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N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}pyridine-2-carboxamide
2-{4-[4-(adamantan-2-yl)piperazine-1-carbonyl]-5-cyclopropyl-1H-pyrazol-1-yl}-4-(furan-2-yl)pyrimidine
(2R,3R,6R)-5-[(2,6-dimethoxyphenyl)methyl]-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(2-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}-4-(thiophen-2-yl)phenoxy)acetic acid
8-fluoro-2-{[2-(pyridin-3-yl)piperidin-1-yl]methyl}quinolin-4-ol
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-2-(2,5-dimethoxyphenyl)acetamide
1-[3-(1H-imidazol-2-yl)piperidin-1-yl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
1-{4-[5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazin-1-yl}ethan-1-one
2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]-4-(1H-1,2,3,4-tetrazol-1-yl)phenol
3-(morpholine-4-carbonyl)-N-[3-(1H-pyrazol-1-yl)propyl]benzene-1-sulfonamide
5-{[4-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}pentan-1-ol
6-cyano-N-[(3R,5S)-5-(diethylcarbamoyl)-1-propylpyrrolidin-3-yl]pyridine-3-carboxamide
N-({2-[2-(3-fluorobenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-2-methylpyridine-3-carboxamide
(1S,5R)-6-[(5-propylfuran-2-yl)methyl]-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-cyclopentyl-N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}acetamide
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)propanamide
2-hydroxy-1-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
4-ethyl-5-methyl-6-[2-(morpholin-4-ylmethyl)-1,4-oxazepan-4-yl]pyrimidin-2-amine
(2R,3R,6R)-5-(cyclopropanesulfonyl)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(3S,5S)-1-methyl-5-[3-(3-methylphenoxy)azetidine-1-carbonyl]pyrrolidin-3-amine
5-{2-amino-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl}-2,3-dimethylbenzene-1-sulfonamide
5-(4-fluoro-2-methylphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
6-methyl-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)imidazo[2,1-b][1,3]thiazole-5-carboxamide
N-(5-tert-butyl-2-methoxyphenyl)-4,4-difluoropiperidine-1-carboxamide
N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-{[5-chloro-7-(1H-indol-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-methyl-1,2-oxazole-3-carboxamide
5-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-2-methyl-3,4-dihydropyrimidin-4-one
1-[3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-3-(thiophen-2-yl)propan-1-one
2-(2-chloro-4-fluorophenoxymethyl)-N-[(6-methylpyridin-2-yl)methyl]-1,3-oxazole-4-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
N-[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]-1-(propan-2-yl)piperidine-4-carboxamide
N-[(4-methanesulfonylphenyl)methyl]-N-methyl-2,3-dihydro-1H-inden-2-amine
7-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]-2-oxa-7-azaspiro[4.5]decan-8-one
4-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(pyrazin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[2-({1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-4-yl}amino)ethyl]methanesulfonamide
1-{pyrazolo[1,5-a]pyridine-3-carbonyl}-3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine
2-(methylamino)-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}pyrimidine-5-carboxamide
3-(3-cyanophenyl)-1-(1-methylpiperidin-4-yl)-1-(pyridin-4-ylmethyl)urea
3-amino-N-benzyl-N-(cyclopropylmethyl)benzamide
(1S,5R)-1,3,3-trimethyl-6-{1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-6-azabicyclo[3.2.1]octane
N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-6-carboxamide
4-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-4-oxobutanoic acid
4-{[ethyl(propan-2-yl)amino]methyl}-N-(4-ethyl-1,3-dimethyl-1H-pyrazol-5-yl)benzamide
(2R,3S,6R)-3-(3-methoxyphenyl)-5-(1,3-thiazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
[(5-{2-[(4-fluorophenyl)methyl]morpholine-4-carbonyl}furan-2-yl)methyl]dimethylamine
N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-methyl-1,2,5-oxadiazole-3-carboxamide
2-[1-cyclopentyl-4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperazin-2-yl]ethan-1-ol
2-{[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]methyl}benzoic acid
3-cyclohexyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1H-pyrazole-4-carboxamide