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5-amino-N-{[2-(dimethylamino)pyridin-3-yl]methyl}-4-phenyl-1H-pyrazole-3-carboxamide
3-[3-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-5-methyl-1H-indazole
N,N-dimethyl-6-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrazin-2-amine
[(3R,4S)-1-[2-(benzyloxy)ethyl]-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-3-azaspiro[5.5]undecan-9-amine
N-(butan-2-yl)-3-{[2-(5-methylfuran-2-yl)ethyl]sulfamoyl}benzamide
2-(3-{4-[(3-cyanophenyl)methyl]piperazine-1-carbonyl}piperidin-1-yl)acetamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-5-[(3-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
N-methyl-3-({9-oxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}sulfonyl)benzamide
1-cyclobutanecarbonyl-N-[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]piperidine-4-carboxamide
(2S,4R)-4-amino-1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-(1,4-dioxan-2-ylmethyl)-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1H-indole-6-carboxamide
1-[4-(pyridin-4-yl)piperidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(3-methoxyphenyl)methyl]acetamide
3-[5-(1,5-dimethyl-1H-indazole-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-2,5,6-trimethylpyrimidin-4-amine
1-[4-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)piperazin-1-yl]ethan-1-one
6-(dimethylamino)-N-[(8-methoxyquinolin-5-yl)methyl]-N-methylpyridine-3-carboxamide
methyl 3-[4-(isoquinoline-3-carbonyl)-6-[(3-methoxyphenyl)methoxy]-2-oxo-1,4-diazepan-1-yl]propanoate
6-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-cyclopropyl-N-(1-methoxybutan-2-yl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
1-[1-(2H-1,3-benzodioxol-5-ylmethyl)piperidin-3-yl]-N-cyclopentyl-1H-1,2,3-triazole-4-carboxamide
N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)thiophene-2-sulfonamide
1-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-4-phenoxypiperidine-4-carboxylic acid
2-[3-(benzyloxy)propyl]-2,7-diazaspiro[4.5]decan-6-one
N,N-dimethyl-6-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidin-4-amine
2-[4-({4-[hydroxy(phenyl)methyl]-1H-1,2,3-triazol-1-yl}methyl)piperidin-1-yl]pyridine-3-carbonitrile
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-1-phenylcyclopropane-1-carboxamide
1-[7-(5-chloropyridin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-methylbutan-1-one
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}acetamide
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-2-(2-methoxyethyl)-1,3-benzoxazole-6-carboxamide
(2S,4S)-4-amino-1-[(2-chloro-4-ethoxy-5-methoxyphenyl)methyl]-N-methylpyrrolidine-2-carboxamide
(3S,4R)-1-(4-cyanooxane-4-carbonyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-[(4-methoxypyridin-2-yl)methyl]-2-(pyridin-2-yl)acetamide
(1R,7S)-N-methyl-4-oxo-3-(pyridin-3-ylmethyl)-N-(thian-4-yl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
5-cyclopropyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-methyl-1,3,4-oxadiazol-2-amine
7-[(2-methyl-1,3-benzothiazol-6-yl)sulfonyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-3-(methylsulfanyl)propanamide
N-{1-oxa-8-azaspiro[4.5]decan-3-yl}-2-(pyridin-3-yl)acetamide
5-[(3S)-3-(dimethylamino)azepane-1-carbonyl]-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
4-(2-{5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-6-yl}ethyl)benzene-1-sulfonamide
4-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-1-[(4-methylphenyl)methyl]piperazin-2-one
(2R,3S,6R)-5-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(3R,4S)-4-cyclopropyl-N,N-dimethyl-1-(2-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)pyrrolidin-3-amine
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[2-(dimethylamino)ethyl]-N-methylacetamide
(2R,3R,6R)-5-(4-methyl-1H-pyrrole-2-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-cyclopentyl-2-{[3-(5-methyl-2H-1,2,3,4-tetrazol-2-yl)adamantan-1-yl]amino}propanamide
(3S,4S)-N-[3-(4-chlorophenyl)phenyl]-4-[(dimethylamino)methyl]-3-hydroxypiperidine-1-carboxamide