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methyl 3-cyclohexaneamido-5-({[4-(morpholin-4-yl)phenyl]formamido}methyl)benzoate
4-[(1-cyclopentylpiperidin-4-yl)oxy]-3-methoxy-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]benzamide
2-benzyl-N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-1,3-thiazole-4-carboxamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-N-(2,2-dimethyloxan-4-yl)-5-methyl-1H-pyrazole-4-carboxamide
2-(2-phenylethyl)-1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
4-(2-methoxyethyl)-N-[2-(pyridin-3-yloxy)phenyl]piperazine-1-carboxamide
(3aR,5S,6S,7aS)-2-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-octahydro-1H-isoindole-5,6-diol
methyl 5-[(cyclohex-3-en-1-ylmethyl)amino]-3-(furan-2-amido)-1-(2-methoxyethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-[2-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-4H-chromen-4-one
1'-[2-(pyrrolidin-3-yl)benzoyl]spiro[indene-1,4'-piperidine]
2-[5-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
[3-(2-phenylethyl)-1-(quinolin-2-yl)piperidin-3-yl]methanol
3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)piperidine
1-[(3-methoxyphenyl)methyl]-4-[(5-methylthiophen-2-yl)methyl]piperazin-2-one
5-[(4-cyclobutanecarbonyl-1,4-diazepan-1-yl)methyl]isoquinoline
(1R,5R)-3-(7-chloro-1-methyl-1H-indole-2-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
N4-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-5,6-dimethylpyrimidine-2,4-diamine
methyl 3-[(2-ethoxyphenyl)methyl]-7-oxo-9-[2-(pyridin-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-[(2-methoxyphenyl)methyl]-N-(2-methyl-1-benzofuran-5-yl)piperazine-1-carboxamide
5-[2-(aminomethyl)-5-fluoro-2,3-dihydro-1-benzofuran-7-yl]pyrimidin-2-amine
2-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-1,2,3,4-tetrahydroisoquinoline
methyl (2S,4S)-4-[2-(methoxycarbonyl)thiophene-3-sulfonamido]-1-methylpyrrolidine-2-carboxylate
N-(2H-1,3-benzodioxol-5-ylmethyl)-7-fluoro-3-methyl-1-benzofuran-2-carboxamide
1'-(3-methylbenzoyl)-5-(3-methylbut-2-en-1-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4,4,4-trifluoro-1-[3-(4-phenoxybenzoyl)piperidin-1-yl]butan-1-one
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-2-(7-fluoro-2-methyl-1H-indol-3-yl)acetamide
N-(1-cycloheptylpiperidin-3-yl)-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
3-{2-[2-(3,5-dimethyl-1-benzofuran-2-yl)-1H-imidazol-1-yl]ethyl}-4-ethyl-4H-1,2,4-triazole
6-methyl-2-(1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
N-[(2-methoxyphenyl)methyl]-6-oxo-N-(pyridin-3-ylmethyl)-1,6-dihydropyridazine-3-carboxamide
(3R,4S)-4-[ethyl({[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl})amino]oxolan-3-ol
(2R,6R)-4-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(2S,4R)-1-[(2-fluorophenyl)methyl]-4-[(4-fluorophenyl)sulfanyl]-N-methyl-N-(1,3-thiazol-4-ylmethyl)pyrrolidine-2-carboxamide
4-(furan-3-yl)-N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-N,6-dimethyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
8-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(3-hydroxy-3-methylbutyl)-N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]benzamide
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
6-(1-phenylcyclohexanecarbonyl)-1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octane
(1R,3S)-7-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-methoxy-7-azaspiro[3.5]nonan-1-ol
2-benzyl-9-(2-ethoxypropanoyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(5-chloro-2,4-dimethoxyphenyl)methyl]-4-[2-(methylsulfanyl)ethyl]piperazine
2-(1H-1,3-benzodiazol-2-ylmethyl)-7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
2-amino-4-{[(5-methyl-1H-pyrazol-3-yl)methyl]amino}quinazoline-6-carboxylic acid
N-{[1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-3-yl]methyl}furan-2-carboxamide
2-{2-methyl-6-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]pyrimidin-4-yl}ethan-1-amine
methyl 3-(2-methoxybenzamido)-5-{[(4-methyl-1,2,5-oxadiazol-3-yl)formamido]methyl}benzoate
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-3-(thiophen-2-yl)propanamide
1-(2,3-dihydro-1H-inden-2-yl)-N-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl){[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}amine
ethyl 3-benzyl-1-{[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]methyl}piperidine-3-carboxylate