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N-({1-[(3,5-dimethoxyphenyl)methyl]pyrrolidin-3-yl}methyl)methanesulfonamide
1-(2,4-dimethoxybenzoyl)-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
N-[(2-ethoxyphenyl)methyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
(4aR,8aS)-6-benzyl-1-[(3,4,5-trimethoxyphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
4-{1-hydroxy-2-[4-(2-phenylethyl)-1H-1,2,3-triazol-1-yl]ethyl}phenol
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-[(1-methyl-1H-imidazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-{2-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}acetamide
1-cycloheptyl-N-[1-(pyridin-3-yl)propan-2-yl]-1H-1,2,3-triazole-4-carboxamide
(1S,5R)-6-(2-methyl-1H-pyrrole-3-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
N-{[(2S,4S)-4-fluoro-1-[3-(furan-2-yl)propanoyl]pyrrolidin-2-yl]methyl}-2-phenoxyacetamide
4-{[2-(2,3-dihydro-1H-indol-1-yl)ethyl]amino}-1λ4-thian-1-one
(3S,4S)-4-({[(2E)-2-methyl-3-phenylprop-2-en-1-yl]amino}methyl)piperidin-3-ol
8-(3,5-dimethyl-1-benzofuran-2-carbonyl)-1-oxa-8-azaspiro[4.6]undecane
N4-ethyl-N2-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}pyrimidine-2,4-diamine
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]ethan-1-one
2-cyclopentyl-N-[3-(4-{[(5-phenyl-4H-1,2,4-triazol-3-yl)methyl]amino}piperidin-1-yl)phenyl]acetamide
3-{5-[3-(2,3-dihydro-1H-isoindol-2-yl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
2'-amino-4'-[5-(hydroxymethyl)furan-2-yl]-7',8'-dihydro-5'H-spiro[piperidine-4,6'-quinoline]-3'-carbonitrile
2-tert-butyl-4-hydroxy-N-[2-(4-sulfamoylphenyl)ethyl]pyrimidine-5-carboxamide
4-{[5-(1-cycloheptylpiperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}morpholine
2-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-4,6-dimethylpyridine-3-carbonitrile
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-propylpiperidine
N-benzyl-4-[5-(3-phenylpropanamido)-1H-pyrazol-1-yl]piperidine-1-carboxamide
3-(2-methoxyphenyl)-1-methyl-3-{2-oxo-2-[3-(3-phenylpropanoyl)piperidin-1-yl]ethyl}pyrrolidine-2,5-dione
4-[(1R,7S)-3-(2-methoxyethyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carbonyl]-1λ6-thiomorpholine-1,1-dione
2-(dimethyl-1,2-oxazol-4-yl)-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
2-(propan-2-yl)-5-{4-[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carbonyl}pyrimidine
2-(3-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}phenoxy)acetamide
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
2-methyl-4-(2-methylphenyl)-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}piperazine
1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(furan-2-yl)ethane-1,2-dione
N-(1H-1,3-benzodiazol-5-yl)-2-(pyrrolidin-3-yl)benzamide
3-{[(7-methanesulfonyl-4-methylquinazolin-2-yl)(methyl)amino]methyl}phenol
methyl 4-[5-({methyl[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]amino}methyl)-1,2,4-oxadiazol-3-yl]benzoate
1-[(diethylcarbamoyl)methyl]-N-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(4-chlorophenyl)methyl]-N-[(2-methoxyphenyl)methyl]pyrrolidine-2-carboxamide
1-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-3-(methylsulfanyl)propan-1-one
[(1-ethylpyrrolidin-2-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})[(2-methyl-1,3-thiazol-5-yl)methyl]amine
(2R,6R)-11-methoxy-4-[2-(morpholin-4-yl)acetyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-{4-[(6-chloro-2H-chromen-3-yl)methyl]-1-(thiophen-3-ylmethyl)piperazin-2-yl}ethan-1-ol
1-[1-(2-amino-2-methylpropanoyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-({1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}methyl)piperidine-4-carboxamide
5-(2,4-difluorophenoxymethyl)-N-[2-(2-methyl-1H-indol-1-yl)ethyl]-1,2-oxazole-3-carboxamide
(1R,5R)-6-benzyl-3-(4-methylpyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-{[1-(2-methoxyethyl)piperidin-3-yl]methyl}-2-methyl-1-benzofuran-5-carboxamide
N-methyl-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide
3-(1-methoxybutan-2-yl)-1-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]urea
2-(4-{[3-(dimethylamino)piperidin-1-yl]methyl}phenyl)-5-fluoro-6-methyl-3,4-dihydropyrimidin-4-one
2-({3-[3-(2,3-dimethoxyphenyl)pyrrolidine-1-carbonyl]phenyl}amino)acetic acid
{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}({1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl})amine