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1-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
3-(2-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-4-(3-fluorobenzenesulfonyl)-9-(oxolan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
methyl 3-[(3S,4R)-1-[(2-ethoxyphenyl)methyl]-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanoate
5-(2-methoxyphenoxymethyl)-N-methyl-N-(oxan-4-yl)-1H-pyrazole-3-carboxamide
(3S,7S)-5-(3,4-difluorobenzoyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
4-[4-(3-methoxyphenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]-1-[(4-methoxyphenyl)methyl]piperidine
2-(1-{[1-(5-ethylthiophene-2-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
2-methyl-7-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
4-[4-(1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]-1-(3-methylphenyl)pyrrolidin-2-one
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-1-ethyl-3-methylpiperidine-3-carboxamide
3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-(4-ethoxy-2-fluorophenyl)-3-methylurea
5-cyclopropyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-1H-pyrazole-4-carboxamide
N-(1-methoxypropan-2-yl)-6-methyl-2-[(2-methylphenyl)methyl]-4-oxo-1-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
1-[4-(3-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxy)piperidin-1-yl]-2-(thiophen-2-yl)ethan-1-one
N-benzyl-N-methyl-1-(pyridin-4-ylmethyl)piperidin-3-amine
2-[1-(1-methylpiperidin-4-yl)-4-[(4-phenylphenyl)methyl]piperazin-2-yl]ethan-1-ol
3-[(4-fluorophenyl)formamido]-N-(1H-indol-4-ylmethyl)propanamide
4-ethyl-3-(1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{[3-(aminomethyl)pyrrolidin-1-yl]methyl}-N-methyl-N-phenylaniline
1-methyl-3-(2-methylpropyl)-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,4R)-1-[(4-hydroxy-3,5-dimethoxyphenyl)methyl]-4-(3-methylthiophen-2-yl)piperidin-3-ol
[(3R,4R)-1-{imidazo[1,2-a]pyridine-2-carbonyl}-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
4-amino-1-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]butan-1-one
(1S,5R)-6-[4-(1H-imidazol-1-yl)benzoyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
({1-[1-(1,4-dithiepan-6-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)urea
(2S)-2-{4-[2-(furan-2-yl)pyrimidin-5-yl]-1H-1,2,3-triazol-1-yl}-4-methylpentan-1-ol
N-[2-(azepan-1-yl)-2-phenylethyl]-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-[(1-methylpiperidin-3-yl)methyl]-2-oxo-2,3-dihydro-1,3-benzothiazole-6-sulfonamide
2-(3-methylfuran-2-carbonyl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-6-one
1-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-N,N-dimethylpyrrolidin-3-amine
{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}(ethyl)(2-methylprop-2-en-1-yl)amine
1-[(4-ethylphenyl)methyl]-5-{5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-yl}-1H-1,2,4-triazole
(2R,3S,6R)-3-(3-methoxyphenyl)-5-(2-methoxypyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(4-benzoylpiperazin-1-yl)-3-(3-methoxy-4-methylphenyl)propan-1-one
N-cyclopropyl-2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-[(3-hydroxyphenyl)methyl]acetamide
3-ethyl-5-{2-[2-(4-methoxynaphthalen-1-yl)-1H-imidazol-1-yl]ethyl}-1,2,4-oxadiazole
6-methyl-2-{[(oxan-3-ylmethyl)amino]methyl}quinolin-4-ol
1-methyl-N-[(5-methylpyrazin-2-yl)methyl]-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
1-ethyl-N,N-bis(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-[5-(furan-2-yl)-1,3,4-thiadiazol-2-yl]-1-[(4-methoxyphenyl)methyl]urea
2-[(4-{imidazo[1,2-b]pyridazin-6-yl}piperazin-1-yl)methyl]benzoic acid
1-[3-(2-chlorophenyl)-3-phenylpropanoyl]piperidine-4-carboxamide
N-{[6-(dimethylamino)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-N-(oxolan-2-ylmethyl)-4-(trifluoromethyl)benzamide
(4aR,7aS)-1-[4-(4-chlorophenyl)butanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(4-methyl-4H-1,2,4-triazol-3-yl)-N-[(3-phenylphenyl)methyl]propanamide
5-chloro-4-{[4-(2,2-dimethylpropyl)-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-2-methoxyphenol
(2S,4S,5R)-4-[ethyl(methyl)carbamoyl]-1-methyl-2-(2-methylpropyl)-5-(pyridin-3-yl)pyrrolidine-2-carboxylic acid
3-{[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]sulfonyl}pyridine
2-[4-(2-methylpyridin-4-yl)piperazin-1-yl]pyridine-4-carboxamide