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(4aR,7aS)-1-benzyl-4-[(1-methyl-1H-imidazol-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[1-(4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzoyl)piperidin-3-yl]propan-1-one
2-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane
N-[1-(3-methylpyridin-2-yl)propan-2-yl]-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
4-{[1-(3,4-diethoxybenzoyl)piperidin-4-yl]methyl}morpholine
N-[2-methyl-3-(pyrrolidin-1-yl)phenyl]-4-(pyrimidin-2-yl)-1,4-diazepane-1-carboxamide
1-[(4-methoxyphenyl)methyl]-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-(4-fluorophenyl)-N-methyl-4-oxobutanamide
3-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-(2-hydroxypropyl)propanamide
4-[(dimethylamino)methyl]-1-(5-phenyl-1,2,4-oxadiazol-3-yl)azepan-4-ol
N-benzyl-6-oxo-N-(1,3-thiazol-2-ylmethyl)-1,6-dihydropyridine-2-carboxamide
N-(4-chloro-3-methylphenyl)-2-{[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]amino}acetamide
6-[2-(3-methoxyphenyl)piperidine-1-carbonyl]-2-methyl-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
3-({5-[1-(4-fluorophenyl)-1H-imidazol-2-yl]furan-2-yl}sulfanyl)-4-methyl-4H-1,2,4-triazole
(benzylsulfamoyl)[2-(4-phenylpyrimidin-2-yl)ethyl]amine
N-[2-(dimethylamino)ethyl]-1-(1-{[4-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide
4-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-2-methylphenol
N-ethyl-2-[1-(2-hydroxyethyl)-1H-pyrazol-4-yl]-7,8-dimethyl-N-(propan-2-yl)quinoline-4-carboxamide
1-[2-(dimethylamino)ethyl]-3-(2-methylphenyl)-3-[2-oxo-2-(piperidin-1-yl)ethyl]pyrrolidine-2,5-dione
2-(4-fluoro-2-methylphenyl)-1-[3-(3-methoxypropyl)piperidin-1-yl]ethan-1-one
2-(2-acetamidoethyl)-N-[4-fluoro-3-(trifluoromethyl)phenyl]piperidine-1-carboxamide
{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}(4-phenylbutan-2-yl)amine
5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)-1-[(4-phenyl-1,3-thiazol-2-yl)methyl]pyrrolidin-2-one
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-4-carboxamide
methyl(oxan-4-ylmethyl){[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}amine
1,3-dimethyl-N-[1-(6-methylpyridin-2-yl)propan-2-yl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[3-ethyl-4-(propan-2-yl)piperazin-1-yl]-4-(1H-imidazol-1-yl)butan-1-one
2-{1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidin-2-yl}pyridine
1-(4-tert-butylbenzoyl)-4-[(3-chlorophenyl)methyl]-1,4-diazepan-5-one
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(5-methylpyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-1-[1-(2-methoxyethyl)-2-methyl-1H-indol-5-yl]urea
ethyl({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)[(4-methoxyphenyl)methyl]amine
3-(3-chloro-1,2-oxazol-5-yl)-N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]propanamide
2-cyclopropyl-N-methyl-6-oxo-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1,6-dihydropyrimidine-5-carboxamide
6-methyl-2-[(2-{[1-(9H-purin-6-yl)piperidin-4-yl]amino}ethyl)amino]-3,4-dihydropyrimidin-4-one
N-[(3-chlorophenyl)methyl]-1,3-dimethyl-N-(2-methylpropyl)-1H-pyrazole-4-carboxamide
N-{2-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}oxolane-2-carboxamide
6-ethyl-N,2-dimethyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]quinoline-4-carboxamide
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1-(furan-2-ylmethyl)piperidine-3-carboxamide
1-(2H-1,3-benzodioxol-4-ylmethyl)-3-(pyrrolidin-1-yl)piperidine
1-(propan-2-yl)-2-{[4-(pyridin-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-1,3-benzodiazole
(3S,4R)-1-(2,1,3-benzoxadiazol-4-ylmethyl)-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-5-ethoxy-2-methyl-1-benzofuran-3-carboxamide
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-2-ethylpyrimidine-5-carboxamide
2-[3-(oxolan-3-yl)-5-[3-(pyridin-2-yl)-1H-pyrazol-5-yl]-1H-1,2,4-triazol-1-yl]acetic acid
2-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1-[1-(thiophen-2-yl)ethyl]-1H-imidazole
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-3-(2-methylphenyl)propan-1-one
(3R,4S)-4-cyclopropyl-1-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]pyrrolidin-3-amine
2-[1-(2,2-dimethylpropyl)-4-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperazin-2-yl]ethan-1-ol
4-methyl-5-{1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1,2,3-thiadiazole