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6-methoxy-N-methyl-N-[2-(pyridin-4-yl)ethyl]pyrimidin-4-amine
2-(4-methoxypiperidin-1-yl)-5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridine
N-[1-(3-chlorophenyl)cyclopropyl]-3-ethyl-4-methyl-1H-pyrazole-5-carboxamide
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-1-methylazepane-2-carboxamide
N,N-dimethyl-2-[4-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazin-1-yl]acetamide
N-{2-[(2,8-dimethylquinolin-4-yl)formamido]ethyl}pyridine-3-carboxamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
methyl (2S,4R)-4-hydroxy-1-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}pyrrolidine-2-carboxylate
N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]imidazo[1,2-a]pyrimidine-2-carboxamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-4-(furan-2-yl)-N-methylbenzamide
(3S,9aR)-8-[(3,4-difluorophenyl)methyl]-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
6-(3,3-diphenylpiperidine-1-carbonyl)-2-methyl-2,3-dihydropyridazin-3-one
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-1-aminocyclopropane-1-carboxamide
{[5-(methoxymethyl)furan-2-yl]methyl}({[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]methylamine
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
9-(5-ethyl-2-methylpyrimidin-4-yl)-3-oxa-9-azaspiro[5.5]undecane
8-[(2,5-difluorophenyl)methyl]-1-(2-methoxyethyl)-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N,8-dimethyl-3-{[(2S)-4-methyl-2-(propan-2-yl)piperazin-1-yl]methyl}-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
3-(2-methyl-1H-imidazol-1-yl)-1-[3-(4-phenylbenzoyl)piperidin-1-yl]propan-1-one
{4-[5-(5-ethyl-1,3-oxazol-4-yl)-1,2,4-oxadiazol-3-yl]phenyl}methanol
ethyl (1R,5S,6R)-3-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-3-azabicyclo[3.1.0]hexane-6-carboxylate
4-[2-(3-phenylpyrrolidin-1-yl)ethyl]-1,4-oxazepane
2-{[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino}-N-(2-methylphenyl)acetamide
1-{2-[2-(3-methoxyphenyl)piperidin-1-yl]-2-oxoethyl}piperidine-4-carboxamide
4,4,4-trifluoro-1-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]butan-1-one
6-[3-(4-ethoxyphenyl)propyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
3-({1-[3-(trifluoromethyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)-1H-pyrazole
(3aR,5S,6S,7aS)-2-{3-methyl-3H-imidazo[4,5-b]pyridine-6-carbonyl}-octahydro-1H-isoindole-5,6-diol
1-[1-(1-cycloheptylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
2-(2-{1-[3-(2-methylpyrimidin-4-yl)phenyl]-1H-imidazol-2-yl}phenoxy)ethan-1-ol
1-[(2,3-difluorophenyl)methyl]-5-[2-(ethylamino)ethyl]pyrrolidin-2-one
4-methyl-3-[3-(2-methylphenoxy)azetidine-1-carbonyl]benzene-1-sulfonamide
N-(1H-indol-3-yl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(2S,4S)-4-amino-N-ethyl-1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]pyrrolidine-2-carboxamide
2-(2-fluorophenyl)-N-{2-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}acetamide
ethyl 1-(2,3-dihydroxypropyl)-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
N-[(6-methylpyridin-2-yl)methyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-[methyl(pyridin-4-ylmethyl)amino]-1-[3-(2-methylphenyl)piperidin-1-yl]ethan-1-one
1-{2-[7-(2-methoxyphenyl)-4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-2-yl]ethyl}-6-methyl-1,2-dihydropyridin-2-one
2-(4,5-dichloro-2-methyl-1H-imidazol-1-yl)-N-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]acetamide
methyl N-(1-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-1-oxopropan-2-yl)carbamate
{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(4-methyl-1,3-thiazol-2-yl)ethyl]amine
1-(4-methoxy-3-propanamidophenyl)-5-oxopyrrolidine-3-carboxylic acid
4-{[(3R,4S)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]methyl}benzoic acid
2-{[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]methyl}pyridine
2-{4-[(3-methyl-1H-indol-2-yl)methyl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
5-cyclopropanecarbonyl-1'-[(2S)-1-methylpyrrolidine-2-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
methyl 3-acetamido-1-(3-methylbutyl)-5-[(2-methylbutyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate