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(4aR,7aS)-1-benzyl-4-(1,3-thiazol-5-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1-methylpiperidine
N-[(5-methylpyrazin-2-yl)methyl]-4-(piperidin-3-ylmethyl)benzamide
9-methoxy-N-methyl-7-oxo-3-(1-phenylcyclopropanecarbonyl)-N-(1,3-thiazol-4-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)propanamide
N-[3-(dimethylamino)propyl]-N-methyl-3-(pyrrolidine-1-carbonyl)-3-azaspiro[5.5]undecan-9-amine
5-[1-(2-methylbutanoyl)piperidin-4-yl]-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
1-{2-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-2-oxoethyl}azepan-2-one
(3aS,6aR)-5-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-[2-(4-fluorophenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-{1-[6-(propan-2-yl)-2-(trifluoromethyl)pyrimidin-4-yl]pyrrolidin-3-yl}benzoic acid
3-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}(methyl)amino)-N-methylpropanamide
4-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(methylsulfanyl)pyrimidine
7-fluoro-2-methyl-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}quinoline-4-carboxamide
N-[(5-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]methanesulfonamide
2-(2,6-dimethoxyphenyl)-5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridine
[4-({[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl](methyl)amino}methyl)oxan-4-yl]methanol
4-(2-ethoxyphenyl)-5,6-dimethyl-2-(trifluoromethyl)pyrimidine
(1R,5R)-6-methyl-3-[1-(4-methylphenyl)cyclopropanecarbonyl]-3,6-diazabicyclo[3.2.2]nonane
9-(5-chloropyridin-2-yl)-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-(cyclohexylmethyl)-3-hydroxy-3-{[(1H-indol-4-ylmethyl)amino]methyl}piperidin-2-one
2-(2,5-dimethoxyphenyl)-4-[(2-ethyl-1H-imidazol-1-yl)methyl]-5-methyl-1,3-oxazole
5-benzyl-5-{1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
3,5-dimethyl-6-[3-methyl-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
4-{2-[1-(thiophen-2-ylmethyl)piperidin-2-yl]ethyl}morpholine
N-butyl-N-(furan-2-ylmethyl)-3-hydroxybenzamide
8-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]quinoline
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[2-(propan-2-yloxy)ethyl]amine
(1R,9aR)-1-[(4-phenyl-1H-imidazol-1-yl)methyl]-octahydro-1H-quinolizin-1-ol
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
N-[4-(furan-2-yl)butan-2-yl]-3-(1,2-oxazinan-2-yl)propanamide
N-{[1-(1,2-oxazol-3-ylmethyl)piperidin-3-yl]methyl}-3-(trifluoromethyl)benzamide
N-methyl-N-[(2-methylpyridin-4-yl)methyl]-4-(piperidin-1-yl)butanamide
6-{[methyl(pyrazin-2-ylmethyl)amino]methyl}pyridine-2-carboxylic acid
2-[(5-methylpyrazin-2-yl)methyl]-8-pentanoyl-2,8-diazaspiro[5.5]undecan-3-one
2-(6-{4-[1-(morpholin-4-yl)ethyl]phenyl}pyridin-3-yl)acetic acid
N,N-diethyl-1-{[4-(furan-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperidine-3-carboxamide
3-[3-methyl-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]aniline
ethyl 4-{[4-(3-oxo-3,4-dihydropyrazin-2-yl)piperazine-1-carbonyl]amino}benzoate
1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-3-[3-methyl-1-(4-methylphenyl)-1H-pyrazol-5-yl]urea
N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]-1-benzofuran-2-sulfonamide
[2-(1H-imidazol-1-yl)ethyl](methyl){[7-methyl-2-(morpholin-4-yl)quinolin-3-yl]methyl}amine
8-chloro-2-{[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]methyl}quinoline
1-[2-methoxy-6-({methyl[2-(pyrrolidin-1-yl)ethyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
1-(4-{[methyl(thian-4-yl)amino]methyl}thiophen-2-yl)ethan-1-one
N-{[3-(3-fluorophenyl)-1,2-oxazol-5-yl]methyl}-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
3-[2-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]carbamoyl}amino)phenyl]-N-methylpropanamide
3-(5-{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)pyridine
1-({3-[2-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methyl)piperidin-4-ol
3-(piperidin-3-yl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]benzamide
2-(1H-indol-1-yl)-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}acetamide