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(2S,4S)-1-cyclopentyl-4-[2-(2,5-dimethylphenyl)acetamido]-N-ethylpyrrolidine-2-carboxamide
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-[(2-phenyl-1H-imidazol-4-yl)methyl]piperazine
4-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-6-methyl-1,2-dihydroquinolin-2-one
2,6-dimethoxy-N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]pyrimidine-4-carboxamide
N-(2-{7-[(3-ethoxy-4-hydroxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-3-carboxamide
3-[(2-amino-5,6,7,8-tetrahydroquinazolin-4-yl)amino]-N-(1,3-thiazol-2-yl)propanamide
3-[(3S,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(naphthalen-1-yl)urea
(1R,5R)-N,N-dimethyl-6-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
6-methyl-N4-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]pyrimidine-2,4-diamine
(1S,5R)-3-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-3,9-diazabicyclo[3.3.2]decan-10-one
3-(1,3-diethyl-6-methyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-1-methyl-1-[3-(oxolan-2-yl)propyl]urea
4-(4-fluorophenyl)-1-[(3R,4R)-3-hydroxy-4-(4-methylpiperazin-1-yl)piperidin-1-yl]butan-1-one
2-[(3S,4R)-4-amino-1-[4-(1H-imidazol-1-yl)benzoyl]pyrrolidin-3-yl]ethan-1-ol
3-{[(3-methylphenyl)methyl]amino}-5-(methylsulfamoyl)-N-[3-(methylsulfanyl)phenyl]benzamide
4-methoxy-1-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)piperidine
(4aS,8aS)-2-{[3-(trifluoromethyl)phenyl]methyl}-decahydroisoquinolin-4a-ol
3-methyl-5-(3-methyl-5-propyl-1-benzofuran-2-yl)-1,2,4-oxadiazole
2-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridine-6-carbonyl]-3,5,7-trimethyl-1H-indole
2-(2-fluorophenoxymethyl)-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]-1,3-oxazole-4-carboxamide
methyl 1-(3-methylbutoxy)-8-(5-methylhex-5-en-2-yl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
2-{2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}-5,6-dimethyl-1H-1,3-benzodiazole
2-(2-chlorophenyl)-N-ethyl-N,3-dimethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N'-(2-ethoxyphenyl)-N-methylpropanediamide
2-[3-(4-hydroxy-4-phenylpiperidine-1-carbonyl)piperidin-1-yl]acetamide
N-[3-(pyridin-4-yl)propyl]-6-[2-(trifluoromethyl)benzoyl]-6-azaspiro[2.5]octane-1-carboxamide
N-(2-hydroxyethyl)-3-(5-{thieno[3,2-d]pyrimidin-4-yl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanamide
4-[3-(1-carbamoylethoxy)phenyl]-N,N-dimethylbenzamide
4-methyl-6-(2,4,6-trimethylphenyl)pyrimidin-2-amine
N-[3-(1H-indazol-1-yl)propyl]-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
1-(3,5-dimethyl-4-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}-1H-pyrrol-2-yl)ethan-1-one
2-oxo-8-[3-oxo-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N'-(2-ethoxyphenyl)-N-[2-(1-methylpyrrolidin-2-yl)ethyl]propanediamide
1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
4-(2-methoxy-6-methylbenzoyl)-2-(trifluoromethyl)morpholine
(3aS,6aS)-2-ethyl-5-{[4-(1H-imidazol-1-yl)phenyl]methyl}-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{4-[(2,4-difluorophenyl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}-2-(thiophene-2-sulfonamido)acetamide
2-butyl-8-(5-propyl-1,2-oxazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
5-(3,4-dihydro-2H-1-benzopyran-2-carbonyl)-3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-(1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-3-yl)-2-phenylethan-1-one
1-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
8-methoxy-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-(2-{7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
1-[4-(4-methoxybenzoyl)piperazin-1-yl]-2-(2-methoxyethoxy)ethan-1-one
7-fluoro-2-methyl-4-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]quinoline
2-{4-[(3-methyl-1H-pyrazol-5-yl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
(1R,2R,6S,7S)-4-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-azatricyclo[5.2.1.02,6]decane
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
2-(propan-2-yl)-5-[4-(pyrazin-2-yl)piperazine-1-carbonyl]-1,3-benzoxazole
1-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(4-fluorophenoxy)ethan-1-one