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{1-[(1-pentylpiperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}methanol
6-(benzyloxy)-1-(oxan-4-ylmethyl)-4-[(3,4,5-trimethoxyphenyl)methyl]-1,4-diazepan-2-one
N,1-dimethyl-6-(propan-2-yl)-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N5-(oxolan-2-ylmethyl)-N5-(pyridin-2-ylmethyl)-N6-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
1-[3-(2-methyl-1,3-thiazol-4-yl)phenyl]-N-[1-(pyridin-3-yl)propan-2-yl]piperidin-4-amine
1-[4-(4-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}piperidin-1-yl)benzoyl]piperidin-3-ol
4-{[3-(dimethylamino)propyl](methyl)amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
ethyl 1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-1H-pyrazole-3-carboxamide
2-(2-methyl-1H-imidazol-1-yl)-N-(1-methyl-1H-pyrazol-5-yl)acetamide
N-cyclopropyl-1-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}piperidine-3-carboxamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
4-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}piperazine-1-sulfonamide
3-[1-(1-methyl-2-oxo-1,2-dihydropyridin-3-yl)-N-(2-phenylethyl)formamido]propanamide
3-[(2-fluorophenyl)formamido]-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}propanamide
4-({3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}methyl)morpholine
4-(1-methyl-3-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-1,2,4-triazol-5-yl)morpholine
methyl 6-[(3,4-difluorophenyl)methyl]-2-(ethylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-[4-(adamantan-1-yl)piperazine-1-carbonyl]-2-cyclopropyl-6-methyl-1-(thiophen-2-ylmethyl)-1,4-dihydropyridin-4-one
5-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-1-ethyl-1H-indole-5-carboxamide
3-{2-[3-cyclopropyl-1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,2,4-triazol-5-amine
7-[(3-methoxyphenyl)methyl]-2-(3-methyl-1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decane
1-[6-(2-hydroxyethyl)pyrazolo[1,5-a]pyrimidine-3-carbonyl]-1,4-diazepan-6-ol
2-ethyl-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-[butyl(methyl)amino]-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-(2-{4-azatricyclo[4.3.1.13,8]undecan-4-yl}-2-oxoethyl)-1-cyclopropyl-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
(2-{2-[1-(5-fluoro-2-methoxybenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
1,3,6-trimethyl-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
7-(4-amino-6,7-dimethoxyquinazolin-2-yl)-2,7-diazaspiro[4.4]nonane-1,3-dione
4-methyl-2-{2-[2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
3-{1-methyl-4-[3-(methylsulfanyl)propyl]-1,4,9-triazaspiro[5.5]undecane-9-carbonyl}benzonitrile
3-[4-(3-chlorophenyl)-3-oxopiperazin-1-yl]-N-[(4-methylphenyl)methyl]propanamide
4-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-4-oxobutanamide
2-{4-[(2-butyl-1H-imidazol-4-yl)methyl]-1-(3-methylbut-2-en-1-yl)piperazin-2-yl}ethan-1-ol
5-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-2-amine
1-(3-{[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}piperidin-1-yl)ethan-1-one
3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}-N-[1-(pyridin-3-yl)propan-2-yl]propanamide
3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-5,6,7-trimethoxy-1,2-dihydroquinolin-2-one
[3-(2-methoxyethyl)-1-(6-methoxypyrimidin-4-yl)piperidin-3-yl]methanol
1-(4-chlorophenyl)-4-(2-ethoxypyridine-3-carbonyl)-5-methylpiperazin-2-one
8-(4,6-dimethoxypyrimidin-2-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
(4aS,8aS)-2-(6-methylpyridin-2-yl)-decahydro-2,7-naphthyridin-4a-ol
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-hydroxypyridine-2-carboxamide
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-3-(4H-1,2,4-triazol-4-yl)benzamide
9-methyl-3-[2-(morpholin-4-yl)pyrimidine-5-carbonyl]-3,9-diazaspiro[5.6]dodecane
6-(methylsulfanyl)-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1,2,3,4-tetrahydroisoquinoline
2,5-dimethyl-3-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]pyrazine
N-{[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}-2-[(prop-2-en-1-yl)amino]benzamide