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(1S,9R)-11-[(7-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
4-[2-(1H-imidazol-2-yl)benzoyl]-1-(2-methoxyphenyl)piperazin-2-one
2-{[(3-ethoxyphenyl)methyl]({[5-(1H-pyrazol-5-yl)furan-2-yl]methyl})amino}ethan-1-ol
2-{5-[(5-cyclopentylthiophen-2-yl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
3-methyl-N-[3-(morpholin-4-yl)propyl]-5-propyl-1-benzofuran-2-carboxamide
5-(3-ethynylbenzoyl)-1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-1,4-oxazepane
4-(2,4-dimethylphenyl)-3-(1-methoxypropyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-cyclopentyl-N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)acetamide
2-{2-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethoxy}ethan-1-ol
methyl({4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl})[1-(pyridin-2-yl)propyl]amine
N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]-1-propanoylpyrrolidine-2-carboxamide
N-(2-hydroxyethyl)-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}-N-(propan-2-yl)acetamide
N-[(1-ethylpiperidin-3-yl)methyl]-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
4-[(5-cyclopropyl-3-methyl-1H-pyrazol-4-yl)formamido]-N,4-dimethylpentanamide
N-ethyl-N-(1-hydroxypropan-2-yl)-6-methoxy-2,3-dihydro-1H-indene-5-carboxamide
2-{[2-amino-6-(3,5-dimethyl-1H-pyrazol-4-yl)pyrimidin-4-yl]amino}ethan-1-ol
dimethyl({[(3S,4R)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl})amine
1-{2-methyl-5-[4-(trifluoromethyl)piperidine-1-carbonyl]phenyl}imidazolidin-2-one
2,5-dimethyl-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
3-[(4aR,7aS)-6,6-dioxo-4-[2-(propylsulfanyl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
prop-2-en-1-yl N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}carbamate
N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methylbutanamide
methyl (2S,4S,5R)-1,2-dimethyl-5-(2-methylphenyl)-4-(piperidine-1-carbonyl)pyrrolidine-2-carboxylate
2-[(2-chlorophenyl)methyl]-4-(pyridin-3-ylmethyl)morpholine
N-ethyl-6-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
N-({2-[4-(furan-3-amido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-1-(pyridin-2-yl)piperidine-3-carboxamide
(3aR,6aR)-2-(4-methylbenzoyl)-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(3-{4-[(3,3-diphenylpropyl)amino]piperidin-1-yl}phenyl)cyclopropanecarboxamide
2-(2-ethoxypyridin-3-yl)-6,7-dimethoxyquinazolin-4-amine
4,6-dimethoxy-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}pyrimidin-2-amine
2-{3-[4-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]piperidin-1-yl}acetamide
7-hydroxy-4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-6-methyl-1,2,3,4-tetrahydroquinolin-2-one
1-(naphthalen-1-ylmethyl)-N-[2-(pyridin-3-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-4-(1H-pyrazol-1-ylmethyl)-1,3-oxazole
2-amino-N-[1-(furan-2-ylmethyl)piperidin-4-yl]-4-methyl-1,3-benzothiazole-6-carboxamide
2-[8-(cyclohex-3-en-1-ylmethyl)-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
(2R)-1-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl]-2-amino-4-methylpentan-1-one
3-[3-methyl-1-(2-methylpropyl)-1H-pyrazol-5-yl]-1-{[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}urea
5-(3,4-difluorophenoxymethyl)-N-[1-(3-methylpyridin-2-yl)ethyl]-1,2-oxazole-3-carboxamide
1-{2-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-2-oxoethyl}-4-methyl-1,2-dihydroquinolin-2-one
ethyl 5-[(3-hydroxyphenyl)methyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-methyl-5-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-1,3-benzothiazole
5-(1H-1,3-benzodiazol-2-ylmethyl)-11-methyl-8-thia-3,5,10-triazatricyclo[7.4.0.02,7]trideca-1(13),2(7),3,9,11-pentaen-6-one
N-[2-(5-cyano-2-methyl-1H-indol-3-yl)ethyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
2-(3-chloro-4-hydroxyphenyl)-1-[2-(pyrrolidine-1-carbonyl)piperazin-1-yl]ethan-1-one
1-[2-(2,3-difluorophenoxymethyl)-1,3-oxazole-4-carbonyl]azepane
3-methoxy-5-methyl-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}thiophene-2-carboxamide
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]propanamide
2-[4-(4-chlorophenyl)-4H-1,2,4-triazol-3-yl]ethan-1-amine