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1-(azepan-1-yl)-3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]propan-1-one
(1R,3S,5S)-8-[6-(aminomethyl)-2-methylpyrimidin-4-yl]-8-azabicyclo[3.2.1]octan-3-ol
N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]-4-oxopentanamide
N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-2,3,4-trimethoxy-N-(oxolan-2-ylmethyl)benzamide
5-{5-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazol-4-yl]-1,2,4-oxadiazol-3-yl}-1H-1,3-benzodiazole
11-{[(2,3-difluorophenyl)methyl]amino}-4-(pyridin-4-ylmethyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-{4-[4-(pyrazin-2-yl)piperazin-1-yl]piperidin-1-yl}-1,3-benzothiazole
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
3-methoxy-1-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
5-[(2-chlorophenyl)methyl]-3-cyclopentyl-5-(piperidin-4-yl)imidazolidine-2,4-dione
N-[2-(4-{[2-(pyridin-3-yl)piperidin-1-yl]methyl}phenoxy)ethyl]-2H-1,3-benzodioxole-5-carboxamide
(2S,4S)-N-[(1R)-1-(4-methoxyphenyl)ethyl]-1-methyl-4-(3-methylbenzamido)pyrrolidine-2-carboxamide
N-benzyl-N-methyl-1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperidin-3-amine
(2E)-N-({7-[(3,5-dimethoxyphenyl)methyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-(2-fluorophenyl)prop-2-enamide
4-methyl-N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}-1,2,5-oxadiazole-3-carboxamide
ethyl 1-{3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}piperidine-4-carboxylate
(2E)-N-[1-(3-phenylpropyl)piperidin-3-yl]-3-(pyridin-4-yl)prop-2-enamide
N,N-dimethyl-2-[(1S,5R)-6-[2-(2-methylphenoxy)acetyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
4-[5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-1-methyl-2-phenylpiperazine
2-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propanoic acid
N-methyl-N-[(3-methyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-methyl-3-(1H-pyrazol-1-ylmethyl)-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-[3-(methylsulfanyl)propyl]piperidin-3-ol
1-benzyl-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-1H-pyrazole-4-carboxamide
(2S,4R)-4-amino-1-(2-amino-5,6,7,8-tetrahydroquinazoline-4-carbonyl)-N,N-diethylpyrrolidine-2-carboxamide
(1R,5R)-6-(cyclobutylmethyl)-3-(1-methyl-1H-indole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(1S,5R)-6-(5-cyclopropyl-3-methyl-1H-pyrazole-4-carbonyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-(2-ethoxyethyl)-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N-[(1-benzylpiperidin-4-yl)methyl]-4-chloro-N,1,5-trimethyl-1H-pyrazole-3-carboxamide
(3aS,6aS)-2-cyclobutanecarbonyl-5-(1,3-thiazol-4-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
methyl 7-oxo-3-[5-oxo-1-(propan-2-yl)pyrrolidine-3-carbonyl]-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[(2S)-2-aminobutanoyl]-4-(4-fluoro-2-methylphenoxy)piperidine-4-carboxylic acid
6-(3-chloro-5-fluorophenyl)pyridine-2-carboxamide
N-[(2-methylphenyl)methyl]-2-[2-(morpholin-4-ylmethyl)piperidin-1-yl]acetamide
5-[(isoquinolin-5-yloxy)methyl]-N-methyl-N-[2-(piperidin-1-yl)ethyl]-1,2-oxazole-3-carboxamide
2-(6-hydroxy-1,4-oxazepane-4-carbonyl)benzonitrile
(2R,3S,6R)-3-(4-methylphenyl)-5-(trimethyl-1H-pyrazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-tert-butyl-N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-1,3,4-oxadiazol-2-amine
3-(3-amino-5-fluoro-1H-indazol-1-yl)-5-(pyrrolidine-1-sulfonyl)benzoic acid
N-cyclopropyl-3-{5-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
1-[2-butyl-5-oxo-4-(3-phenylphenyl)piperazin-1-yl]propane-1,2-dione
1-{1-[2-(dimethylamino)benzoyl]piperidin-3-yl}-2-phenylethan-1-one
N-{1-[4-(3-chlorophenyl)-5-[(cyclohexylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}cyclobutanecarboxamide
(3aR,6aS)-5-{[7-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
2-(3-tert-butyl-1H-pyrazol-5-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2,5-dimethyl-3-(4-{[5-(oxan-2-yl)thiophen-2-yl]methyl}piperazin-1-yl)pyrazine
(2S)-N-{[5-chloro-7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-acetamido-4-(methylsulfanyl)butanamide
(1S,5R)-6-(benzenesulfonyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
[(3R,5R)-1-[4-(methylamino)pyrimidin-2-yl]-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
4-benzyl-1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-1,4-diazepan-5-one