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N-({3-methoxy-4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}methyl)pyrrolidin-3-amine
2-[1-({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidine-3-carbonyl]pyridine
dimethyl({[(3S,4R)-1-[2-(methylsulfanyl)pyridine-3-carbonyl]-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl})amine
2-[3-(hydroxymethyl)phenyl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-[(4aR,7aS)-4-[(1-methyl-1H-imidazol-2-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
N-cyclopropyl-2,6-dimethyl-N-(1,3-thiazol-2-ylmethyl)quinoline-3-carboxamide
6-(3-chlorophenyl)-8-oxo-7-(prop-2-en-1-yl)-N-propyl-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-[1-(2-chloropyridine-4-carbonyl)piperidin-3-yl]-4-(2-fluorophenyl)piperazine
8-(4-methylpyrimidine-5-carbonyl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-{5-[6-(dimethylamino)pyridin-3-yl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
3-{5-[({1-[(3-methoxyphenyl)methyl]piperidin-3-yl}amino)methyl]thiophen-3-yl}prop-2-yn-1-ol
1-[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
3-[5-({[2-(2,4-dimethylphenoxy)ethyl](methyl)amino}methyl)thiophen-3-yl]prop-2-yn-1-ol
1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
5-(3-{[(7-methoxy-4-methylquinolin-2-yl)amino]methyl}pyrrolidin-1-yl)-2-methyl-2,3-dihydropyridazin-3-one
6-methoxy-2-oxo-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-3-(4,5-dimethyl-1H-pyrazol-3-yl)propan-1-one
(3S,5R)-1-(4-methyl-1H-imidazole-5-carbonyl)-5-(4-methylpiperazine-1-carbonyl)piperidine-3-carboxylic acid
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-2,4-dimethoxy-N-(2-methoxyethyl)benzamide
5-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}pyridin-2-amine
(3S,9aR)-3-[(1R)-1-(benzyloxy)ethyl]-8-(4-methylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
(2S,4R)-N-ethyl-4-({[4-(methylsulfanyl)phenyl]methyl}amino)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
5-[(3-hydroxypiperidin-1-yl)methyl]-N-[2-(3-methylpyridin-2-yl)ethyl]-1,2-oxazole-3-carboxamide
3-(3-methylbutyl)-8-(2-methyloxane-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[4-({[2-(dimethylamino)ethyl]amino}methyl)-2-methoxyphenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
1-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-3-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}urea
3-ethoxy-1-[3-(1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
[(5-fluoro-1H-indol-2-yl)methyl][(4-methanesulfonylphenyl)methyl]methylamine
3-(1-cycloheptylpiperidin-3-yl)-1-[2-(methylsulfanyl)phenyl]urea
7-fluoro-3-methyl-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1-benzofuran-2-carboxamide
2-[1-(2,3-dihydro-1H-inden-5-yl)-5-{[methyl(pyridin-3-ylmethyl)amino]methyl}-1H-1,2,4-triazol-3-yl]acetamide
N,N-dimethyl-2-[6-(piperidine-1-carbonyl)pyrazin-2-yl]aniline
8-[1-(2,3-dimethylphenyl)piperidin-4-yl]-2-methyl-2,8-diazaspiro[4.5]decan-3-one
3-(3-fluorophenoxymethyl)-1-(1,3-thiazol-4-ylmethyl)piperidine
8-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[benzyl(methyl)amino]-3-[4-({[(3-fluoro-4-methylphenyl)methyl]amino}methyl)phenoxy]propan-2-ol
2-cyclopropyl-4-hydroxy-N-{1-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]ethyl}pyrimidine-5-carboxamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-(adamantan-1-yl)-N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methylacetamide
1-[(4aS,8aS)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-(4-phenylpiperidin-1-yl)ethan-1-one
3-[(3S,4R)-1-benzyl-4-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-3-yl]-N-(2,3-dihydro-1H-inden-5-yl)propanamide
2-(4-{4-cyclopropyl-5-[(dimethylamino)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyridine-4-carbonitrile
1-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-3-(methoxymethyl)piperidine
2-(cyclopropylmethyl)-7-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[1-(pyrazin-2-yl)piperidin-3-yl]-1H-1,2,3-benzotriazole-5-carboxamide
6-methyl-5-{2-oxo-2-[2-(3-phenylpropyl)morpholin-4-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-({7-[(4-fluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-phenylacetamide
1-{[1-(hydroxymethyl)cyclobutyl]methyl}-5,5-diphenylpiperidin-2-one