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3-(2H-1,3-benzodioxole-5-carbonyl)-1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperidine
methyl 3-(2,3-dihydro-1-benzofuran-5-ylmethyl)-9-[3-(1-methyl-1H-pyrazol-4-yl)propoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-[3-(2H-1,3-benzodioxol-5-ylmethyl)-1,2-oxazole-5-carbonyl]thiomorpholine
N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-2,3-dihydro-1,4-benzodioxine-2-carboxamide
methyl(2-methylprop-2-en-1-yl){[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl}amine
4-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-1-[(3,5-dimethylphenyl)methyl]piperazin-2-one
N-[2-(dimethylamino)ethyl]-3-(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)propanamide
4-{[1-(furan-3-carbonyl)piperidin-4-yl]methyl}morpholine
4-{[(3aS,6aS)-5-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-octahydropyrrolo[3,4-b]pyrrol-1-yl]methyl}pyridine
N-(5-chloro-2-methoxyphenyl)-4-(hydroxymethyl)-4-(oxan-2-ylmethyl)piperidine-1-carboxamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1-methylcyclopropane-1-carboxamide
N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}-1-benzofuran-2-sulfonamide
[(5-chloro-2-methoxyphenyl)methyl](ethyl)(pyridin-2-ylmethyl)amine
N-{[1-(2-methylphenyl)pyrrolidin-3-yl]methyl}-2-(pyridin-4-yl)pyrimidine-5-carboxamide
1-[(4-fluorophenyl)methyl]-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-methyl-3-{2-[(4-methylphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[1-(thiophen-2-yl)ethyl]propanamide
1-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperidin-4-ol
2-{1-[(6-methylpyridin-2-yl)methyl]-4-(2-methylquinolin-4-yl)piperazin-2-yl}ethan-1-ol
N-(2,4-dimethylphenyl)-N'-(2-methoxyethyl)-N'-[(2-methylphenyl)methyl]propanediamide
ethyl({[2-(prop-2-en-1-yloxy)phenyl]methyl})(1,3-thiazol-2-ylmethyl)amine
methyl 2-{[5-(2-methylphenyl)-1,2,4-triazin-3-yl]amino}-4-(methylsulfanyl)butanoate
{[(1R,5S,6R)-3-(dimethyl-1,2-oxazole-4-carbonyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl}[(1-ethyl-1H-imidazol-2-yl)methyl]methylamine
3-[2-(3-ethoxy-4-hydroxyphenyl)-1H-imidazol-1-yl]-4-methylbenzamide
(1S,3R)-3-amino-N-(2-{[(3-chlorophenyl)methyl]sulfanyl}ethyl)cyclopentane-1-carboxamide
1-[5-(2,5-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]-2-(methoxymethyl)piperidine
2-(4-fluoro-3-methylphenyl)-2-(4-{[(propan-2-yl)carbamoyl]methyl}piperazin-1-yl)acetic acid
N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2-(2,3,6-trimethylphenoxy)acetamide
5-(2-methoxy-4-methylphenoxymethyl)-N-methyl-N-(pyridin-3-ylmethyl)-1,2-oxazole-3-carboxamide
(2E)-3-(1H-imidazol-4-yl)-1-{7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}prop-2-en-1-one
8-(oxan-4-yl)-3-{2-[4-(propan-2-yl)piperazin-1-yl]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-(ethylamino)pyrimidine-5-carboxamide
methyl (2S,4S)-4-[2-chloro-5-(trifluoromethyl)benzamido]-1-[(2,4-dimethoxyphenyl)methyl]pyrrolidine-2-carboxylate
N-benzyl-N-methyl-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
5-[6-amino-5-cyano-4-(4-hydroxyphenyl)pyridin-2-yl]thiophene-3-carboxylic acid
N-[(2,4-dimethoxyphenyl)methyl]-3-(1-{imidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-yl)propanamide
1-(4,7-dimethylquinazolin-2-yl)-N-[1-(thiophen-2-yl)propan-2-yl]azepan-4-amine
(3-benzyl-1-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}piperidin-3-yl)methanol
3-(2-methoxy-3-methylbenzoyl)-3,9-diazaspiro[5.5]undecane
3-[5-(dimethyl-1,2-oxazol-4-yl)-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl]pyridine
(2S)-3-methyl-2-[2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamido]butanamide
N-benzyl({5H,6H,7H-cyclopenta[b]pyridin-7-yl}amino)sulfonamide
2-(methylsulfanyl)-N-[(1R,3S)-3-[(thiophen-2-ylmethyl)carbamoyl]cyclopentyl]pyridine-3-carboxamide
4-[(3-fluorophenyl)methyl]-3-oxo-N-(1,3,4-thiadiazol-2-yl)piperazine-1-carboxamide
1-[(2-chlorophenyl)methyl]-N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
8-(cyclohex-3-en-1-ylmethyl)-3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]methyl}-2-phenyl-2H-1,2,3-triazole
propan-2-yl 4-chloro-3-[2-(5-oxopyrrolidin-2-yl)acetamido]benzoate
8-(5-fluoro-2-methylbenzoyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decane
4-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
2-[4-(2H-1,3-benzodioxol-5-yl)-3,5-dimethyl-1H-pyrazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide