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2-[3-(1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-1H-pyrazol-3-yl)phenyl]-1,3-thiazole
6-amino-1-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]hexan-1-one
N-cyclopropyl-4-methoxy-3-({1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidin-4-yl}oxy)benzamide
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-(2-methoxyethoxy)piperidine
2-methyl-6-{4-[3-(1,2-oxazol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1H-imidazol-1-yl}pyridine
N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-{8-methyl-3-oxo-2,8-diazaspiro[4.5]decan-2-yl}acetamide
1-cyclohexyl-4-(2,5-difluorobenzoyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
2-[3-(4-chlorophenyl)-5-[2-(1-methylpiperidin-3-yl)ethyl]-1H-1,2,4-triazol-1-yl]ethan-1-ol
N-{[2-(azepan-1-yl)-7-fluoroquinolin-3-yl]methyl}-2-(2,5-dimethoxyphenyl)-N-(2-methoxyethyl)acetamide
N-({4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)cyclohexanecarboxamide
2,6-dimethyl-N-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)pyridine-4-carboxamide
(3R,4R)-1-(4-ethyl-5-methylpyrimidin-2-yl)-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
2-(1-ethyl-1H-pyrazole-4-carbonyl)-N-(oxolan-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
N-(3,4-dimethoxyphenyl)-1-[5-(4-methoxyphenyl)furan-2-carbonyl]piperidin-3-amine
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]acetamide
2-amino-6-(1,3-dimethyl-1H-pyrazol-4-yl)-4-[2-(propylamino)pyrimidin-5-yl]pyridine-3-carbonitrile
7-(4-methylphenyl)-4-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[3-(1-phenylcyclopropyl)-5-[2-(1H-1,2,3,4-tetrazol-1-yl)ethyl]-1H-1,2,4-triazol-1-yl]acetic acid
6-[4-(4-methoxyphenyl)-2-methyl-5-oxopiperazine-1-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
3-[(2,3-difluoro-6-methoxyphenyl)methyl]-3,9-diazaspiro[5.6]dodecan-10-one
(2R,3R)-N-(furan-2-ylmethyl)-2-hydroxy-3-(pyrrolidin-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-carboxamide
5-butyl-4-[3-(methanesulfonylmethyl)piperidin-1-yl]-6-methylpyrimidin-2-amine
2,6,8-trimethyl-4-[4-(oxolan-2-ylmethyl)piperazine-1-carbonyl]quinoline
(4aR,8aR)-2-cyclopentanecarbonyl-7-(1,3-thiazol-5-ylmethyl)-decahydro-2,7-naphthyridin-4a-ol
2-(1-ethylpiperidin-4-yl)-1-(2-phenylazetidin-1-yl)ethan-1-one
4-chloro-N-methyl-3-({[(1-methyl-1H-imidazol-2-yl)methyl](propyl)carbamoyl}amino)benzamide
2-{2-oxa-7-azaspiro[4.5]decane-7-carbonyl}-4H-chromen-4-one
{4-[6-(benzyloxy)pyridin-3-yl]-3-(hydroxymethyl)phenyl}methanol
N-(4-butanamido-3-methoxyphenyl)-1,1-dioxo-1λ6-thiane-4-carboxamide
4-[3-(2-fluorophenyl)pyrrolidin-1-yl]-5-methylpyrimidin-2-amine
methyl 6-(3-methylpentanoyl)-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-methyl-5-[3-methyl-1-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1,3-thiazole
1-(oxan-4-ylmethyl)-4-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
N-[1-(methoxymethyl)cyclopropyl]-N,2-dimethyl-1,3-thiazole-4-carboxamide
N-methyl-3-(4-methyl-1,3-thiazol-5-yl)-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}propanamide
1-(azepan-1-yl)-3-[3-({[(3,4-dimethoxyphenyl)methyl](methyl)amino}methyl)phenoxy]propan-2-ol
4-[({1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}amino)methyl]-2,6-dimethylphenol
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-6-(methoxymethyl)pyrimidin-4-amine
4-{[5-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-methylpiperidine
3-[1-(6-methylpyridin-2-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]pyridin-2-ol
4-(1-{[3-(furan-2-yl)phenyl]methyl}azetidin-3-yl)morpholine
N,5-dimethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-amino-6-(2-methoxyphenyl)-4-[1-(propan-2-yl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
N-{[3-(2H-1,3-benzodioxol-5-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
4-[(5-chloro-2-hydroxyphenyl)methyl]-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-[1-(3-hydroxypropyl)-4-phenyl-1H-imidazol-5-yl]-2-methoxy-6-(prop-2-en-1-yl)phenol
N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}furan-2-carboxamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(1H-1,2,4-triazol-1-yl)benzamide
2,3-difluoro-5-(4-methyl-1H-pyrazol-1-yl)phenol
2-(3-hydroxyphenyl)-2-[methyl(1H-pyrazol-3-ylmethyl)amino]acetic acid