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(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-(4-methyl-1,3-thiazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-[6-(piperidine-1-carbonyl)pyrazin-2-yl]-2-(trifluoromethyl)morpholine
3-{2-[4-(propan-2-yl)piperazin-1-yl]ethyl}-3,4-dihydroquinazolin-4-one
3-[1-(propan-2-yl)-1H-imidazol-2-yl]-1-{[2-(1H-pyrazol-1-yl)phenyl]methyl}piperidine
{2-[3-(2-ethylphenoxy)azetidin-1-yl]-2-oxoethyl}urea
2-[1-(3-methylbutyl)-4-{[3-(methylsulfanyl)phenyl]methyl}piperazin-2-yl]ethan-1-ol
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)sulfonyl]piperidin-3-ol
6-{[(2-phenylethyl)(pyridin-2-ylmethyl)amino]methyl}-1,4-oxazepan-6-ol
3-(2-methyl-1H-imidazol-1-yl)-1-[2-methyl-4-(4-methylphenyl)piperazin-1-yl]propan-1-one
3-(3-chlorophenyl)-3-(3-hydroxyphenyl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]propanamide
1-[2-(2-methyl-1H-indol-3-yl)acetyl]-4-(pyrimidin-2-yl)piperazine-2-carboxylic acid
3-[(3R,4S)-1-(5-ethyl-1H-pyrrole-2-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
4-{7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}-N-methylpyridin-2-amine
8-(6-cyclopropylpyrimidin-4-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-{4-[(1-methoxybutan-2-yl)amino]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
(3S,4R)-1-[(4-acetylphenyl)methyl]-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-(2-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)methanesulfonamide
1-{[3-cyclopropyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-4-methyl-1,2-dihydroquinolin-2-one
3-[(2-hydroxyethyl)[(2-methylphenyl)methyl]sulfamoyl]-N,N-dimethylbenzamide
N-[(3-fluorophenyl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-6-oxopiperidine-3-carboxamide
2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-{1-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
5-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carbonyl}pyridine-2-carbonitrile
(1r,4r)-4-({4-[4-(2-chlorophenyl)piperidin-4-yl]pyrimidin-2-yl}amino)cyclohexan-1-ol
1-[(2-chlorophenyl)methyl]-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
3-(4-methanesulfonylphenyl)-6-(pyrrolidin-1-yl)pyridazine
3-acetamido-5-({[(2-hydroxynaphthalen-1-yl)methyl]amino}methyl)-N-(2-methoxyphenyl)benzamide
N-({1-[(3-phenyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)methanesulfonamide
3-{methyl[2-(pyridin-2-yl)ethyl]amino}-N-[2-(methylsulfanyl)phenyl]piperidine-1-carboxamide
(2S,4R)-1-[(2,6-difluorophenyl)methyl]-4-[(4-fluorophenyl)sulfanyl]-N-{imidazo[1,2-a]pyridin-2-ylmethyl}pyrrolidine-2-carboxamide
(1S,5R)-6-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
(2E)-N-{[3-methyl-7-(1-methyl-1H-pyrazole-3-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-phenylprop-2-enamide
9-ethyl-3-{1-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-imidazol-2-yl}-9H-carbazole
5-methoxy-3-[1-(pyrazin-2-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3-(pyrazin-2-yl)propanamide
3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)propanamide
N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)-1,2,5-thiadiazole-3-carboxamide
4-(2-methoxy-5-{[1,3]oxazolo[4,5-b]pyridin-2-yl}phenyl)-4H-1,2,4-triazole
2-[5-(2H-1,2,3-benzotriazol-2-ylmethyl)-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-1-yl]ethan-1-ol
5-[2-(methylsulfanyl)phenoxymethyl]-N-[2-(pyridin-3-yloxy)propyl]-1,2-oxazole-3-carboxamide
(3S,4S)-4-cyclopropyl-1-[3-(4-methyl-1,4-diazepan-1-yl)propanoyl]pyrrolidine-3-carboxylic acid
3-({4-[bis(4-fluorophenyl)methyl]piperazin-1-yl}methyl)piperidin-3-ol
dimethyl({4-[1-(3-methyl-1H-pyrazole-5-carbonyl)piperidin-2-yl]phenyl}methyl)amine
2-(1H-indol-3-yl)-1-{4-[2-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}ethan-1-one
N-[2-(dimethylamino)ethyl]-N-[(4-methylphenyl)methyl]-4-propylpyrimidine-5-carboxamide
1-benzyl-4-{[4-(dimethylamino)-5-fluoropyrimidin-2-yl]amino}pyrrolidin-2-one
6-(propan-2-yl)-N4-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}pyrimidine-2,4-diamine
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N-methyl-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N-methyl-3-[({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]benzamide
2-[1-(1-methanesulfonylpiperidin-4-yl)-1H-imidazol-2-yl]pyridine
(2R)-N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-hydroxy-2-phenylacetamide