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2-[3-(5-methylfuran-2-yl)-5-[1-(1H-pyrazol-1-yl)propan-2-yl]-1H-1,2,4-triazol-1-yl]pyridine
N-[(7R,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetamide
1-(carbamoylmethyl)-N-methyl-N-[1-(pyridin-3-yl)propyl]piperidine-4-carboxamide
[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)(1,3-thiazol-2-ylmethyl)amine
3-phenyl-N-{4-[4-({[3-(1H-pyrazol-1-yl)phenyl]methyl}amino)piperidin-1-yl]phenyl}propanamide
2-[4-(3,5-dimethylphenyl)-3-oxopiperazin-1-yl]pyridine-4-carboxamide
methyl 3-({2-ethyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}methyl)-4-methoxybenzoate
3-[1-(3-cyclohexylpropanoyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
ethyl 4-{[(1-methyl-1H-indazol-5-yl)carbamoyl]amino}piperidine-1-carboxylate
2-[4-(4-ethylpiperazine-1-carbonyl)-5-methyl-1H-pyrazol-1-yl]-4-(2-fluorophenyl)pyrimidine
1-{[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]amino}-3-(pyrrolidin-1-yl)propan-2-ol
2-{1-[(7-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperidin-4-yl}acetamide
(3S,4R)-3-ethyl-4-methyl-1-(pyrazine-2-carbonyl)piperidin-4-ol
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}propan-1-one
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-2-(1H-pyrazol-1-yl)butanamide
2-(1-benzofuran-5-carbonyl)-7-(3-methoxypropyl)-2,7-diazaspiro[4.5]decan-6-one
1-benzoyl-4-(2H-1,3-benzodioxol-4-ylmethyl)piperazine
(1S,5R)-6-(2-methoxyethyl)-3-[6-(4H-1,2,4-triazol-4-yl)pyridine-2-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-cyclopentyl-4-[(3-methyl-1,2-oxazol-5-yl)methyl]-1,4-diazepan-6-ol
2-[3-(2-ethylphenoxy)azetidine-1-carbonyl]thiophen-3-amine
3-(cyclopentylmethyl)-5-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
3-{1-[2-(2,2-difluoro-2H-1,3-benzodioxol-4-yl)-1H-imidazol-1-yl]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[2-(propylsulfanyl)phenyl]urea
2-[4-(3-acetamidophenyl)-3,5-dimethyl-1H-pyrazol-1-yl]acetic acid
4-(1-tert-butyl-3-methyl-1H-1,2,4-triazol-5-yl)-1-methylimidazolidin-2-one
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}propan-1-one
3-(azepane-1-sulfonyl)-5-(3-fluoropyridin-4-yl)benzoic acid
N-methyl-4-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-2-amine
N-[(1-ethylpyrrolidin-2-yl)methyl]-1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-4-amine
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carboxamide
N-butyl-N-(furan-2-ylmethyl)-4-oxo-1H,4H-benzo[h]quinoline-3-carboxamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-{imidazo[1,2-a]pyridin-3-ylmethyl}-5-methylpiperidin-2-one
3-(oxolan-3-yl)-5-(3-phenyl-1,2-oxazol-5-yl)-1,2,4-oxadiazole
N-[1-(cyclohexylmethyl)piperidin-3-yl]-4-(4-methylpiperazin-1-yl)benzamide
1-cyclopentyl-N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-6-oxopiperidine-3-carboxamide
8-[(2-ethylpyrimidin-5-yl)methyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
2-ethyl-N-[(7-fluoro-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-4-methyl-1,3-oxazole-5-carboxamide
{1-[1-(pyridin-3-ylmethyl)piperidin-3-yl]piperidin-4-yl}methanol
(oxolan-2-ylmethyl)({[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl})(thiophen-3-ylmethyl)amine
2-[(2-phenyl-1,3-thiazol-4-yl)methyl]-5-(piperazin-1-yl)-2,3-dihydropyridazin-3-one
4-(5-{2-[2-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)-1H-imidazol-1-yl]ethyl}-1H-1,2,4-triazol-3-yl)pyridine
4-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}-2,3-dihydro-1H-imidazol-2-one
4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]-1-(1H-pyrrole-2-carbonyl)piperidine
1'-(furan-3-carbonyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-[(2-fluoro-4-methoxyphenyl)methyl]-9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-(2-methyl-1,3-oxazol-4-yl)-1-(thiophen-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-(2-chlorophenyl)-1-cyclopentyl-3-{2-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
5-(3-phenylpropyl)pyridine-3-carboxamide
1-(1-cyclopentanecarbonylpiperidin-4-yl)-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
N-(furan-2-ylmethyl)-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-(prop-2-yn-1-yl)benzamide