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2-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-amine
3-cyclopentyl-1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazole
(1H-imidazol-2-ylmethyl)({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)methylamine
N-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-[1,2,3,4]tetrazolo[1,5-a]pyridine-5-carboxamide
8-{5-methyl-6-[(2-methylpyridin-3-yl)oxy]pyrimidin-4-yl}-1-oxa-8-azaspiro[4.5]decane
4-({2-[2-(1-ethyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]phenyl}methyl)morpholine
(2S,4R)-4-{[(3,4-difluorophenyl)methyl]amino}-N-(2-methoxyethyl)-1-(propan-2-yl)pyrrolidine-2-carboxamide
3-[(3R,4S)-1-(1H-imidazol-4-ylmethyl)-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
(4aR,7aS)-1-cyclopropanecarbonyl-4-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-benzyl-3-[2-(4-ethylpiperazin-1-yl)-2-oxoethyl]-1-methyl-2,3-dihydro-1H-indol-2-one
2-(5-fluoro-2-methyl-1H-indol-3-yl)-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
1-[3-(2-chlorophenyl)pyrrolidin-1-yl]-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N-(3-hydroxy-3-phenylpropyl)-N-methylimidazo[2,1-b][1,3]thiazole-6-carboxamide
4-({3-[3-(2H-1,3-benzodioxol-5-yl)phenyl]-1H-pyrazol-1-yl}methyl)-3-methylpyridine
2-[(3R,4S)-3-(3-hydroxypropanamido)-4-(propan-2-yl)pyrrolidin-1-yl]acetic acid
methyl 1-[(3R,5S)-5-[(diphenylmethyl)carbamoyl]-1-[(4-ethylphenyl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-{[5-chloro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(trifluoromethyl)benzamide
1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)(methyl){[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}amine
{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[2-(1H-pyrazol-4-yl)ethyl]amine
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl][2-(2-fluorophenyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]ethyl]methylamine
2-{1-benzyl-4-[1-(2-fluorophenyl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
1-(furan-2-carbonyl)-N-[4-(1H-indol-3-yl)butan-2-yl]piperidin-4-amine
N-methyl-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[1-(4-methylpyridin-2-yl)propan-2-yl]acetamide
(4aS,8aR)-1-(2-aminoethyl)-6-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]-decahydro-1,6-naphthyridin-2-one
ethyl 1-(cyclopropylmethyl)-5-[2-(6-methoxy-2-oxo-2,3-dihydro-1H-indol-3-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-(naphthalen-2-yl)-4-(pyrrolidin-3-ylmethyl)piperazine
1-[(3-fluorophenyl)methyl]-5-(1,2-oxazolidine-2-carbonyl)piperidin-2-one
(4aS,8aR)-1-(3-hydroxypropyl)-6-(1H-indazole-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
3-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)propanamide
N,N-diethyl-1-[(1s,4s)-4-(3,4,5-trimethoxybenzamido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
(4aS,7aR)-1-(1H-pyrazole-3-carbonyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(1H-imidazol-4-yl)ethyl]-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
N-(1-cyclopropylethyl)-6-(2,5-dimethylfuran-3-yl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
5-cyclopropyl-4-phenyl-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-imidazole
N-(3-methoxypropyl)-3-methyl-N-{[6-(2-methylphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}thiophene-2-carboxamide
N-cyclohexyl-4-oxo-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carboxamide
(3S,4R)-1-[(4-fluoro-3-methoxyphenyl)methyl]-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
1-(2-fluorophenyl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(2,2,3,3-tetrafluoropropoxy)ethan-1-one
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(3-methylpyridin-2-yl)ethyl]acetamide
2-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}phenyl)-4,6-dimethoxypyrimidine
N-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-5-yl)-2-(1,3-thiazol-2-yl)pyrrolidine-1-carboxamide
7,7-dimethyl-2-(oxan-2-ylmethyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
5-{[1-(2-cyclohexylethyl)-3-hydroxy-2-oxopiperidin-3-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonitrile
(2H-1,3-benzodioxol-4-ylmethyl)({[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})methylamine
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-2-(morpholin-3-yl)acetamide
N-(1-{1-[(3,5-difluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-phenylbutanamide
3-[4-(dimethylamino)phenyl]-1-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]propan-1-one
{1-[1-(4-chloro-2-methoxybenzoyl)piperidin-3-yl]piperidin-4-yl}methanol