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N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-4-hydroxy-3-methoxybenzamide
N-(2-{7-[(4-hydroxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclohexanecarboxamide
8-[4-(4-fluorophenyl)butanoyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-{3-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-(5-methylhexan-2-yl)-1H-pyrazole-3-carboxamide
6-methoxy-N4-methyl-N4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]pyrimidine-2,4-diamine
N-[2-(azepan-1-yl)-2-phenylethyl]-2-methyl-1,3-thiazole-4-carboxamide
(1R,2R,6S,7S)-4-[(1-phenyl-1H-pyrazol-5-yl)methyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane
N-[(3-chlorophenyl)methyl]-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-benzyl-4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
1-[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
3-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-1-(2-methylpropyl)-1-(pyridin-2-ylmethyl)urea
2-butyl-5-chloro-4-{1-[2-(1H-imidazol-1-yl)ethyl]-1H-imidazol-2-yl}-1H-imidazole
1-methyl-3-phenyl-8-[(1s,4s)-4-hydroxycyclohexanecarbonyl]-1,8-diazaspiro[4.5]decan-2-one
1-(isoquinoline-5-carbonyl)spiro[azepane-4,2'-chromene]
2-methyl-3-{[3-(oxolan-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-indole
ethyl 5-({[5-(tert-butylcarbamoyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridin-3-yl]formamido}methyl)furan-2-carboxylate
2-chloro-N-[2-({[1-(propan-2-yl)-1H-pyrazol-5-yl]carbamoyl}amino)ethyl]benzamide
3-{2-[4-hydroxy-4-(pyridin-2-yl)piperidin-1-yl]-2-oxoethyl}-4-[(2-methoxyphenyl)methyl]piperazin-2-one
2-[5-(4-cyano-1-methyl-1H-pyrrol-2-yl)-1-(2,3-dihydro-1H-inden-4-yl)-1H-1,2,4-triazol-3-yl]acetamide
2-cyclopentyl-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)acetamide
1-{2-[(3-fluorophenyl)methyl]morpholin-4-yl}-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
N-cyclopropyl-6-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyridazin-3-amine
1-[6-(3-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-4-phenyl-1,2,3,6-tetrahydropyridine
N-(2-ethylphenyl)-3-[2-(4-ethylpiperazin-1-yl)acetamido]benzamide
1-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-3-[1-(4-methoxyphenyl)-3-methyl-1H-pyrazol-5-yl]-1-methylurea
N-{1-[(3-chlorophenyl)methyl]-1H-pyrazol-5-yl}-3-ethoxypropanamide
ethyl 4-{6-[(1-methyl-1H-indol-3-yl)methyl]-6-azaspiro[2.5]octane-1-carbonyl}piperazine-1-carboxylate
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(5-methyl-1,3-oxazole-4-carbonyl)piperidin-3-ol
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-cyclopropanecarbonylpyrrolidine-2-carboxamide
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl][2-(2-fluorophenyl)-1-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-4-yl}ethyl]methylamine
(3R,4S)-4-cyclopropyl-N,N-dimethyl-1-[(1-propyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-amine
5-{5-[1-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1,2,4-oxadiazol-3-yl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
3-(2-fluorophenyl)-5-phenylmethanesulfonyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
2-amino-6-(3-fluoro-4-methoxyphenyl)-4-(3-hydroxyphenyl)pyridine-3-carbonitrile
N,N-diethyl-4-(1H-pyrazol-3-yl)aniline
2-{[1-(pyrrolidin-1-yl)hex-5-en-2-yl]oxy}-5-(trifluoromethyl)pyridine
1-({[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)cyclohexan-1-ol
4-[(2,4-difluorophenyl)methyl]-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
ethyl 4-[(4-methoxyphenyl)methyl]-1-(2-methyl-1,3-thiazole-4-carbonyl)piperidine-4-carboxylate
4-[4-(1,2-oxazole-3-carbonyl)piperazin-1-yl]-2-(trifluoromethyl)quinoline
(3S,5S)-1-[(3-chlorophenyl)methyl]-N-cyclooctyl-5-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)pyrrolidin-3-amine
1-[(3S,4R)-1-(1-benzofuran-5-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
4-cyclopentyl-N-(3-fluoro-4-methylphenyl)-3-oxopiperazine-1-carboxamide
1-[(4aR,8aR)-7-[(3,4-difluorophenyl)methyl]-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
2-{1-[2-(2-hydroxyethoxy)ethyl]-4-phenyl-1H-imidazol-5-yl}quinolin-4-ol
N,1,3-trimethyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-(2H-1,3-benzodioxol-5-yl)-3-{[4-(propan-2-yl)phenyl]amino}piperidine-1-carboxamide
(3aS,6aS)-2-[(3-methyl-1,2-oxazol-5-yl)methyl]-5-[2-(thiophen-3-yl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid