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1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one
N-[4-(1-methyl-1H-pyrazol-4-yl)phenyl]methanesulfonamide
1,3-dimethyl-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
(1-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrrolidin-3-yl)methanamine
N-(2-hydroxyethyl)-2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-methylacetamide
N-[2-(3-methoxyphenyl)-1-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]ethyl]-N-methylfuran-2-carboxamide
1-(3-methoxyphenoxy)-3-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]propan-2-ol
N-(5-acetamido-2-fluorophenyl)-4-(pyridin-3-yloxy)piperidine-1-carboxamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-hydroxy-1-(thian-4-yl)ethyl]benzamide
1-{1-[2-(methylamino)-1,3-thiazole-4-carbonyl]piperidin-4-yl}pyrrolidin-2-one
N-[(3R,4S)-1-(2-carbamoylethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-2-ethoxybenzamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-5-methyl-6-[4-(morpholin-4-yl)piperidine-1-carbonyl]thieno[2,3-d]pyrimidin-4-amine
N-(1-{7-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-methoxypropanamide
1-[(4aR,8aR)-6-[(2E)-3-phenylprop-2-en-1-yl]-decahydro-1,6-naphthyridin-1-yl]-2-(2,4,6-trifluorophenyl)ethan-1-one
N-(1-ethyl-1H-1,2,3-triazol-4-yl)-2-[2-(4-methylbenzoyl)-1H-imidazol-1-yl]acetamide
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-[2-(dimethylamino)ethyl]-N-methylpiperidine-3-carboxamide
{[(1R,5S,6S)-3-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-3-azabicyclo[3.1.0]hexan-6-yl]methyl}dimethylamine
5-[1-(furan-2-ylmethyl)-1H-imidazol-2-yl]-2-(pyrrolidin-1-yl)-1,3-thiazole
1-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(thiophen-3-yl)ethan-1-one
(4aS,7aR)-1-(furan-2-ylmethyl)-4-(3-methylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}morpholine
7-methyl-11-[3-(1H-pyrazol-1-yl)propyl]-3,7,11-triazaspiro[5.6]dodecane
7-(cyclopropylmethyl)-2-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-2,7-diazaspiro[4.5]decane
2-(2H-indazol-2-yl)-1-(4-methyl-3-phenylpiperazin-1-yl)ethan-1-one
8-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-hydroxy-2-methyl-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)pyrimidine-5-carboxamide
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-4-[(2,4-dimethoxyphenyl)methyl]-9-(oxolan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-(2-methylpropyl)-3-(2-oxo-2-{4-[2-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}ethyl)piperazin-2-one
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-7-methoxy-4-methylquinazoline
5-ethyl-6-methyl-N4-[(3,4,5-trimethoxyphenyl)methyl]pyrimidine-2,4-diamine
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-2-(pyrimidin-2-ylsulfanyl)acetamide
5-[4-(1H-pyrazol-1-yl)phenyl]pyrimidine
N-[2-(pyridin-4-yl)ethyl]-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
N-{5H,6H,7H,8H,9H,10H,11H-cycloocta[b]indol-2-ylmethyl}-1,2-dimethyl-1H-imidazole-4-sulfonamide
1-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopentyl-2-(propan-2-yl)pyrimidine-5-carboxamide
5-(2,3-difluorophenyl)pyrimidin-2-amine
N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)pyrazine-2-carboxamide
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
4-[(4-methoxy-2,5-dimethylphenyl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N,N-dimethyl-2-{1-[(3-methylphenyl)methyl]-1H-pyrazol-4-yl}quinoline-4-carboxamide
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
methyl 3-[2-oxo-4-(oxolane-3-carbonyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-1-yl]propanoate
2-{1-[(2E)-3-(5-chloro-2-hydroxyphenyl)-2-methylprop-2-en-1-yl]piperidin-4-yl}-N-methylacetamide
2-(dimethylamino)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(2-methylphenyl)acetamide
2-{5-[3-(1H-imidazol-2-yl)benzoyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
1-(2-methoxyethyl)-3-(3-methoxyphenyl)-3-{2-[4-(6-methylpyridin-2-yl)piperazin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
N-methyl-N'-(4-methylphenyl)-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}propanediamide
3-[4-(2-oxo-1,3-oxazolidin-3-yl)piperidine-1-carbonyl]-6-phenyl-1,2-dihydropyridin-2-one
N-(3-methylphenyl)-3-[1-(quinoline-6-carbonyl)piperidin-4-yl]propanamide