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N-[2-(2-chlorophenyl)ethyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
3-[ethyl({[4-(pyridin-2-yl)phenyl]methyl})amino]-1λ6-thiolane-1,1-dione
3-(furan-3-ylmethyl)-9-methoxy-N-[(2-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
[(3,5-dimethoxyphenyl)methyl]({[7-methoxy-2-(thiophen-3-yl)quinolin-3-yl]methyl})amine
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,2,5-trimethylfuran-3-carboxamide
N,N-diethyl-1-{1-[(2,4,5-trimethoxyphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
1-{1-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]piperidin-4-yl}-N-(propan-2-yl)piperidine-4-carboxamide
N,N-dimethyl-4-[1-(piperidin-4-yl)-1H-imidazol-2-yl]aniline
[(3R,4R)-4-[(dimethylamino)methyl]-1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl]methanol
(2S,4R)-4-[(4-fluorophenyl)sulfanyl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1-{[4-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxamide
7-(cyclohexylmethyl)-2-(pent-4-enoyl)-2,7-diazaspiro[4.5]decan-6-one
N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
1-{1-[(3,4-dimethylphenyl)methyl]piperidin-4-yl}pyrrolidin-2-one
7-fluoro-2-methyl-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}quinoline-4-carboxamide
(1-{[1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
N-(1,3-dimethyl-1H-pyrazol-4-yl)-2-[2-(2-methoxyethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]acetamide
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-1-methyl-1H-pyrrole-2-carboxamide
6-methyl-N-[3-(4-methylpiperazin-1-yl)propyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
(3E)-1-{9-[(3-fluorophenyl)methyl]-1-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl}pent-3-en-1-one
N-[2-(cyclohex-1-en-1-yl)ethyl]-4-acetamido-N-{[2-(4-hydroxypiperidin-1-yl)-7-(methylsulfanyl)quinolin-3-yl]methyl}benzamide
N-cyclopropyl-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
4-cyclopropanecarbonyl-7-(5-methylthiophen-2-yl)-9-(oxan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-benzyl-N-(2-hydroxyethyl)-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]acetamide
methyl 6-(morpholin-4-ylmethyl)-3-(2-phenylacetamido)thieno[2,3-b]pyridine-2-carboxylate
N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
N,N-dimethyl-6-(2-phenylphenyl)pyridine-3-carboxamide
4-(1-ethyl-1H-1,2,4-triazol-5-yl)-3-(thiophen-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-cyclopropyl-N-{[2-(dimethylamino)-7-methylquinolin-3-yl]methyl}-2,3,4-trimethoxybenzamide
N-[4-({8-cyclopropyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}methyl)phenyl]acetamide
N,N-dimethyl-6-{3-[1-(pyridin-3-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyrimidin-4-amine
2-({[1-(2,2-dimethylpropyl)-3-hydroxy-2-oxopiperidin-3-yl]methyl}amino)-N-(2-methylphenyl)acetamide
1-methyl-2-(2-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}phenyl)-1H-imidazole
3-(4-benzyl-4-hydroxypiperidine-1-carbonyl)piperidine-1-carboxamide
6-ethyl-1,5-dimethyl-2-oxo-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,2-dihydropyridine-3-carboxamide
9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-3-[(5-methylfuran-2-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(5S,9aS,9bS)-2-(2,3-dihydro-1H-inden-2-yl)-5-[2-(dimethylamino)-1,3-thiazol-5-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
9-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
6-{9-oxo-8-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-2-yl}pyridine-2-carbonitrile
N-methyl-3-{spiro[azepane-4,2'-chromene]-1-ylmethyl}pyridin-2-amine
1-(azepan-1-yl)-3-[3-({[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]amino}methyl)phenoxy]propan-2-ol
4-[1-(1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)ethyl]morpholine
N-(oxan-4-ylmethyl)-1-(3-phenylphenyl)piperidin-4-amine
1-(2,3-dihydro-1H-inden-5-yl)-3-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]urea
2-{1-cyclohexyl-4-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperazin-2-yl}ethan-1-ol
(3S,5S)-1-cyclopentanecarbonyl-5-[(pyridin-4-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-3-(piperidin-1-yl)propanamide
N-(2-methylpropyl)-3-(2-oxopyrrolidin-1-yl)-N-[(2E)-3-phenylprop-2-en-1-yl]propanamide
2-[1-(2,2-dimethylpropyl)-4-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}piperazin-2-yl]ethan-1-ol
methyl 2-(3-methyl-4-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-2-oxopiperazin-1-yl)acetate