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3-{[methyl({2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl})amino]methyl}phenol
3-methyl-8-[2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)acetyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)propanamide
1-[3-({7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}methyl)phenyl]ethan-1-one
[(3R,4R)-1-(2,3-dimethyl-1H-indole-5-carbonyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
1-cyclopropyl-N-methyl-6-oxo-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]piperidine-3-carboxamide
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidine
6-ethoxy-3-{[3-(pyrimidin-4-yl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
2-methyl-6-(thiophen-3-yl)-3,4-dihydroquinazolin-4-one
N-(3-methanesulfonamidophenyl)-4-(3-methylpyridin-4-yl)piperazine-1-carboxamide
5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]methyl}-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
2-(4-chlorophenoxy)-1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
1-[6-(2,5-dimethylphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]azepane
1-cyclohexyl-N-[2-(1,3-thiazol-4-yl)ethyl]piperidine-4-carboxamide
4-{1-[1-(1-methylcyclohexanecarbonyl)piperidin-4-yl]piperidine-4-carbonyl}morpholine
N-(2-methoxyethyl)-2-(3-methyl-1,2-oxazole-5-carbonyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
3-(pentan-2-yl)-8-[4-(1H-pyrazol-4-yl)butanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[1-(1-{[4-(propan-2-yl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]pyridine-3-carboxamide
N-(2-acetamidophenyl)-2-{[2-(ethylsulfanyl)ethyl]amino}acetamide
5-[2-(hydroxymethyl)phenyl]-N-[2-(propan-2-yl)phenyl]furan-2-carboxamide
4-{[(4-hydroxy-1-methylpiperidin-4-yl)methyl]amino}pyrimidine-5-carboxylic acid
1-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-methoxy-2-methylpropan-1-one
2-(4-{[1-ethyl-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]methyl}piperazin-1-yl)pyrimidine
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-N-(3-fluorophenyl)propanamide
N-cyclohexyl-N-(2-phenylethyl)-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
1-{5-[3-(5-fluoro-2-methoxybenzoyl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
2-methyl-4-(4-{[(1S,6R)-3-methyl-3,9-diazabicyclo[4.2.1]nonan-9-yl]methyl}phenyl)butan-2-ol
N'1-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]cyclopropane-1,1-dicarboxamide
[(5-{[2-(3-methoxyphenyl)pyrrolidin-1-yl]methyl}thiophen-3-yl)methyl]dimethylamine
(2S,4R)-4-(furan-3-amido)-1-(1H-imidazol-2-ylmethyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-[1-(pyridin-3-yl)propan-2-yl]-5-(trifluoromethyl)-3,4-dihydroquinazolin-4-one
9-(2-hydroxy-3-methylbenzoyl)-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-methyl-6-[4-(pyrazin-2-yl)piperazine-1-carbonyl]-1H-indole
[(3R,4R)-1-[(2,6-dimethoxyphenyl)methyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
8-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
1-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)pyrimidin-4-yl]piperidin-3-ol
(4aR,7aS)-1-(2-{[2-(dimethylamino)ethyl](methyl)amino}pyrimidin-4-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-methyl-5-{[(3S,4R)-4-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)oxolan-3-yl]methyl}-1,2-oxazole
(oxolan-2-ylmethyl)(propyl){[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amine
1-methyl-2-oxo-N-[2-(pyrrolidin-1-yl)ethyl]-1,2-dihydroquinoline-3-carboxamide
4-[6-(morpholine-4-carbonyl)pyrazin-2-yl]-1,4-oxazepan-6-ol
5-{4-[(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidine-1-carbonyl}pyridine-2-carbonitrile
8-[(4-chlorophenyl)methyl]-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[5-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepine-3-carbonyl)-1H-1,3-benzodiazol-1-yl]ethan-1-ol
2-cyclopentyl-1-{4-[3-({methyl[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)phenoxy]piperidin-1-yl}ethan-1-one
[(4-fluorophenyl)methyl]({[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})(oxolan-2-ylmethyl)amine
(3R,4R)-1-(2,6-diaminopyrimidin-4-yl)-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
4-(4-{[3-(morpholin-4-ylmethyl)piperidin-1-yl]methyl}phenyl)but-3-yn-1-ol
1-{3-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[(3R,4S)-4-(dimethylamino)-1-{[5-(1H-pyrazol-5-yl)furan-2-yl]sulfonyl}piperidin-3-yl]propanoic acid