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4-ethyl-3-({1-[2-(oxolan-2-ylmethoxy)acetyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl 3-(2-methoxyacetamido)-1-(3-methylbutyl)-5-{[1-(4-methylphenyl)propan-2-yl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[3-(2-chlorophenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methylacetamide
2-cyclopropyl-1-[(4-fluorophenyl)methyl]-6-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1,4-dihydropyridin-4-one
1-[2-methyl-2-(morpholin-4-yl)propyl]-4-(pyridin-3-yl)piperidin-4-ol
3-fluoro-N-[(2-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)pyridine-4-carboxamide
1-(2-methoxy-5-{[4-(methoxymethyl)piperidin-1-yl]methyl}phenoxy)-3-(piperidin-1-yl)propan-2-ol
2-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propane-1,3-diol
2-[2-(dimethylamino)ethyl]-9-[(2-fluoro-4-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(1-{1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
2-[2-(6-fluoro-1H-1,3-benzodiazol-2-yl)phenoxy]-1-(piperidin-1-yl)ethan-1-one
[4-(3-fluoro-4-phenylphenyl)pyridin-2-yl]methanol
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}acetamide
N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
1-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
4-benzyl-3-ethyl-1-[2-(propan-2-yl)pyrimidine-4-carbonyl]-1,4-diazepan-5-one
(2S,4S)-1-[(4-chlorophenyl)methyl]-4-{[(2,5-dimethylphenyl)methyl]amino}-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[2-(4-methyl-1,3-thiazol-2-yl)ethyl]acetamide
1-cyclopentyl-4-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-1,4-diazepane
7-(cyclobutylmethyl)-2-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-2,7-diazaspiro[4.5]decane
1-ethyl-N-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-5-methyl-1H-pyrazole-4-carboxamide
5-[2-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1H-indole
3-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
2-(2-chlorophenyl)-4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridine
1-ethyl-8-(4-phenoxybutanoyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[1-(3-methylbutyl)-2,4-dioxo-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
4-{2-[(5,6-dimethylpyrimidin-4-yl)amino]-1-hydroxyethyl}benzene-1,2-diol
1-(benzyloxy)-8-[2-(cyclohex-1-en-1-yl)acetyl]-1,8-diazaspiro[4.5]decan-2-one
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-[3-(trimethyl-1H-pyrazol-1-yl)propanoyl]-1,4-diazepan-5-one
(1S,5R)-6-(2-methoxyethyl)-3-{2-[methyl(pyridin-2-ylmethyl)amino]acetyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[2-(3-methoxyphenyl)piperidin-1-yl]ethan-1-one
(4aS,8aR)-1-butyl-6-[3-(pyridin-3-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
5-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]pyrazin-2-ol
N-[2-(2-methyl-1H-indol-3-yl)ethyl]-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
2-(2-ethyl-1H-imidazol-1-yl)-1-[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]ethan-1-one
6-(2-chlorophenyl)-2-(4-{[(3R)-3-hydroxypyrrolidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
2-ethoxy-5-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]pyridine
(4aR,8aS)-6-[(2E)-3-(3,4-dimethoxyphenyl)prop-2-enoyl]-1-(2-methoxyethyl)-decahydro-1,6-naphthyridin-2-one
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-(pyrimidin-2-yl)pyrrolidin-3-yl]acetamide
2-fluoro-N-[4-(4-{[phenyl(pyridin-4-yl)methyl]amino}piperidin-1-yl)phenyl]benzamide
[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl](methyl)[(5-methylfuran-2-yl)methyl]amine
[(3,4-dimethoxyphenyl)methyl][(2,3,5-trimethyl-1H-indol-7-yl)methyl]amine
8-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
4-(1H-imidazol-2-yl)-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidine
2-{1-[2-methoxy-1-(3-methylphenyl)-2-oxoethyl]-1H-imidazol-2-yl}benzoic acid
2-{1-[(2-ethoxyphenyl)methyl]-4-(1-propylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
2-(1-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-3-yl)-1H-1,3-benzodiazole
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
(2-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-oxoethyl)urea
3-({3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridin-2-amine