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N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-1,2-oxazole-3-carboxamide
3-(6-fluoropyridin-3-yl)-1-{[4-(pyrrolidin-1-ylmethyl)phenyl]methyl}urea
3-acetamido-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)benzamide
6-[3-(2-methoxyphenoxy)propyl]-1H-indazole
(2S,4R)-4-amino-N-methyl-1-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}pyrrolidine-2-carboxamide
(4aS,8aR)-6-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-decahydro-1,6-naphthyridine-4a-carboxylic acid
6-(2-methyl-1,4-oxazepan-4-yl)-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
3-propoxy-N-[3-(sulfamoylmethyl)phenyl]piperidine-1-carboxamide
2-[4-({imidazo[1,2-a]pyrimidin-2-ylmethyl}amino)-6-methylpyrimidin-2-yl]phenol
5-[(3-hydroxy-2,2-dimethylpropyl)amino]-1-methyl-N-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-methyl-6-{4-[2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}pyrimidine
methyl 5-[5-(oxolan-2-yl)thiophene-2-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
(2R)-2-amino-N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-4-methylpentanamide
1-[2-(pyridin-2-yl)pyrrolidin-1-yl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenoxy]ethan-1-one
2-(2-hydroxyphenyl)-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]acetamide
2-{[2-(1H-pyrazol-1-yl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
[1-(3-fluorophenyl)propan-2-yl][(2-methyl-1,3-thiazol-4-yl)methyl]amine
3-[(3S,4R)-1-[(2,3-dimethoxyphenyl)methyl]-4-(dimethylamino)piperidin-3-yl]-N-[2-(2-methoxyphenyl)ethyl]propanamide
(3R,4R)-1-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
6-fluoro-4-(pyridin-3-ylmethyl)-3,4-dihydro-2H-1,4-benzoxazin-3-one
2-{4-[(2-methyl-1,3-thiazol-5-yl)methyl]-1-(thiophen-3-ylmethyl)piperazin-2-yl}ethan-1-ol
2-[(3R,4S)-3-[(2-methylpyrimidin-4-yl)amino]-4-propylpyrrolidin-1-yl]-1-(morpholin-4-yl)ethan-1-one
1-[7-(4-hydroxy-1-methylpiperidin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(3-methoxyphenyl)ethan-1-one
5-(1-benzothiophen-2-ylmethyl)-N-[(1-ethylpyrrolidin-2-yl)methyl]-1-(2-methoxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-cyclopentyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]-N-{[6-(thiophen-2-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}acetamide
4-(pyridin-3-yl)-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrimidin-2-amine
3-(5-tert-butyl-1,3,4-thiadiazol-2-yl)-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}urea
3-{[4-(4-aminopyrimidin-2-yl)-6-hydroxy-1,4-diazepan-1-yl]methyl}benzoic acid
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-(pyridin-4-ylmethoxy)-4-(thiophene-3-carbonyl)-1,4-diazepan-2-one
N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-2-(pyridin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-1,4-dithiepan-6-amine
N-[(1S,2R)-2-[(1-ethylpiperidin-4-yl)amino]cyclobutyl]-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanamide
4-[4-({4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}methyl)piperazin-1-yl]phenol
1-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-2-[2-(thiophen-2-yl)ethyl]piperidine
2-(3-fluorophenoxymethyl)-N-[2-(1H-pyrazol-1-yl)ethyl]-1,3-oxazole-4-carboxamide
1-[(2-chloro-4-fluorophenyl)methyl]-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
4-[({[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}amino)methyl]-1-ethylpyrrolidin-2-one
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-(1H-indazole-3-carbonyl)pyrrolidin-3-yl]methanol
2-[4-(1,4-diazepan-1-ylmethyl)phenyl]-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
3-{[1-(4-methylphenyl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
6-[2-(3,4-dichlorophenyl)morpholin-4-yl]-N-ethylpyridine-3-carboxamide
9-[4-(difluoromethoxy)benzoyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
ethyl[({1-[(2-fluorophenyl)methyl]pyrrolidin-3-yl}methyl)sulfamoyl]methylamine
1-butyl-4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidine
2-methyl-6-(1H-pyrazol-4-yl)quinolin-4-ol
N-methyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
methyl({3-methyl-1-[4-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl}methyl)amine
N-methyl-N-[2-(oxan-4-yl)ethyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
methyl 5-[(4-hydroxy-4-methylpentan-2-yl)amino]-3-(oxolane-3-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate