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2-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}-5-(piperazin-1-yl)-2,3-dihydropyridazin-3-one
1-[(2-chlorophenyl)methyl]-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-4-ol
(3S,4S)-4-methoxy-1-{[4-phenyl-5-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}pyrrolidin-3-ol
N-(butan-2-yl)-5-hydroxy-N-(3-phenylprop-2-yn-1-yl)pyrazine-2-carboxamide
(3aR,6aR)-2-(cyclobutylmethyl)-5-[2-(thiophen-3-yl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(2-amino-1,3-thiazol-4-yl)-1-[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]propan-1-one
4-[5-cyclopropyl-4-(piperidine-1-carbonyl)-1H-pyrazol-1-yl]-3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaene
2-cyclopropyl-9-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(oxolan-2-ylmethyl)-6-phenyl-N-(pyridin-4-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-(6-methyl-2-phenylpyrimidin-4-yl)piperazine-2-carboxylic acid
4-[(2-methyl-1H-imidazol-1-yl)methyl]-1-(3,3,3-trifluoro-2-methylpropyl)piperidine
1-[(2-chlorophenyl)methyl]-4-[3-(propan-2-yl)-1,2-oxazol-5-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-butyl-5-[3-(methoxymethyl)piperidine-1-carbonyl]-1,3-benzoxazole
1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-8-(1,2,3,4-tetrahydronaphthalen-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(5-{1-benzyl-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl}furan-2-yl)methanol
(2E)-N-{[5-(benzylsulfanyl)-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}-3-(3-fluorophenyl)prop-2-enamide
6-({4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}methyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(4-fluorophenyl)-4-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]-1,4-diazepane
8-(4-ethyl-5-methylthiophene-3-carbonyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
3-hydroxy-3-{[4-(2-hydroxypropan-2-yl)piperidin-1-yl]methyl}-1-(2-phenylethyl)piperidin-2-one
N-[2-(1H-imidazol-4-yl)ethyl]-2-methyl-1-benzofuran-7-carboxamide
2-(4-{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrazine
4-ethyl-1-methyl-3-{1-[(4-methylpiperazin-1-yl)sulfonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
5-chloro-N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-1H-1,2,4-triazole-3-carboxamide
8-{[4-(1H-imidazol-1-yl)phenyl]methyl}-2-methyl-2,8-diazaspiro[4.5]decan-3-one
N-(2-{[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)acetamide
5-[9-hydroxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]pyridine-2,4-diol
4-benzyl-3-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]piperazin-2-one
4-[4-(2-hydroxypropan-2-yl)-1H-1,2,3-triazol-1-yl]-N-[(3-methoxyphenyl)methyl]piperidine-1-carboxamide
(1S,5R)-3-benzyl-6-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
4-(hydroxymethyl)-1-(1-methyl-1H-indazole-3-carbonyl)piperidin-4-ol
N-{[1-(2-acetamidoacetyl)piperidin-3-yl]methyl}naphthalene-1-carboxamide
(2R)-2-amino-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-methoxypropanamide
N-cyclohexyl-2-ethyl-N-[2-(ethylsulfanyl)ethyl]pyrimidine-5-carboxamide
1-(2-aminoethyl)-N-methyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-1H-1,2,3-triazole-4-carboxamide
3-chloro-N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)benzamide
5-chloro-2-oxo-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}-1,2-dihydropyridine-3-carboxamide
N,N-dimethyl-1-{[2-(pyridine-3-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]sulfonyl}pyrrolidin-3-amine
(3R,4R)-4-(azepan-1-yl)-1-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-ol
N-methyl-3-phenyl-N-[1-(pyridin-3-yl)propyl]-1H-pyrazole-4-carboxamide
2-{1-[1-(2-phenylbenzoyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
2-[(3,4-difluorophenyl)methyl]-8-(6-hydroxyhexyl)-2,8-diazaspiro[4.5]decan-3-one
methyl 2-({1-methyl-2-oxo-3-phenyl-1,8-diazaspiro[4.5]decane-8-carbonyl}amino)acetate
(3aR,6aS)-5-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}-4-chloro-1-methyl-1H-pyrazole-3-carboxamide
2-{1-[1-cyclohexyl-3-(cyclopropylmethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl]-N-methylformamido}-N-methylacetamide
1-[1-(1H-imidazole-4-carbonyl)piperidin-3-yl]-4-(2-methoxyphenyl)piperazine
2-{4-[(2-chloro-6-fluorophenyl)methyl]-1-cyclohexylpiperazin-2-yl}ethan-1-ol
2-(2H-1,3-benzodioxol-5-yl)-1-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-2-(1H-pyrrol-1-yl)propanamide