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(1R,9aR)-1-{[methyl({[3-(1H-pyrazol-1-yl)phenyl]methyl})amino]methyl}-octahydro-1H-quinolizin-1-ol
1-{7-[(4-acetylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-4-(4-methoxyphenyl)butane-1,4-dione
N-(3-hydroxypropyl)-N-methyl-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
N-[3-(1H-indol-1-yl)propyl]-1H-1,2,3-triazole-5-carboxamide
4-(4-methyl-1H-pyrazol-1-yl)-1-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperidine-4-carboxylic acid
[(4aS,8aR)-6-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}-decahydro-1,6-naphthyridin-4a-yl]methanol
2-(dimethyl-1,2-oxazol-4-yl)-1-[3-(4-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxymethyl)piperidin-1-yl]ethan-1-one
3-(3,5-dimethylphenyl)-1-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]propan-1-one
3-(1H-1,2,3-benzotriazol-1-yl)-N-[2-(3,5-dimethylphenoxy)ethyl]-N-methylpropanamide
N-{2-[(2-butyl-6-methylpyrimidin-4-yl)amino]ethyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
3-(3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl)benzoic acid
2-chloro-N-methyl-5-[(E)-2-phenylethenyl]benzamide
7-{1-butyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}-3-methyl-3,4-dihydroquinazolin-4-one
dimethyl[(6-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridin-3-yl)methyl]amine
methyl 7-oxo-3-(3-phenylprop-2-ynoyl)-9-(thiophen-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-(2-methoxyethyl)-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-1,3-benzoxazole-6-carboxamide
N-[5-(2-methanesulfonamidopropanamido)-2-methoxyphenyl]pentanamide
1-[(2,3-dimethoxyphenyl)methyl]-3-{[(1-ethylcyclopropyl)amino]methyl}-3-hydroxypiperidin-2-one
methyl 2-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-1-oxo-1,2-dihydroisoquinoline-7-carboxylate
2-(4-fluorophenoxy)-N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]acetamide
N-tert-butyl-3-(4-phenylbenzoyl)piperidine-1-carboxamide
1-[3-(2-fluorophenyl)-1H-pyrazole-4-carbonyl]-N-methyl-N-(2-phenylethyl)piperidin-3-amine
1-methyl-2-[1-(1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
2-cyclohexyl-5-{[4-(1H-pyrazol-3-yl)piperidin-1-yl]methyl}pyrimidine
2,4,5-trimethyl-6-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
5-(5-{3-[(4-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)pyrimidine
2-[3-({methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)phenoxy]acetamide
1-(methoxymethyl)-N-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)cyclobutane-1-carboxamide
1-[3-(benzyloxy)phenyl]-3-[(4-hydroxy-1-methylpiperidin-4-yl)methyl]urea
2-[(2,4-dimethoxyphenyl)methyl]-9-oxa-2-azaspiro[5.5]undecane
(1R,5R)-3-cyclobutanecarbonyl-6-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-[2-(1-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethyl]acetamide
8-hydroxy-5,7-dimethyl-N-[(1-methylpyrrolidin-3-yl)methyl]quinoline-2-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-3-[5-oxo-2-(thiophen-3-ylmethyl)pyrrolidin-2-yl]propanamide
N-(propan-2-yl)-1-{1-[4-(1H-pyrazol-4-yl)butanoyl]piperidin-4-yl}piperidine-4-carboxamide
2-[4-(isoquinolin-1-yl)-1-[(3-methoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
N-[2-(5-chloro-2-methyl-1H-indol-3-yl)ethyl]-2-[(dimethylcarbamoyl)amino]acetamide
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
1-(2,3-dihydro-1H-inden-2-yl)-4-[(4-ethyl-5-methylpyrimidin-2-yl)amino]pyrrolidin-2-one
(3S,5R)-1-[(1-propyl-1H-imidazol-2-yl)methyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxylic acid
1-benzyl-N-(2-oxopyrrolidin-3-yl)-4-phenylpiperidine-4-carboxamide
8-(4-methyl-1,3-thiazole-5-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-3-(1H-pyrazol-1-yl)propan-1-one
3-(4-hydroxyphenyl)-N-{2-[(pyridin-3-yl)amino]ethyl}-1H-pyrazole-5-carboxamide
9-methoxy-3-[2-(morpholin-4-yl)propanoyl]-10-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
4-{2-[(6-methylpyridazin-3-yl)oxy]hex-5-en-1-yl}thiomorpholine
2-amino-6-(1-propyl-1H-1,2,3-benzotriazol-5-yl)-4-(pyridin-3-yl)pyridine-3-carbonitrile
1-(difluoromethyl)-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-5-carboxamide
(2S)-1-acetyl-N-{1-[(3-chlorophenyl)methyl]-1H-pyrazol-5-yl}pyrrolidine-2-carboxamide
1-(3-{3-[(4-fluorophenyl)amino]piperidin-1-yl}-3-oxopropyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one