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5-methyl-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-1,3,4-oxadiazol-2-amine
N-[(2S,4R,6S)-2-(6-chloro-4-oxo-4H-chromen-3-yl)-6-(2-methylpropyl)oxan-4-yl]acetamide
(4aR,7aS)-1-cyclopropanecarbonyl-4-[3-(4-methyl-1H-pyrazol-1-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pent-4-en-1-one
N-({7-[4-(4-methoxyphenyl)-4-oxobutanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-3-carboxamide
N-[(3S,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3,5-difluorobenzamide
N-[3-fluoro-5-(trifluoromethyl)phenyl]-3-oxopiperazine-1-carboxamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[2-(4-methylpiperidin-1-yl)ethyl]-1H-pyrazole-3-carboxamide
N-[1-(cyclohex-1-en-1-yl)ethyl]-1H,4H,6H,7H-pyrano[4,3-c]pyrazole-3-carboxamide
1-{2-[methyl({[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl})amino]ethyl}piperidin-2-one
N-(2-fluorophenyl)-2-{4-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]morpholin-3-yl}acetamide
1-{2-[(2,5-difluorophenyl)carbamoyl]ethyl}-5-oxopyrrolidine-3-carboxylic acid
1-[(1-benzyl-3-methyl-1H-1,2,4-triazol-5-yl)methyl]-1,2-dihydropyrimidin-2-one
N-(1-{1-[(5-chloro-2-hydroxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
3-(3,4-dimethoxyphenyl)-N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)propanamide
N-{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}-N-methylcyclohexanamine
ethyl 4-{1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}piperazine-1-carboxylate
N-{1-[2-(1,2-oxazolidin-2-yl)-2-oxoethyl]-1H-pyrazol-4-yl}-2-(phenylsulfanyl)acetamide
(4S)-N-(5-chloro-2-methylphenyl)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidine-1-carboxamide
N-(5-chloro-2-methoxyphenyl)-3-{1-[2-(2-oxopiperidin-1-yl)acetyl]piperidin-3-yl}propanamide
(2S,4R)-N-ethyl-4-[(1-methylpiperidin-4-yl)amino]-1-(naphthalen-1-ylmethyl)pyrrolidine-2-carboxamide
2-[(dimethylamino)methyl]-N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-1,3-thiazole-4-carboxamide
2-[2-({cyclopropyl[(2-methoxyphenyl)methyl]amino}methyl)phenoxy]ethan-1-ol
2-[4-(3-chlorothiophene-2-carbonyl)piperazin-1-yl]-N-ethylacetamide
3-chloro-N-cyclohexyl-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-1-[4-(methoxymethyl)piperidin-1-yl]propan-1-one
[(4aS,8aR)-6-(3-methoxypyrazin-2-yl)-decahydro-1,6-naphthyridin-4a-yl]methanol
2,3-dimethyl-N-[2-(3-{[methyl(thiophen-2-ylmethyl)amino]methyl}phenoxy)propyl]-1H-indole-7-carboxamide
N-{3-[(3S,4S)-3,4-dihydroxypiperidine-1-carbonyl]-4-(2,5-dimethyl-1H-pyrrol-1-yl)phenyl}acetamide
2-methyl-N-{[6-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1,3-thiazole-4-carboxamide
N-[(3-{1-[(4-fluorophenyl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}-1,2-oxazol-5-yl)methyl]-N-methylacetamide
N-cyclopropyl-1-[(1s,4s)-4-[2-(4-methylphenoxy)acetamido]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
(5-{1-[2-fluoro-3-(trifluoromethyl)phenyl]-1H-imidazol-2-yl}furan-2-yl)methanol
2-[4-(6-chloro-1,3-benzothiazol-2-yl)-1H-pyrazol-1-yl]-N-(2-ethyl-2H-1,2,3-triazol-4-yl)acetamide
(3S,4R)-1-(8-methoxy-4-methylquinolin-2-yl)-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
5-(4-chloro-2-methoxyphenoxymethyl)-N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
N-benzyl-5-methyl-N-(oxolan-2-ylmethyl)-1-propyl-1H-pyrazole-4-carboxamide
N-cyclobutyl-3-{methyl[2-(methylcarbamoyl)ethyl]sulfamoyl}benzamide
methyl 2-oxo-1-(prop-2-en-1-yloxy)-8-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-1,8-diazaspiro[4.5]decane-4-carboxylate
1-{1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}-N-(2-phenylethyl)piperidine-4-carboxamide
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(methylamino)acetamide
N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-1-(pyrimidin-2-yl)piperidin-3-amine
2-({3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)-3-methyl-1H-indole
N-[(3R,4S)-4-propyl-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]pyrrolidin-3-yl]methanesulfonamide
N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-1-(propan-2-yl)-1H-pyrazole-5-carboxamide
(2S,4R)-4-amino-N-ethyl-1-(5-methoxy-2,4-dimethylbenzenesulfonyl)pyrrolidine-2-carboxamide
(1S,5R)-6-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-{1-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]propyl}aniline
2-{[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]methyl}quinoline
N,4,6-trimethyl-2-oxo-N-[(5-phenyl-1H-pyrazol-4-yl)methyl]-1,2-dihydropyridine-3-carboxamide