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7-acetamido-1-[(4-fluorophenyl)methyl]-N-methyl-N-(thiophen-3-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
(3S,4S)-1-[2-(benzyloxy)ethyl]-4-cyclopropylpyrrolidine-3-carboxylic acid
2-{[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-1H-indole
1-(1H-imidazol-2-ylmethyl)-4-(3-phenylpropyl)-1,4-diazepane
N-{5-[(2R,6S)-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]pyridin-2-yl}acetamide
1-(3-methylfuran-2-carbonyl)-4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
2-cyclopentyl-9-(pyrimidin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(3aS,6aS)-1-oxo-5-(3-phenylpropyl)-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-N-(6-methylpyridin-3-yl)piperazine-2-carboxamide
[(2-chloro-4,5-dimethoxyphenyl)methyl][2-methoxy-1-(pyridin-2-yl)ethyl]methylamine
1,6-dimethyl-N-[2-(2-methyl-1H-indol-1-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-cyclohexyl-N-[(2-methylphenyl)methyl]-2,7-dioxo-1,3-diazepane-4-carboxamide
N-[3-(furan-2-yl)propyl]-1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
1-{2-[4-(1-hydroxy-3-phenylpropyl)piperidin-1-yl]-2-oxoethyl}azepan-2-one
5-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
5-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
1,3-dimethyl-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4-(thian-4-yl)piperazine
2-chloro-4-{4-phenyl-1-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]-1H-imidazol-5-yl}phenol
N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-4-(pyridin-2-yl)pyrimidin-2-amine
1-[7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-2-yl]-4,4,4-trifluorobutan-1-one
7-fluoro-N-[1-(thiophen-2-yl)propan-2-yl]quinazolin-4-amine
N-(1-{7-[(4-methoxy-2,3-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxane-4-carboxamide
1-({2,4-dimethyl-5H,6H-furo[2,3-d]pyrimidin-6-yl}methyl)-4-ethyl-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[1-(2,3-dimethylphenyl)piperidin-4-yl]piperazine-2-carboxylic acid
1-[(3-methylphenyl)methyl]-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
N-[2-(4-chlorophenyl)ethyl]-2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-{4-[(dimethylsulfamoyl)amino]phenyl}-N-[2-(5-phenyl-4H-1,2,4-triazol-3-yl)ethyl]piperidin-4-amine
1-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(4-methylphenyl)ethan-1-one
methyl 3-{[1-(cyclopropylmethyl)-5-[3-(3,5-dimethylphenyl)propanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]formamido}propanoate
8-(6-methylpyridine-3-carbonyl)-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-{[(2R,3R)-2-methoxy-3-(2-phenoxyacetamido)-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]carbonyl}pyridin-1-ium-1-olate
N-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
1-(2-{[cyclohexyl(methyl)amino]methyl}phenyl)-3-[2-(1H-pyrazol-4-yl)ethyl]urea
4-[(4S)-4-hydroxy-3,3,4-trimethylpiperidine-1-carbonyl]-1,2-dihydroisoquinolin-1-one
(1R,5R)-6-benzyl-3-(3-methyl-1,2-oxazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
5-(5-fluoro-2-methylphenyl)-3-(2-phenylethyl)-1H-1,2,4-triazole
6-(dimethylamino)-N-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]pyridine-3-carboxamide
6-ethyl-2-(morpholin-4-yl)-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyrimidin-4-amine
3-[(2-chloro-5-acetamidophenyl)formamido]-N-(1,3-thiazol-2-yl)propanamide
N-[(1-hydroxycyclohexyl)methyl]-2-(4H-1,2,4-triazol-4-yl)benzamide
1-cyclohexyl-N-methyl-N-[(2-methylpyridin-4-yl)methyl]piperidine-4-carboxamide
2-(4-{1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carbonyl}piperazin-1-yl)ethan-1-ol
(2R,6R)-4-(2-hydroxyethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
6-acetyl-2-amino-4-(thiophen-3-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
6-[(2-hydroxynaphthalen-1-yl)methyl]-N-[2-(2-methoxyphenyl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
3-(N-methyl-1-{1-methyl-3-phenyl-1H-thieno[2,3-c]pyrazol-5-yl}formamido)propanamide
1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-N,N-diethylpiperidine-3-carboxamide
2,5-dimethyl-4-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]pyrimidine