]-4-(3-methylpyridin-4-yl)piperazine
1-{1-[(2,4-dimethylphenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
N-[(7R,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-ethyl-3,5-dimethyl-1H-pyrazole-4-carboxamide
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
(cyclopentylmethyl)[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
(3S,5R)-1-benzyl-3-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-5-(pyrrolidine-1-carbonyl)piperidine
N-[2-(3-chlorophenyl)ethyl]-5-methyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
N-cyclohexyl-N-[(4-fluorophenyl)methyl]oxolane-3-carboxamide
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
2-{2-[3-(1H-imidazol-1-yl)propoxy]phenyl}-6,7-dimethyl-1H-1,3-benzodiazole
4-[4-(5-chloropyridin-2-yl)piperazine-1-carbonyl]-1-cyclopropylpyrrolidin-2-one
4-{3-[2-(2,4-difluorophenyl)ethyl]piperidine-1-carbonyl}-2,6-dimethylpyrimidine
2-{4-[(5-chloro-2,3-dimethoxyphenyl)methyl]-1-(3-methylbutyl)piperazin-2-yl}ethan-1-ol
N-(cyclopropylmethyl)-1-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[cyclohexyl(methyl)amino]-3-(2-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}phenoxy)propan-2-ol
{4-[3-(trifluoromethyl)phenyl]pyridin-2-yl}methanol
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2,3-dihydro-1-benzofuran-7-carboxamide
3-(but-3-en-1-yl)-1-(cyclopropylmethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)(thiophen-3-ylmethyl)amine
4-{4-[(4-fluorophenyl)methyl]piperazin-1-yl}-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
3-[(5-methyl-1,2-oxazol-3-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[2-(4-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-2,2-dimethyloxan-4-amine
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-(ethylamino)pyrimidine-5-carboxamide
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-4-[(2-methylprop-2-en-1-yl)oxy]benzamide
1-{[1-(2-methylpyridin-4-yl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}piperidin-2-one
N-(1,3-dihydroxypropan-2-yl)-6-(2-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-[6-(trifluoromethyl)pyridin-2-yl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(1S,5R)-3-cyclobutanecarbonyl-6-(2-methylfuran-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[(3,5-dimethylphenyl)methyl]-4-[(4-hydroxy-2-methoxyphenyl)methyl]piperazin-2-one
N-cyclohexyl-N-[2-(ethylsulfanyl)ethyl]-1-(2-hydroxyethyl)-1H-1,3-benzodiazole-5-carboxamide
4-(2-ethoxyacetyl)-5-methyl-1-(2-phenylphenyl)piperazin-2-one
N-(2-{4-[(3-hydroxyphenyl)methyl]morpholin-2-yl}ethyl)pyridine-3-carboxamide
3-{[5-(2-fluoro-4,5-dimethoxyphenyl)-1H,4H-pyrazolo[3,4-d]imidazol-1-yl]methyl}pyridine
N-(2-methoxyethyl)-3-{[1-(5-methylhex-5-en-2-yl)piperidin-4-yl]oxy}benzamide
1-cyclohexyl-N3-cyclopropyl-N5-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-[(3R,4S)-1-(oxan-4-yl)-4-propylpyrrolidin-3-yl]-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
4-(3,3-dimethylpyrrolidine-1-carbonyl)-2-[2-(propan-2-yl)pyrimidin-5-yl]quinoline
4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-1,3λ6,4-oxathiazinane-3,3-dione
N-{[4-(benzyloxy)-3-methoxyphenyl]methyl}-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)-3,5-dimethyl-1H-indole