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3-({1-[2-(cyclohex-1-en-1-yl)ethyl]-1H-1,2,3-triazol-4-yl}methyl)-2,3-dihydro-1,3-benzoxazol-2-one
1-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(propan-2-yloxy)ethan-1-one
1-{2-[3-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]-2-oxoethyl}-5,5-dimethylimidazolidine-2,4-dione
N-[4-(3-methylphenyl)phenyl]-1-[(2-propylpyrimidin-5-yl)methyl]piperidine-4-carboxamide
6-(propan-2-yloxy)-N4-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}pyrimidine-2,4-diamine
2-[(4-chlorophenyl)methyl]-8-(2-hydroxybenzoyl)-2,8-diazaspiro[4.5]decan-3-one
3-ethyl-1-(pyrrolidine-1-carbonyl)piperidine-3-carboxylic acid
2-(4-fluorophenyl)-2-hydroxy-1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
8-[(1-methyl-1H-imidazol-2-yl)methyl]-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
1-(1H-pyrrole-2-carbonyl)-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(2-methoxyphenyl)piperazine
3-(1H-pyrazol-4-yl)-N-(2-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
4-(2-chlorobenzenesulfonyl)-7-(2-methylphenyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(pyridin-4-yl)-7-(pyridine-2-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(3R,4R)-3,4-dimethyl-1-[4-(piperidine-1-carbonyl)pyridin-2-yl]pyrrolidin-3-ol
N-{2-methyl-2H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-2-[4-propyl-3-(pyridin-3-yl)-1H-pyrazol-1-yl]acetamide
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-[(3R,4S)-1-[(5-ethylpyridin-2-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
2-[3-(dimethylamino)pyrrolidin-1-yl]-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide
2-{4-[6-(methoxymethyl)pyrimidin-4-yl]piperazin-1-yl}-4-methyl-6-(trifluoromethyl)pyrimidine
N-[(1-hydroxycyclohexyl)methyl]-1-(4,6,7-trimethylquinazolin-2-yl)piperidine-4-carboxamide
N-(oxan-3-ylmethyl)-2-[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
7-chloro-2-methyl-4-(quinolin-5-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-{1-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-3-yl}-N-(4-methoxy-2-methylphenyl)propanamide
4-(2-methoxyacetyl)-1-[(4-methoxyphenyl)methyl]piperazin-2-one
5-(2-chlorophenyl)-1-methyl-1H,4H-pyrazolo[3,4-d]imidazole
N-[3-(4-methoxyphenyl)propyl]-6-(quinolin-8-yl)pyridine-3-carboxamide
2-(1,4-diazepan-1-yl)-N-[1-(4-propylphenyl)ethyl]acetamide
methyl (1R,3S,3aR,6aS)-3-(3-cyanophenyl)-1-(2-methoxy-2-oxoethyl)-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
1-{3-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]phenyl}imidazolidin-2-one
3-{1-[(2-chloro-6-fluorophenyl)methyl]piperidin-4-yl}-1-(pyrrolidin-1-yl)propan-1-one
3-(difluoromethoxy)-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-2-(1,1,2,2-tetrafluoroethoxy)benzamide
[(3R,5R)-5-[(dimethylamino)methyl]-1-(9H-fluorene-9-carbonyl)piperidin-3-yl]methanol
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]methanesulfonamide
2-{2-[2-(4-methoxy-3-methylphenyl)-1H-imidazol-1-yl]phenyl}ethan-1-ol
3-[(4-fluorophenyl)methyl]-5-{1-[3-(methylsulfanyl)propanoyl]piperidin-4-yl}-5-(pyridin-3-yl)imidazolidine-2,4-dione
N-[1-benzyl-7-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-carbonyl)-2-methyl-1H-1,3-benzodiazol-5-yl]acetamide
N-[3-(furan-2-yl)phenyl]-1-[2-(thiophen-2-yl)acetyl]piperidine-4-carboxamide
3-[3-(dimethylamino)propyl]-5-[(3-fluorophenyl)methyl]-5-[1-(thiophene-3-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
N-[2-(4-fluorophenyl)-1-(1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-4-yl)ethyl]-2-methoxy-N-methylacetamide
2-{4-[2-(2-aminoethyl)morpholin-4-yl]-6-oxo-1,6-dihydropyridazin-1-yl}-N-ethyl-N-methylacetamide
3-{4-[3-(aminomethyl)pyrrolidin-1-yl]-6-oxo-1,6-dihydropyridazin-1-yl}-N-(propan-2-yl)propanamide
4-[7,8-dimethyl-2-(2-methylpyrimidin-5-yl)quinoline-4-carbonyl]-1,3-dimethylpiperazin-2-one
methyl({[4-(pyridin-2-yl)phenyl]methyl})[1-(pyridin-3-yl)ethyl]amine
2-amino-6-(2H-1,3-benzodioxol-5-yl)-4-(4-methyl-1H-imidazol-5-yl)pyridine-3-carbonitrile
N-{[4-(3-methoxyphenyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
4-(2-ethylmorpholine-4-carbonyl)-7,8-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methyl-N-[2-(oxan-4-yl)ethyl]acetamide
6-(3-fluorophenyl)-N-[(3-fluorophenyl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide